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Quercetin dihydrate
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Quercetin dihydrate
CAS No. : 6151-25-3
MCE 站:Quercetin dihydrate
产品活性:Quercetin dihydrate 是一种天然黄酮类化合物,可激活或抑制许多蛋白质的活性。Quercetin (dihydrate) 可激活 SIRT1,也可抑制 PI3K,抑制 PI3K γ,PI3K δ,PI3K β 的 IC50 值分别为 2.4 μM, 3.0 μM, 5.4 μM。
研究领域:PI3K/Akt/mTOR | Apoptosis
In Vitro: Quercetin dihydrate is a type of plant-based chemical, or phytochemical, used as an ingredient in supplements, beverages or foods. In several studies, it may have anti-inflammatory and antioxidant properties, and it is being investigated for a wide range of potential health benefits.Quercetin dihydrate is a PI3K inhibitor with IC50s of 2.4-5.4 μM. Quercetin dihydrate strongly abrogates PI3K and Src kinases, mildly inhibits Akt1/2, and slightly affected PKC, p38 and ERK1/2.Quercetin dihydrate inhibits TNF-induced LDH% release, EC-dependent neutrophils adhesion to bovine pulmonary artery endothelial cells (BPAEC), and BPAEC DNA synthesis and proliferation.
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