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Nicergoline
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Nicergoline
CAS No. : 27848-84-6
MCE 站:Nicergoline
产品活性:Nicergoline,溴烟碱酸的麦角林衍生物,是一种有效,选择性和具有口服活性的
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Adrenergic Receptor
In Vitro: Nicergoline (0.3-30 μM; 24 h) attenuates activated microglia- and astrocytes-induced neuronal cell death.
Nicergoline (0.3-30 μM; 48 h) suppresses the production of proinflammatory cytokines and superoxide anion by activated microglia.
In Vivo: Nicergoline (10 mg/kg; i.v. once daily for 60 d) improves impaired neurogenesis and cognitive competence in mice with Alzheimer's disease.
Nicergoline (10 mg/kg; i.v. once daily for 60 d) inhibits apoptosis, inflammation and oxidative stress in hippocampal cells, and regulates the activity of hippocampal cells through the PI3K/AKT signaling pathway in mice.
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