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FTI-277 hydrochloride
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FTI-277 hydrochloride
CAS No. : 180977-34-8
MCE 站:FTI-277 hydrochloride
产品活性:FTI-277 hydrochloride 是法尼基转移酶 FTase 抑制剂,高效 Ras CAAX 肽模拟物,可抑制 H-Ras 和 K-Ras 信号转导。FTI-277 hydrochloride 可抑制 hepatitis delta virus (HDV) 感染。
研究领域:Metabolic Enzyme/Protease | Apoptosis | GPCR/G Protein
作用靶点:Farnesyl Transferase | Apoptosis | Ras
In Vitro: Treatment with FTI-277 (20 microM) for 48 h prior to irradiation led to a significant decrease in survival of radioresistant cells expressing the 24-kDa isoform (HeLa 3A) but had no effect on the survival of control cells (HeLa PINA). The radiosensitizing effect of FTI-277 is accompanied by a stimulation of postmitotic cell death in HeLa 3A cells and by a reduction in G(2)/M-phase arrest in both cell types [1]. Treatment of PC-3 cells with GGTI-298 and FTI-277 inhibited migration and invasion in a time- and dose-dependent manner [3].
In Vivo: FTI-277 treatment prevented increased PTP-1B and PTEN protein expression in burned mice as compared with vehicle alone. In contrast, FTI-277 did not significantly alter protein expression of PTP-1B and PTEN in sham-burned mice [2].
相关产品:Covalent Screening Library Plus | Bioactive Compound Library Plus | Anti-Infection Compound Library | Apoptosis Compound Library | GPCR/G Protein Compound Library | Kinase Inhibitor Library | Metabolism/Protease Compound Library | Anti-Cancer Compound Library | Peptidomimetic Library | Covalent Screening Library | Ferroptosis Compound Library | Glutamine Metabolism Compound Library | Anti-Pancreatic Cancer Compound Library | Anti-Blood Cancer Compound Library | MG-132 | LY294002 | Doxorubicin hydrochloride | Bafilomycin A1 | Paclitaxel | Y-27632 dihydrochloride | Acetylcysteine | Angiotensin II human | SP600125 | 5-Fluorouracil | Staurosporine | Bortezomib | Tamoxifen | 2-Deoxy-D-glucose | Gemcitabine | Verteporfin | Decitabine | Actinomycin D | Temozolomide | BAY 11-7082 | Etoposide | Mitomycin C | CCCP | DAPT | Rote | Etomoxir | Stattic | Docetaxel | Fulvestrant
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