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Src Inhibitor 1

CAS No. : 179248-59-0

MCE 站：Src Inhibitor 1

产品活性：Src Inhibitor 1是高效选择性的，ATP-竞争性的双位点Src酪氨酸激酶抑制剂，对Src和Lck的IC₅₀值分别为44 nM和88 nM。

研究领域：Protein Tyrosine Kinase/RTK

作用靶点：Src

In Vitro: Src-I1 is competitive with both ATP and peptide binding sites of the kinase. The IC₅₀ values are 44 and 88 nM for Src and Lck, respectively. Src-I1, is found to be a potent inhibitor of Src (IC₅₀=0.18 μM), but also inhibited other Src family members, such as Lck, Csk and Yes with similar potency to Src, and RIP2 (IC₅₀=0.026 μM) with even greater potency. In addition, it inhibited CHK2 with similar potency to Src, and Aurora B with slightly lower potency.

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