当前位置: 易推广 > 生物试剂/抗体/细胞 > 生化试剂 > 其他 > MedChemExpress > 产品展示 > MCE信号通路 > 凋亡 > Zoledronic acid disodium tetrahydrate
Zoledronic acid disodium tetrahydrate
企业档案
会员类型:会员
已获得易推广信誉 等级评定
(0 -40)基础信誉积累,可浏览访问
(41-90)良好信誉积累,可接洽商谈
(91+ )优质信誉积累,可持续信赖
易推广会员:8年
最后认证时间:
注册号: 【已认证】
法人代表: 【已认证】
企业类型:生产商 【已认证】
注册资金:人民币万 【已认证】
产品数:91195
参观次数:10506585
联系我们
MedChemExpress
电话:021-58955995
联系人:客服部 (请说明是在易推广看到的!谢谢)
手机:13611715263
邮编:201203
邮箱:sales@medchemexpress.cn
地址:上海上海
详细内容
MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
Zoledronic acid disodium tetrahydrate
CAS No. : 165800-07-7
MCE 站:Zoledronic acid disodium tetrahydrate
产品活性:Zoledronic Acid (Zoledronate) disodium tetrahydrate 是第三代含氮二磷酸盐,具有高效的抗骨质再吸收活性。Zoledronic Acid disodium tetrahydrate 能抑制破骨细胞的分化和凋亡。Zoledronic Acid disodium tetrahydrate 也有抗癌作用。
In Vitro: Zoledronic Acid disodium tetrahydrate (0.1-1 M; 48 hours) increases receptor activator of nuclear factor kB ligand (RANKL) and sclerostin mRNA expressions in osteocyte-like MLO-Y4 cells.
Zoledronic Acid disodium tetrahydrate increases the expression of osteoclastogenesis supporting factor from MLO-Y4 cells.
Zoledronic Acid disodium tetrahydrate enhances the RANKL expression via IL-6/ JAK2/STAT3 pathway in MLO-Y4 cells.
Zoledronic acid disodium tetrahydrate inhibits osteoclast differentiation and function through the regulation of NF-κB and JNK signalling pathways.
Zoledronic Acid disodium tetrahydrate (10-100 M; 1-7 days) markedly reduces the viability of MC3T3-E1 cells and induces apoptosis in MC3T3-E1 cells.
Zoledronic Acid disodium tetrahydrate (10-100 M; 4 days) inhibits cell viability due to the induction of apoptosis.
Zoledronic Acid disodium tetrahydrate exerts inhibitory effects on the differentiation and maturation of MC3T3-E1 cells at concentrations <1 M.
In Vivo: Zoledronic Acid disodium tetrahydrate (0.05 mg/kg; i.p.; weekly; for 3 weeks) increases bone mineral density and content.
Zoledronic Acid disodium tetrahydrate (0.5-1 mg/kg; i.p.; weekly; for 3 weeks) inhibits both osteoclast and osteoblasts function and bone remodeling in vivo interfering with bone mechanical properties.
相关产品:MG-132 | LY294002 | Doxorubicin hydrochloride | Bafilomycin A1 | Y-27632 dihydrochloride | Paclitaxel | Acetylcysteine | Tamoxifen | Deferoxamine mesylate | Angiotensin II human | Staurosporine | Bortezomib | 2-Deoxy-D-glucose | 5-Fluorouracil | Sorafenib | SP600125 | Trametinib | Temozolomide | Gemcitabine | MK-2206 dihydrochloride | Decitabine | Verteporfin | Etoposide | Gefitinib | Rote | DAPT | CCCP | Ruxolitinib | Actinomycin D
热门产品线:重组蛋白 | 化合物库 | 天然产物 | 染料试剂 | PROTAC | 同位素标记物 | 寡核苷酸
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Dye Reagents | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
品牌介绍:
• MCE (MedChemExpress) 拥有数百种全球独家化合物,我们致力于为全球科研客户提供*新*全的高品质小分子活性化合物;
• 10,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领域;
• 设有专业的实验中心和严格的质控、验证体系;
• 提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;
• 产品的生物活性多经各国客户实验验证;
• Nature, Cell, Science 等多种期刊及制药收录了MCE客户的科研成果;
• 专业团队跟踪*新的制药及生命科学研究进展,为您提供全球*新的活性化合物;
• 与世界各大制药公司及知名科研机构建立了长期的合作。