TP1559LZiconotide Acetate (107452-89-1 free base)analgesic,non-opioid,Ziconotide Acetate (107452891 free

Ziconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.

价 格：￥电议型 号：TP1559L产 地：中国大陆

T27371FR-167356

FR-167356 is a specific inhibitor of a3 isoform vacuolar type H?-ATPase with IC50s of 170 nM, 370 nM and 220 nM for osteoclast plasma membranes, renal brush border membranes and macrophage microsomes. FR-167356 reduces bone metastasis of B16-F10 cells.

价 格：￥电议型 号：T27371产 地：中国大陆

T58772,6-Dichloroaniline

2,6-Dichloroaniline is used as intermediate.

价 格：￥电议型 号：T5877产 地：中国大陆

T6675Sodium Picosulfateinhibit,Inhibitor,Sodium Picosulfate

Sodium Picosulfate inhibits absorption of water and electrolytes, and increases their secretion.

价 格：￥电议型 号：T6675产 地：中国大陆

TN12955-O-Caffeoylshikimic acidinhibit,5 O Caffeoylshikimic acid,Inhibitor,5OCaffeoylshikimic acid

5-O-Caffeoylshikimic acid shows anti-oxidative activity; it also shows anti-inflammatory activity, the underlying mechanism was associated with downregulation of nuclear factor-κB.

价 格：￥电议型 号：TN1295产 地：中国大陆

PDK04236-METHYL-1H-INDOLE-2-CARBOXYLIC ACID6METHYL1HINDOLE2CARBOXYLICACID

价 格：￥电议型 号：PDK0423产 地：中国大陆

T22849ICI 199,441 hydrochlorideICI 199,441 hydrochloride

ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.

价 格：￥电议型 号：T22849产 地：中国大陆

TP1789LMalantide acetate(86555-35-3 free base)Malantide acetate(86555 35 3 free base),Malantide acetate(865

Malantide acetate is a dodecapeptide phosphorylated by cyclic AMP-dependent protein kinase (PKA), and increases PKA activity.Malantide is a synthetic peptide that is phosphorylated by PKA and is used to measure PKA activity in vitro.

价 格：￥电议型 号：TP1789L产 地：中国大陆

T16536Pimonidazole hydrochlorideinhibit,Pimonidazole hydrochloride,Pimonidazole,Inhibitor

Pimonidazole hydrochloride accumulates in hypoxic cells via covalent binding with macromolecules or by forming reductive metabolites after the reduction of its nitro group. It can be used for qualitative and quantitative assessment of tumor hypoxia. Pimonidazole hydrochloride is a novel hypoxia marker for the complementary study of tumor hypoxia and cell proliferation in tumors.

价 格：￥电议型 号：T16536产 地：中国大陆

TN1438beta-Amyrin acetateHMG-CoA,betaAmyrin acetate,LDL,Fungal,inhibit,Inhibitor,arthritic,hemolysis,antif

beta-Amyrin acetate inhibits HMG-CoA Reductase (HMGCR) and sEH activity with IC50 of 3.4 μM. beta-Amyrin acetate has anti-inflammatory, antifungal, antioxidant, and anti-hyperlipidemic activities.

价 格：￥电议型 号：TN1438产 地：中国大陆

T22761EIT hydrobromide

EIT hydrobromide is an iNOS inhibitor.

价 格：￥电议型 号：T22761产 地：中国大陆

TP1898HS024selective,melanocortin,intake,Inhibitor,Melanocortin Receptor,MC Receptor,HS-024,food,HS024,inh

Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.

价 格：￥电议型 号：TP1898产 地：中国大陆

TN2079(-)-Pinoresinol()Pinoresinol,( ) Pinoresinol

(-)-Pinoresinol is isolated from the whole plant of Serissa japonica (Thunb.) Thunb.

价 格：￥电议型 号：TN2079产 地：中国大陆

T60146USP8-IN-1USP8inhibitor

USP8-IN-1 is an inhibitor of USP8 with an IC 50 of 1.9 μM. USP8-IN-1 inhibits H1975 cell growth with a GI 50 of 82.04 μM [1].

价 格：￥电议型 号：T60146产 地：中国大陆

TN2100PratenseinInhibitor,Nuclear factor-kappaB,Nuclear factor-κB,cognitive,inhibit,BDNF,synapse,Pratensei

Pratensein as a novel transcriptional up-regulator of scavenger receptor class B type I in HepG2 cells.

价 格：￥电议型 号：TN2100产 地：中国大陆

TP1882L1Orphanin FQ(1-11) acetate(178249-41-7 free base)Orphanin FQ(1 11) acetate(178249 41 7 free base),Orp

Peptide fragment containing amino acids 1-11 of Nociceptin. Potent agonist of the ORL1/KOR-3 receptor (Ki = 55 nM); displays no affinity for opioid receptors, including μ, δ, κ1 and κ3 receptors (Ki >1000 nM). Displays analgesic properties in CD-1 mice.

价 格：￥电议型 号：TP1882L1产 地：中国大陆

T8595Practololreceptor,inhibit,arrhythmias,β1-adrenergic,Practolol,Beta Receptor,Adrenergic Receptor,card

Practolol is a selective β-adrenoceptor blocker.

价 格：￥电议型 号：T8595产 地：中国大陆

T8796CAN508inhibit,CAN 508,ATP-competitive,Cyclin dependent kinase,esophageal,cells,CDK,CAN508,Inhibitor,

CAN508 is a potent, ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 μM. It is also a competitive inhibitor of Cdk2-cyclin E with respect to ATP, with Ki and IC50 values of 13.3 and 20 μM, respectively.CAN508 exhibits a 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes. Antitumor activity.

价 格：￥电议型 号：T8796产 地：中国大陆

T6924Riviciclib hydrochlorideinhibit,Inhibitor,Riviciclib,CDK,Riviciclib hydrochloride,Cyclin dependent k

P276-00 is a novel CDK1, CDK4 and CDK9 inhibitor with IC50 of 79 nM, 63 nM and 20 nM, respectively. Phase 2/3.

价 格：￥电议型 号：T6924产 地：中国大陆

T6767TCS7010Aurora Kinase,inhibit,TCS 7010,Apoptosis,TCS-7010,TCS7010,Inhibitor

Aurora A Inhibitor I is a novel, potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM in a cell-free assay. It is 1000-fold more selective for Aurora A than Aurora B.

价 格：￥电议型 号：T6767产 地：中国大陆