T31204Darapladib-impurityDarapladib impurity,Darapladibimpurity

Darapladib-impurity is the impurity of Darapladib. Darapladib inhibits lipoprotein-associated phospholipase A2 (Lp-PLA2)

价 格：￥电议型 号：T31204产 地：中国大陆

T67698WAY-300374WAY300374

WAY-300374 inhibits the p53-MDM2 protein-protein interaction.

价 格：￥电议型 号：T67698产 地：中国大陆

T7848PT-2385Inhibitor,inhibit,Hypoxia-inducible factors,HIF/HIF Prolyl-Hydroxylase,HIF-PH,PT 2385,HIFs,PT

PT-2385 is a selective HIF-2α inhibitor (Kd<50 nM).

价 格：￥电议型 号：T7848产 地：中国大陆

T15018CUDC-427

CUDC-427 is an orally bioactive and pan antagonist of inhibitor of apoptosis proteins(IAPs). CUDC-427 can be used in research on cancers.

价 格：￥电议型 号：T15018产 地：中国大陆

TP1559LZiconotide Acetate (107452-89-1 free base)analgesic,non-opioid,Ziconotide Acetate (107452891 free

Ziconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.

价 格：￥电议型 号：TP1559L产 地：中国大陆

T8439Clobenpropit dihydrobromideApoptosis,inhibit,Clobenpropit dihydrobromide,histamine H3R,antagonist,in

Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)

价 格：￥电议型 号：T8439产 地：中国大陆

T15641K777

K777 is a potent, orally active and irreversible inhibitor of cysteine protease. K777 is a potent CYP3A4 inhibitor (IC50= 60 nM). K777 is also a selective CCR4 antagonist featuring the potent chemotaxis inhibition. K777 irreversibly inhibits Cruzain, which is the major cysteine protease of Trypansoma cruzi, and cathepsins B and L. K777 targets cathepsin-mediated cell entry and wxibits a broad-spectrum antiviral activity. K777 inhibits EBOV and SARS-CoV pseudovirus entry with IC50 values of 0.87

价 格：￥电议型 号：T15641产 地：中国大陆

T8331NUN82647NUN82647,Inhibitor,NUN 82647,inhibit,Apoptosis,QBS,NUN-82647

NUN82647 is an Inhibitor of cell cycle at G2 phase, and apoptosis inducer.

价 格：￥电议型 号：T8331产 地：中国大陆

T9840AtaquimasAtaquimas

Ataquimast inhibits IL-5 secretion along with that of TNF-a, IL-4 and GM-CSF from human cells.

价 格：￥电议型 号：T9840产 地：中国大陆

T27371FR-167356

FR-167356 is a specific inhibitor of a3 isoform vacuolar type H?-ATPase with IC50s of 170 nM, 370 nM and 220 nM for osteoclast plasma membranes, renal brush border membranes and macrophage microsomes. FR-167356 reduces bone metastasis of B16-F10 cells.

价 格：￥电议型 号：T27371产 地：中国大陆

T58772,6-Dichloroaniline

2,6-Dichloroaniline is used as intermediate.

价 格：￥电议型 号：T5877产 地：中国大陆

T6675Sodium Picosulfateinhibit,Inhibitor,Sodium Picosulfate

Sodium Picosulfate inhibits absorption of water and electrolytes, and increases their secretion.

价 格：￥电议型 号：T6675产 地：中国大陆

T16940STAT5-IN-2STAT-5-IN-2,STAT5IN2,STAT5 IN 2

STAT5-IN-2 is an inhibitor of STAT5 with antileukemic effects (EC50s: 9 μM and 5 μM in K562 and KU812 cells, respectively).

价 格：￥电议型 号：T16940产 地：中国大陆

TN2275Tinnevellin glucosideTinnevellin glucoside,inhibit,Inhibitor

Tinnevellin glucoside is a natural product from Cassia angustifolia.

价 格：￥电议型 号：TN2275产 地：中国大陆

TN12955-O-Caffeoylshikimic acidinhibit,5 O Caffeoylshikimic acid,Inhibitor,5OCaffeoylshikimic acid

5-O-Caffeoylshikimic acid shows anti-oxidative activity; it also shows anti-inflammatory activity, the underlying mechanism was associated with downregulation of nuclear factor-κB.

价 格：￥电议型 号：TN1295产 地：中国大陆

PDK04236-METHYL-1H-INDOLE-2-CARBOXYLIC ACID6METHYL1HINDOLE2CARBOXYLICACID

价 格：￥电议型 号：PDK0423产 地：中国大陆

TP1881L1Pep 2-8 ammonium salt(1541011-97-5 free base)Pep 2 8 ammonium salt(1541011 97 5 free base),Pep 28 am

Pep 2-8 ammonium salt is Proprotein convertase subtilisin/kexin type 9 (PCSK9) inhibitor. Potent inhibitor of PCSK9 binding to LDL receptor (IC50 = 0.8 μM). Restores LDL uptake in HepG2 cells treated with PCSK9.

价 格：￥电议型 号：TP1881L1产 地：中国大陆

T22849ICI 199,441 hydrochlorideICI 199,441 hydrochloride

ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.

价 格：￥电议型 号：T22849产 地：中国大陆

TQ0150LevcromakalimPotassium Channel,KcsA,Inhibitor,inhibit,BRL38227,BRL-38227,Levcromakalim

Levcromakalim is an activator of the ATP-sensitive K+ channel.

价 格：￥电议型 号：TQ0150产 地：中国大陆

TN12373-O-Methylgallic acidAnthocyanin,3 O Methylgallic acid,inhibit,3OMethylgallic acid,metabolite,anti-c

3,4-Dihydroxy-5-methoxybenzoic acid reduces cell proliferation in Caco-2 cells(IC50 = 24.1 μM) more effectively than anthocyanins and may offer protection against colon cancer after its formation in the gut. 3,4-Dihydroxy-5-methoxybenzoic acid inhibits transcription factors NF-κB, AP-1, STAT-1, and OCT-1 which are known to be activated in colorectal cancer.

价 格：￥电议型 号：TN1237产 地：中国大陆