T11023DHODH-IN-14DHODH IN 14,DHODHIN14

DHODH-IN-14 is an analog of hydroxyfuran pyrimidine A771726. DHODH-IN-14 is a dihydroorotate dehydrogenase (DHODH) inhibitor IC50 0.49 μM mouse liver DHODH. DHODH-IN-14 can be used for rheumatoid arthritis.

价 格：￥电议型 号：T11023产 地：中国大陆

TQ0230BTK IN-1Btk,SNS062,Inhibitor,SNS-062,BTK IN 1,Bruton tyrosine kinase,SNS 062,inhibit,BTK IN-1,BTK IN

BTK IN-1 (SNS062 analog) is an effective BTK inhibitor (IC50: <100 nM).

价 格：￥电议型 号：TQ0230产 地：中国大陆

T40023Pomalidomide-PEG3-CO2H

Thalidomide-NH-PEG3-propionic acid is a synthesized E3 ligase ligand-linker conjugate. Thalidomide-NH-PEG3-propionic acid incorporates the Thalidomide based cereblon ligand and 3-unit PEG linker used in PROTAC technology.

价 格：￥电议型 号：T40023产 地：中国大陆

T6883SamotolisibInhibitor,mTOR,LY-3023414,Phosphoinositide 3-kinase,DNA-dependent protein kinase,inhibit,

LY3023414 is an oral ATP competitive inhibitor of the class I PI3K isoforms, DNA-PK, and mTOR. LY3023414 has been used in trials studying the treatment of Neoplasm, Solid Tumor, COLON CANCER, BREAST CANCER, and Advanced Cancer, among others.

价 格：￥电议型 号：T6883产 地：中国大陆

T8219VU0238441mAChR,Inhibitor,VU-0238441,VU0238441,Muscarinic acetylcholine receptor,VU 0238441,inhibit

VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.

价 格：￥电议型 号：T8219产 地：中国大陆

PDK0236Compound PDK0236Compound PDK0236

价 格：￥电议型 号：PDK0236产 地：中国大陆

T60023CL-278474CL278474,CL 278474

CL-278474 (compound I-79) is a potent inhibitor of β-N-acetylhexosaminidase OfHex1. CL-278474 can be used in control of insect.

价 格：￥电议型 号：T60023产 地：中国大陆

T6S2023HarpagosideCOX,inhibit,Cyclooxygenase,NO Synthase,Harpagoside,NOS,Nitric oxide synthases,Inhibitor

1. Harpagoside has anti-inflammatory activity. 2. Harpagoside at 3 mM concentration, shows moderate inhibition of seed germination. 3. Harpagoside can inhibit lipopolysaccharide-induced mRNA levels and protein expression of cyclooxygenase-2 and inducible nitric oxide in HepG2 cells.

价 格：￥电议型 号：T6S2023产 地：中国大陆

TQ0236Tirabrutinib

Tirabrutinib (ONO-4059) is an orally active Bruton’s Tyrosine Kinase (Btk) inhibitor (can cross the blood-brain barrier (BBB)), with an IC50 of 6.8 nM. Tirabrutinib irreversibly and covalently binds to Btk and inhibits aberrant B cell receptor signaling. Tirabrutinib can be used in studies of autoimmune diseases and hematological malignancies.

价 格：￥电议型 号：TQ0236产 地：中国大陆

TPL0023Compound 80875-98-5Compound 80875985,Compound 80875 98 5

价 格：￥电议型 号：TPL0023产 地：中国大陆

T6896TolimidoneSrc,Tolimidone,MLR 1023,MLR1023,Inhibitor,inhibit

MLR-1023 is a chemical compound which inhibits acid secretion in animal models and also acts as a bronchodilator in histamine-challenged animals.

价 格：￥电议型 号：T6896产 地：中国大陆

TQ0292GrapiprantRQ 00000007,Inhibitor,Grapiprant,CJ 023423,RQ00000007,Prostaglandin Receptor,AAT 007,inhib

Grapiprant is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM).

价 格：￥电议型 号：TQ0292产 地：中国大陆

T9023AtuliflaponInhibitor,inhibit,FLAP,AZD-5718,AZD 5718,artery,Atuliflapon,disease,Coronary,5-LO activat

AZD5718 is a novel 5-Lipoxygenase Activating Protein(FLAP) inhibitor for Treatment of Coronary Artery Disease.

价 格：￥电议型 号：T9023产 地：中国大陆

TQ0023LorediplonGABA Receptor,γ-Aminobutyric acid Receptor,inhibit,Inhibitor,Lorediplon,Gamma-aminobutyric

Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.

价 格：￥电议型 号：TQ0023产 地：中国大陆

TP1111LTirzepatide Acetate(2023788-19-2 free base)Tirzepatide Acetate(2023788 19 2 free base),Tirzepatide A

Tirzepatide acetate is a dual GIP / GLP-1 receptor agonist.

价 格：￥电议型 号：TP1111L产 地：中国大陆

T7522GI254023XSRI 028594,SRI028594,GI 4023,inhibit,GI-254023X,Matrix metalloproteinases,SRI-028594,Inhibi

GI254023X is a potent MMP9 and ADAM10 inhibitor (IC50s: 2.5 and 5.3 nM) with 100-fold selectivity for the α-secretase ADAM10 over ADAM17 (TACE). GI254023X can remarkably inhibit the proliferation and induce the apoptosis of H929 cells. Its mechanism may be associated with inbihition of Notch1 activation.

价 格：￥电议型 号：T7522产 地：中国大陆

T7419SutezolidU 100480,oxazolidinone,Antibiotic,protein,Sutezolid,synthesis,Bacterial,Inhibitor,PF 023412

Sutezolid is an oxazolidinone antimicrobial for the treatment of tuberculosis.

价 格：￥电议型 号：T7419产 地：中国大陆

T6S0232EriodictyolEriodictyol,Inhibitor,DNA/RNA Synthesis,inhibit,Keap1-Nrf2,Influenza Virus,Endogenous Met

1. Eriodictyol is a flavonoid with anti-inflammatory and antioxidant activities. 2. Eriodictyol may possess antidiabetic properties through increasing glucose uptake and improving insulin resistance. 3. Eriodictyol may be a potential therapeutic resource for Atopic dermatitis and an adjunctive agent to control itchiness inAtopic dermatitis.

价 格：￥电议型 号：T6S0232产 地：中国大陆

T9611PF-04802367PF367,PF 367,protein,disease,Alzheimer,PF-04802367,PF-367,Glycogen synthase kinase-3,kina

PF-04802367 is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3β enzyme assay and 1.1 nM based on ADP-Glo assay. It shows desirable central nervous system (CNS) properties and potency. It is equally effective at inhibition of the two known GSK-3 isoforms (GSK-3α and GSK-3β) with IC50 values of 10.0 and 9.0 nM in mobility shift assays, respectively.

价 格：￥电议型 号：T9611产 地：中国大陆

TQ0232UNC0646H3K9me2,KMT1D,chromatin,EHMT1,Histone Methyltransferase,UNC-0646,SAR,inhibit,G9a,GLP,PKMT,UNC

UNC 0646 is a potent and selective inhibitor of the homologous protein lysine methyltransferases, G9a and GLP (IC50s: 6 nM/15 nM for G9a/GLP). UNC0646 potently blocks G9a/GLP methyltransferase activity in cells (IC50: 10 nM in MCF7 cells); exhibits low cellular toxicity (EC50: 4.7 μM in MCF7 cells).

价 格：￥电议型 号：TQ0232产 地：中国大陆