Fr12535Compound Fr12535Compound Fr12535

价 格：￥电议型 号：Fr12535产 地：中国大陆

T27683JNJ-42253432JNJ42253432,JNJ 42253432

JNJ-42253432 is a potent and selective antagonist of central nervous system-penetrant P2X7.

价 格：￥电议型 号：T27683产 地：中国大陆

T12530PPTNPPTN

PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.

价 格：￥电议型 号：T12530产 地：中国大陆

T8933JNJ-63576253 free baseJNJ 63576253 free base,resistant,TRC 253,JNJ63576253,TRC-253,CRPC,JNJ63576253

JNJ-63576253 is a potent and orally active full antagonist of androgen receptor (AR), with IC50s of 37 and 54 nM for F877L mutant AR and wild-type AR in LNCaP cells. JNJ-63576253 can be used for the research of castration-resistant prostate cancer (CRPC).

价 格：￥电议型 号：T8933产 地：中国大陆

T7727Se-Methylselenocysteinecaspase-3,A253,neck,SKOV-33,FaDu,Apoptosis,chemopreventive,cancer,cells,Se-Me

Se-Methylselenocysteine is a potent chemopreventive agent in many test systems and has been shown to inhibit tumor promotion and induce apoptosis.

价 格：￥电议型 号：T7727产 地：中国大陆

T25253Cinnamtannin B-1

Cinnamtannin B1 is an A-type proanthocyanidin contained in several plant species such as Vaccinium vitis-idaea, Laurus nobilis L., Cinnamomum zeylanicum, and Lindera umbellata. It is a potent antioxidant and protective agent against oxidative stress and apoptosis in human platelets. It is a Cox-2 inhibitor.

价 格：￥电议型 号：T25253产 地：中国大陆

TP1253Argirelineskin-permeable,BoNTs,inhibit,neurotransmitter,Inhibitor,peptide,Acetyl hexapeptide 3,Argir

Argireline (Acetyl hexapeptide-3) is composed of chains of amino acids known as peptides. Argireline significantly inhibits Ca2+ dependent neurotransmitter release (acetylcholine) at the neuromuscular junction. Argireline has antiwrinkle and anti-aging activity[1][2][3].

价 格：￥电议型 号：TP1253产 地：中国大陆

T23005MM 11253

MM 11253 is a RARγ antagonist with IC50 of 44nM.

价 格：￥电议型 号：T23005产 地：中国大陆

T12531PQCAPQCA

PQCA is a highly selective muscarinic M1 receptor positive allosteric modulator(EC50 value of 49 nM and 135 nM on rhesus and human M1 receptor, respectively).

价 格：￥电议型 号：T12531产 地：中国大陆

T13253UmibecestatBACE,Beta-secretase,inhibit,CNP-520,β-Secretase,CNP 520,Inhibitor

Umibecestat is an inhibitor of beta-site amyloid precursor protein cleaving enzyme-1 (BACE-1), with IC50s of 11 nM and 10 nM for human BACE-1 and mouse BACE-1, respectively. Umibecestat can be used for the research of alzheimer´s disease.

价 格：￥电议型 号：T13253产 地：中国大陆

T25310Dersimelagon

Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m) and rat (r) MC1R, respectively. Dersimelagon shows good affinity for hMC1R and hMC4R with Ki values of 2.26, 32.9 nM, respectively. Dersimelagon can be used for the research of skin pigmentation.

价 格：￥电议型 号：T25310产 地：中国大陆

T22538A-7 hydrochlorideA7 hydrochloride,A 7 hydrochloride

A-7 hydrochloride is a calmodulin antagonist and causes alterations in the subpopulation of CD44+CD24- in MDA-MB-231 cells.

价 格：￥电议型 号：T22538产 地：中国大陆

T9246JNJ-63576253TRC-253,mutant,JNJ 63576253,resistant,wild-type,JNJ63576253,TRC 253,prostate,inhibit,And

JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).

价 格：￥电议型 号：T9246产 地：中国大陆

TQ0253PLX51107PLX 51107,Epigenetic Reader Domain,PLX51107,inhibit,PLX-51107,Inhibitor

PLX51107 is a potent and selective BET inhibitor (Kds: 1.6, 2.1, 1.7, and 5 nM for BRD2-BD1, BRD3-BD1, BRD4-BD1, and BRDT-BD1).

价 格：￥电议型 号：TQ0253产 地：中国大陆

T23253RS 100329

RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.

价 格：￥电议型 号：T23253产 地：中国大陆

T7680GSNKGAIIGLM(131602-53-4(free base))GSNKGAIIGLM(131602 53 4(free base)),GSNKGAIIGLM(131602534(free ba

GSNKGAIIGLM is the fragment Aβ(25-35) of the Alzheimer´s amyloid β-peptide.

价 格：￥电议型 号：T7680产 地：中国大陆

T9239RS-25344RS25344,RS 25344

RS-25344 is a potent and selective phosphodiesterase (PDE) 4 inhibitor. It inhibits eosinophil chemotaxis and increases progressive motility of spermatozoa in vitro.

价 格：￥电议型 号：T9239产 地：中国大陆

TN12533-hydroxymorindoneinhibit,3-Hydroxymorindone,anthraquinone,Inhibitor,dye,3 hydroxymorindone,3hydroxy

3-hydroxymorindone is a natural product from Morinda citrifolia. 3-hydroxymorindone is a pigment.

价 格：￥电议型 号：TN1253产 地：中国大陆

TP2135LcAC 253 acetate

cAC 253 acetate is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.

价 格：￥电议型 号：TP2135L产 地：中国大陆

TQ0266MSC2530818Cyclin dependent kinase,Inhibitor,CDK,MSC2530818,inhibit,MSC 2530818,MSC-2530818

MSC2530818 is an effective, selective and orally available CDK8 inhibitor (IC50: 2.6 nM).

价 格：￥电议型 号：TQ0266产 地：中国大陆