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T70063GYKI 52466 HCl；化合物 GYKI 52466 HClGYKI 52466 HCl
GYKI 52466 is an allosteric AMPA receptor antagonist. It selectively inhibits AMPA-induced inward currents (IC50 = 7.5 ?M) over NMDA- or GABA-induced inward currents in primary rat hippocampal neurons at 50 ?M but also inhibits kainate-induced inward currents in the same cells (IC50 = 11 ?M).2 GYKI 52466 (10 ?M) reduces the amplitude of spontaneous excitatory postsynaptic currents (EPSCs) in the same cells. It increases the latency to seizure onset and reduces mortality in a rat model of general
价 格：￥电议型 号：T70063产 地：中国大陆
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T21449GYKI-52466；化合物 T21449GYKI 52,466|||GYKI-5,2466|||GYKI52,466；GYKI 52,466|||GYKI-5,2466|||GYKI52,466
GYKI-52466 is a selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >50 μM for AMPA-, kainate- and NMDA-induced responses, respectively) used as a Skeletal muscle relaxant, orally active anticonvulsant, neuroprotective and anxiolytic in vivo.
价 格：￥电议型 号：T21449产 地：中国大陆
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T11522GYKI 52466 dihydrochloride；化合物 T11522GYKI 52466 dihydrochloride
GYKI 52466 dihydrochloride is orally active and non-competitive kainate- and AMPA-activated currents antagonist (IC50s: 7.5 μM and 11 μM). It is inactive against NMDA or γ-aminobutyric acid responses. It is a muscle relaxant and anticonvulsant agent and has good blood-brain barrier permeability.
价 格：￥电议型 号：T11522产 地：中国大陆
