T9192BIIB068ADME,inhibit,FcγR,Autoimmune,Bruton tyrosine kinase,TNFα,BIIB 068,ROS,Inhibitor,reversible,Bt

BIIB068 is an selective, reversible and orally active BTK inhibitor (IC50 = 1 nM, Kd = 0.3 nM). BIIB068 is 400 times more selective for BTK than other kinases.

价 格：￥电议型 号：T9192产 地：中国大陆

TN1768IriflophenoneInhibitor,MCF-7,proliferation,Iriflophenone,cells,T-47D,inhibit

Iriflophenone?stimulates cells proliferation in?MCF-7 and T-47D human breast cancer.

价 格：￥电议型 号：TN1768产 地：中国大陆

T9268UlinastatinUlinastatin

Ulinastatin is a multivalent Kunitz-type serine protease inhibitor with anti-inflammatory properties.

价 格：￥电议型 号：T9268产 地：中国大陆

T6874Lercanidipine hydrochlorideantihypertensive,Inhibitor,calcium,Lercanidipine,Lercanidipine hydrochlor

Lercanidipine is a calcium channel blocker of the dihydropyridine class.

价 格：￥电议型 号：T6874产 地：中国大陆

T6683STF-62247renal,STF-62247,VHL,carcinoma,inhibit,cytotoxic,cell,RCC,Inhibitor,STF62247,intracytoplasmi

STF-62247 is TGN inhibitor with IC50 of 0.625 μM and 16 μM in RCC4 and RCC4/VHL cells, respectively.

价 格：￥电议型 号：T6683产 地：中国大陆

T6990LSNAP8 Acetate(868844-74-0,free base)SNAP8 Acetate(868844 74 0,free base),SNAP8 Acetate(868844740,fre

Diminishing the appearance of wrinkles.

价 格：￥电议型 号：T6990L产 地：中国大陆

T6476Dofetilidecardiovascular,potent,specific,class,antiarrhythmic,orally,Inhibitor,UK68789,UK-68789,Dofe

Dofetilide is a sulfonamide class III antiarrhythmic agent and potassium channel blocker. Dofetilide selectively blocks cardiac ion channels of the rapid component of the delayed rectifier potassium current Ikr. This antiarrhythmic agent prolongs cardiac action potential duration and effective refractory period due to delayed repolarization without affecting conduction velocity. This results in a normal sinus rhythm. Dofetilide is used in the treatment of atrial fibrillation and flutter.

价 格：￥电议型 号：T6476产 地：中国大陆

T6S1683DemethoxycurcuminBacterial,Inhibitor,Autophagy,Demethoxycurcumin,inhibit,Apoptosis

1. Demethoxycurcumin has antioxidant activity. 2. Demethoxycurcumin has anti-inflammatory activity. 3. Demethoxycurcumin has anti-proliferative activity. 4. Demethoxycurcumin has anti-acanthamoebic effect. 5. Demethoxycurcumin is a potential additive natural product in combination with chemotherapeutic agents in drug-resistant cancers. 6. Demethoxycurcumin inhibits energy metabolic and oncogenic signaling pathways through AMPK activation in triple-negative breast cancer cells.

价 格：￥电议型 号：T6S1683产 地：中国大陆

TQ0011PF-06869206inhibit,PF-06869206,Na+ channels,Sodium Channel,Na channels,PF 06869206,Inhibitor,PF06869

PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).

价 格：￥电议型 号：TQ0011产 地：中国大陆

Fr16683Compound Fr16683Compound Fr16683

价 格：￥电议型 号：Fr16683产 地：中国大陆

T14681BMS-935177BMS 935177,BMS935177

BMS-935177 is a reversible BTK inhibitor with IC50 value of 3 nM.

价 格：￥电议型 号：T14681产 地：中国大陆

T6864IxabepiloneBMS247550,inhibit,Inhibitor,Aza-epothilone B,Apoptosis,Microtubule/Tubulin,Ixabepilone,BM

Ixabepilone is an orally bioavailable microtubule inhibitor. It binds to tubulin and promotes tubulin polymerization and microtubule stabilization, thereby arresting cells in the G2-M phase of the cell cycle and inducing tumor cell apoptosis.

价 格：￥电议型 号：T6864产 地：中国大陆

T9573GSK3685032Inhibitor,GSK 3685032,lymphoma,DNMTs,cancer,DNA MTases,GSK-3685032,inhibit,GSK3685032,DNA

GSK3685032 is a non-covalent and selective DNMT1 inhibitor(IC50 = 36 nM). The inhibitory effect is time-independent and reversible. GSK3685032 induces loss of DNA methylation and transcriptional activation and inhibits cancer cell growth.

价 格：￥电议型 号：T9573产 地：中国大陆

T6841FumagillinFumagillin,NSC 9168,Antibiotic,inhibit,Human immunodeficiency virus,Parasite,Inhibitor,NSC

Fumagillin is a selective and potent irreversible inhibitor of Methionine aminopeptidase 2 (MetAP2), used as an antibiotic to treat microsporidiosis.

价 格：￥电议型 号：T6841产 地：中国大陆

PDK0168Compound PDK0168Compound PDK0168

价 格：￥电议型 号：PDK0168产 地：中国大陆

T6635EMD638683inhibit,EMD-638683,EMD638683,Serum and glucocorticoid-regulated kinase,EMD 638683,Inhibitor

EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).

价 格：￥电议型 号：T6635产 地：中国大陆

TP1086Men 10376 TFA(135306-85-3,free)Men 10376 TFA(135306853,free),Men 10376 TFA(135306 85 3,free)

Men 10376 TFA is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.

价 格：￥电议型 号：TP1086产 地：中国大陆

T6885MarimastatTA-2516,Marimastat,inhibit,Inhibitor,BB 2516,BB-2516,TA 2516,Matrix metalloproteinases,MMP

Marimastat (BB-2516) is a potent, broad spectrum matrix metalloprotease (MMP) inhibitor. MMP-9 (IC50=3 nM), MMP-1 (IC50=5 nM), MMP-2 (IC50=6 nM), MMP-14 (IC50=9 nM)and MMP-7 (IC50=13 nM).

价 格：￥电议型 号：T6885产 地：中国大陆

TN7068Sinomenine N-oxideSinomenine N oxide,Sinomenine Noxide

Sinomenine N-oxide is one of the major metabolites of the cyclic metabolic mechanism of Sinomenine.

价 格：￥电议型 号：TN7068产 地：中国大陆

T6815HS-1371HS-1371,Inhibitor,Receptor-interacting protein kinases,RIPK,inhibit,HS 1371,RIP kinase,HS1371

HS-1371 is a novel kinase inhibitor of receptor-interacting protein kinase 3 (RIP3) with an IC50 of 20.8 nM.

价 格：￥电议型 号：T6815产 地：中国大陆