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产品数：86101
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T8418DCLK1-IN-1DCLK1 IN 1,signaling,PDAC,KRAS,cancer,low,ERK,Inhibitor,selective,DCLK1IN1,inhibit,DCLK-1-
DCLK1-IN-1 is a selective and in vivo-compatible chemical probe of the DCLK1 kinase domain .
价 格：￥电议型 号：T8418产 地：中国大陆
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T7703PK11007PK11007,inhibit,MDM-2/p53,Reactive Oxygen Species,Inhibitor,PK 11007,PK-11007
PK11007 is an anti-p53 drug.
价 格：￥电议型 号：T7703产 地：中国大陆
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T9177BPAM344Ionotropic glutamate receptors,GluK3a,PAM,iGluR,BPAM344,BPAM 344,Inhibitor,BPAM-344,KAR,GluK1
BPAM344 is a potent positive allosteric modulator (PAM) of the KAR subunits GluK1b, GluK2a, and GluK3a.
价 格：￥电议型 号：T9177产 地：中国大陆
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T9095Necrostatin-34Necrostatin 34,RIP kinase,FADD,Necrostatin-34,RIPK,inhibit,RIPK1,Receptor-interacting
Necrostatin-34 is a RIPK1 kinase inhibitor, stabilizing RIPK1 kinase in an inactive conformation by occupying a distinct binding pocket in the kinase domain.
价 格：￥电议型 号：T9095产 地：中国大陆
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T8900SeralutinibPK 10571,Seralutinib,inhibit,arterial,PDGFR,PK10571,PK-10571,PAH,Pulmonary,hypertension,G
Seralutinib is an inhibitor of inhaled PDGFRα and PDGFRβ. It is used in the study for pulmonary arterial hypertension.
价 格：￥电议型 号：T8900产 地：中国大陆
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T6848GSK1016790Ainhibit,Ca2+ channels,Inhibitor,embryonic,GSK-1016790A,Ca channels,HEK,vanilloid,transien
GSK1016790A (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.
价 格：￥电议型 号：T6848产 地：中国大陆
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T8861GSK199GSK 199,GSK-199,GSK199,Inhibitor,Peptidylarginine Deiminase,Protein Arginine Deiminase,inhibit
GSK199 is a selective PAD4 inhibitor(IC50 of 200 nM in the absence of calcium).
价 格：￥电议型 号：T8861产 地：中国大陆
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TN1493Chrysosplenol Dcancer,Apoptosis,inhibit,ERK1/2,Inhibitor,antitrypanosomal,breast,Chrysosplenol D,ant
Chrysosplenol D, an efflux pump inhibitor that can potentiate the activity of commercially important antibiotics and antimalarials.
价 格：￥电议型 号：TN1493产 地：中国大陆
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T10792LCHK1-IN-4 hydrochloride
CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1). CHK1-IN-4 hydrochloride potently inhibits chk1 phosphorylation in the tumor cells. CHK1-IN-4 hydrochloride has anti-tumor activity.
价 格：￥电议型 号：T10792L产 地：中国大陆
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T6422Brimonidine TartrateUK-14304,UK14304,AGN190342,Brimonidine,Adrenergic Receptor,AGN-190342,AGN 190342
Brimonidine tartrate is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated with open-angle glaucoma or ocular hypertension.
价 格：￥电议型 号：T6422产 地：中国大陆
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T9849HQ461cyclin K degrader,Cyclin dependent kinase,molecular glue,HQ461,HQ 461,HQ-461,CDK12 substrate ph
HQ461 is a molecular glue that promotes CDK12-DDB1 interaction to trigger cyclin K degradation, resulting in decreased CDK12 substrate phosphorylation, downregulation of DNA damage response genes, and cell death.
价 格：￥电议型 号：T9849产 地：中国大陆
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T64373CDK1-IN-2
CDK1-IN-2 is a CDK1 inhibitor with IC50 of 5.8 μM. A broad-spectrum kinase profiling of CDK1-IN-2 revealed nonselective inhibition of several kinases.
价 格：￥电议型 号：T64373产 地：中国大陆
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T3079GSK1838705ACD246,Anaplastic lymphoma kinase,inhibit,Cluster of differentiation 246,Anaplastic lympho
GSK1838705A is an effective IGF-1R inhibitor (IC50: 2.0 nM), modestly potent to IR (IC50: 1.6 nM) and ALK (IC50: 0.5 nM), respectively, and little inhibition to other protein kinases.
价 格：￥电议型 号：T3079产 地：中国大陆
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T39752CDK12-IN-2
CDK12-IN-2 is an effective and selective inhibitor of CDK12 with an IC50 of 52 nM, >100 μM, >10 μM and 16 μM for CDK12, CDK2, CDK7, and CDK9. CDK12-IN-2 can be used in studies about the function of CDK12.
价 格：￥电议型 号：T39752产 地：中国大陆
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T9688CC-90001CC90001,kinase,IPF,JNK,c-Jun,idiopathic,JNK1,Inhibitor,N-terminal,inhibit,CC-90001,CC 90001,
CC-90001 is an orally administered c-Jun N-terminal kinase (JNK) inhibitor with bias for JNK1 over JNK2.
价 格：￥电议型 号：T9688产 地：中国大陆
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TQ0138K145 hydrochlorideK-145,K 145,ERK,K145 hydrochloride,K145,Sphingosine kinase,anti-proliferative,SphK
K145 hydrochloride is a selective sphk2 inhibitor with substrate competitiveness and oral activity, with IC50 of 4.3 ?M and Ki of 6.4 ?M. K145 hydrochloride can induce apoptosis and has strong antitumor activity.
价 格：￥电议型 号：TQ0138产 地：中国大陆
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T9758dCeMM3?degradation,dCeMM 3,dCeMM3?,Inhibitor,inhibit,CDK,CDK12,Cyclin dependent kinase,glue degrader
dCeMM3 is a glue degrader. dCeMM3 prompts an interaction of CDK12-cyclin K with a CRL4B ligase complex, result in inducing ubiquitination and degradation of cyclin K.
价 格：￥电议型 号：T9758产 地：中国大陆
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T6636RefametinibMEK1,allosteric,RDEA 119,BAY-869766,inhibit,Inhibitor,MAP2K,MEK2,orally,MAPKK,RDEA-119,Mi
Refametinib (RDEA119, Bay 86-9766) is an effective, ATP non-competitive and specific inhibitor of MEK1/2 (IC50: 19/47 nM).
价 格：￥电议型 号：T6636产 地：中国大陆
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T8850sbp-7455SBP-7455,ULK,TNBC,ULK2,ULK1,Unc-51 like kinase,sbp7455,Ser318,sbp 7455,Inhibitor,inhibit,Aut
SBP-7455 potently inhibited ULK1/2 enzymatic activity in vitro and in cells, reduced the viability of TNBC cells and had oral bioavailability in mice.
价 格：￥电议型 号：T8850产 地：中国大陆
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T9195SHR0302Th17,SHR-0302,B-cell,Inhibitor,inhibit,arthritis,collagen,migration,hepatic,SHR0302,JAK1,phos
SHR0302 is a JAK inhibitor that binds JAK1 with stronger affinity than others (Selectivity for JAK1 is more than 10 times for JAK2, 77 times for JAK3, 420 times for Tyk2).
价 格：￥电议型 号：T9195产 地：中国大陆
