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T6S0232EriodictyolEriodictyol,Inhibitor,DNA/RNA Synthesis,inhibit,Keap1-Nrf2,Influenza Virus,Endogenous Met
1. Eriodictyol is a flavonoid with anti-inflammatory and antioxidant activities. 2. Eriodictyol may possess antidiabetic properties through increasing glucose uptake and improving insulin resistance. 3. Eriodictyol may be a potential therapeutic resource for Atopic dermatitis and an adjunctive agent to control itchiness inAtopic dermatitis.
价 格：￥电议型 号：T6S0232产 地：中国大陆
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TQ0207SulforaphaneInhibitor,Keap1-Nrf2,Apoptosis,Sulforaphane,Histone deacetylases,inhibit,HDAC
Sulforaphane is derived from the consumption of cruciferous vegetables, such as broccoli. It has shown anticancer and cardioprotective activities.
价 格：￥电议型 号：TQ0207产 地：中国大陆
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TN1674Garcinone DKeap1-Nrf2,inhibit,Reactive Oxygen Species,Garcinone D,Inhibitor,STAT
Garcinone D shows significant cytotoxicity against the CEM-SS cell line, with IC(50) value of 3.2 microg/ml; it exhibits dose-dependent enzyme-based microsomal aromatase inhibitory activity. Garcinone D inhibits p65 activation with IC50 values of 3.2 microM.
价 格：￥电议型 号：TN1674产 地：中国大陆
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T8979AEM1AEM-1,AEM1,inhibit,AEM 1,Inhibitor,Keap1-Nrf2
AEM1 is an inhibitor of deregulated NRF2 transcriptional activity in cancer. AEM1 acts by broadly decreasing the expression of NRF2 controlled genes, sensitizing A549 cells to various chemotherapeutic agents, and inhibiting the growth of A549 cells in vitro and in vivo.
价 格：￥电议型 号：T8979产 地：中国大陆
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TQ0211BrusatolNrf2,oxygen,CT-26,NSC172924,NSC-172924,defense,stress,Keap1-Nrf2,Brusatol,chemosensitization
Brusatol is a natural product isolated from the Brucea javanica plant. It inhibits Nrf2.
价 格：￥电议型 号：TQ0211产 地：中国大陆
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T6S2356Corynolineinhibit,Corynoline,Inhibitor,Cholinesterase (ChE),Keap1-Nrf2
1. Corynoline is an acetylcholinesterase inhibitor.
价 格：￥电议型 号：T6S2356产 地：中国大陆
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TQ0120CDDO-Iminhibit,Ferroptosis,Keap1-Nrf2,CDDO Im,Inhibitor,CDDO-Im,Peroxisome proliferator-activated re
CDDO-Im is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).
价 格：￥电议型 号：TQ0120产 地：中国大陆
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T6S1302CarnosolRibosomal S6 Kinase (RSK),Keap1-Nrf2,Endogenous Metabolite,S6K,inhibit,Carnosol,Inhibitor
Carnosol has anti-oxidative, anti-inflammatory, antiproliferative and apoptosis inducing properties. Carnosol enhances the sensitivity of chemoresistant cancer cells to chemotherapeutic agents. 3. Carnosol may as a novel agonist of TRPA1 with an EC5 value of 12.46 μM.
价 格：￥电议型 号：T6S1302产 地：中国大陆
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T81984Keap1-Nrf2-IN-10；化合物 Keap1-Nrf2-IN-10Keap1-Nrf2-IN-10
Keap1-Nrf2-IN-10 (compound 15) is a potent inducer of NQO1 and efficaciously mitigates oxidative stress in gamma-irradiated mice by reducing MDA and ROS levels, as well as NQO1 in the liver, which enhances the survival rate of these mice [1].
价 格：￥电议型 号：T81984产 地：中国大陆
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T80522Keap1-Nrf2 probe；化合物 Keap1-Nrf2 probeKeap1-Nrf2 probe
Keap1-Nrf2 probe [1] is a fluorescent molecule designed to target the interaction between the Kelch-like ECH-associated protein 1 (Keap1) and nuclear factor erythroid 2-related factor 2 (Nrf2).
价 格：￥电议型 号：T80522产 地：中国大陆
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T80260Keap1-Nrf2-IN-16；化合物 Keap1-Nrf2-IN-16Keap1-Nrf2-IN-16
Keap1-Nrf2-IN-16 is a biologically active peptide with KEAP1 binding activity.
价 格：￥电议型 号：T80260产 地：中国大陆
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T78697Keap1-Nrf2-IN-15；化合物 Keap1-Nrf2-IN-15Keap1-Nrf2-IN-15
Keap1-Nrf2-IN-15 (Compound 24a) is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction, displaying IC50 values of 77 nM in a fluorescence polarization (FP) assay and 2.5 nM in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay [1].
价 格：￥电议型 号：T78697产 地：中国大陆
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T74600Keap1-Nrf2-IN-9；化合物 Keap1-Nrf2-IN-9Keap1-Nrf2-IN-9
Keap1-Nrf2-IN-9 (compound 11) is a potent inhibitor of the Keap1-Nrf2 protein?protein interaction (PPI) with an IC50 value of 0.575 ?M. It enhances the expression of Nrf2 target genes, including heme oxygenase 1 (Hmox1), glutathione S-transferase P (GstP), and glutamate-cysteine ligase catalytic (Gclc) and modulatory (Gclm) subunits. Notably, Keap1-Nrf2-IN-9 is not cytotoxic to ARPE19 cells [1].
价 格：￥电议型 号：T74600产 地：中国大陆
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T72760Keap1-Nrf2-IN-6；化合物 Keap1-Nrf2-IN-6Keap1-Nrf2-IN-6
Keap1-Nrf2-IN-6 is a potent, selective inhibitor of the Keap1-Nrf2 protein?protein interaction (PPI), demonstrating an inhibitory concentration (IC50) of 41 nM and a dissociation constant (Kd) of 68 nM.
价 格：￥电议型 号：T72760产 地：中国大陆
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T72706Keap1-Nrf2-IN-13；化合物 Keap1-Nrf2-IN-13Keap1-Nrf2-IN-13
Keap1-Nrf2-IN-13 is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction (PPI), exhibiting an IC50 value of 0.15 μM, indicative of its high efficacy. It binds strongly to the Keap1 protein by forming hydrogen bonds with critical polar residues (Asn414, Arg415, Arg483, Gln530), showcasing its specificity. This compound has implications for research into diseases associated with oxidative stress and inflammation, such as pulmonary fibrosis, chronic obstructive pulmonary disorder (COPD)
价 格：￥电议型 号：T72706产 地：中国大陆
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T72687Keap1-Nrf2-IN-11；化合物 Keap1-Nrf2-IN-11Keap1-Nrf2-IN-11
Keap1-Nrf2-IN-11 (Compound 6k), a potent Keap1-Nrf2 inhibitor, exhibits a dissociation constant (KD) of 0.21 nM. It hampers the production of reactive oxygen species (ROS) and nitric oxide (NO), as well as the expression of tumor necrosis factor-alpha (TNF-α). By promoting Nrf2 nuclear translocation, it mitigates inflammation and is utilized in anti-inflammatory studies [1].
价 格：￥电议型 号：T72687产 地：中国大陆
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T64218Keap1-Nrf2-IN-1 TFA；化合物 Keap1-Nrf2-IN-1 TFAKeap1-Nrf2-IN-1 TFA
Keap1-Nrf2-IN-1 TFA (compound35) is a Keap1-Nrf2 protein-protein interaction inhibitor (IC50: 43 nM) that activates Nrf2-regulated cytoprotective responses. Keap1-Nrf2-IN-1 TFA antagonizes acetaminophen-induced liver injury in cellular and in vivo models.
价 格：￥电议型 号：T64218产 地：中国大陆
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T64190Keap1-Nrf2-IN-12；化合物 Keap1-Nrf2-IN-12Keap1-Nrf2-IN-12
eap1-Nrf2-IN-12 is a potent inhibitor of Keap1-Nrf2 (IC50: 2.30 μM). eap1-Nrf2-IN-12 is metabolically stable in human liver microsomes.
价 格：￥电议型 号：T64190产 地：中国大陆
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T63987Keap1-Nrf2-IN-14；化合物 Keap1-Nrf2-IN-14Keap1-Nrf2-IN-14
Keap1-Nrf2-IN-14 is a KEAP1-NRF2 inhibitor that effectively disrupts the KEAP1-NRF2 interaction (IC50: 75 nM) with a Kd=24 nM for KEAP1. Keap1-Nrf2-IN-14 induces the expression of NRF2 target genes and is able to enhance downstream antioxidant and anti-inflammatory effects. -Nrf2-IN-14 can be used to study oxidative stress-related inflammation.
价 格：￥电议型 号：T63987产 地：中国大陆
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T63294Keap1-Nrf2-IN-5；化合物 Keap1-Nrf2-IN-5Keap1-Nrf2-IN-5
Keap1-Nrf2-IN-5 is a potent inhibitor of Keap1-Nrf2 PPI (Keap1-Nrf2 protein-protein interaction) (IC50: 4.1 μM, Kd: 3.7 μM).
价 格：￥电议型 号：T63294产 地：中国大陆
