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T4170PKM2-IN-1PKM2 inhibitor；compound 3k
PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.
价 格：￥电议型 号：T4170产 地：中国大陆
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T81446PKM2 activator 6；化合物 PKM2 activator 6PKM2 activator 6
Compound Z10 (PKM2 activator 6) serves as both a PKM2 activator and a PDK1 inhibitor, exhibiting dissociation constants (K D ) of 121 μM and 19.6 μM, respectively. It promotes apoptosis in colorectal cells while suppressing their proliferation and migration, additionally inhibiting glycolysis. Compound Z10 demonstrates inhibitory effects on the proliferation of various cell lines, including DLD-1, HCT-8, HT-29, and MCF-10A, with half-maximal inhibitory concentrations (IC 50 ) of 10.04 μM, 2.16 μ
价 格：￥电议型 号：T81446产 地：中国大陆
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T79636PKM2-IN-4；化合物 PKM2-IN-4PKM2-IN-4
Compound 5C, referred to as Pkm2-in-4, is a selective PKM2 inhibitor (IC50 = 0.35 ?M) that modulates pyruvate-dependent respiration and promotes mitochondrial H2O2 production rate and electron transport system coupling [1].
价 格：￥电议型 号：T79636产 地：中国大陆
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T74814PKM2/PDK1-IN-1；化合物 PKM2/PDK1-IN-1PKM2/PDK1-IN-1
PKM2/PDK1-IN-1, a shikonin thioether derivative, serves as a dual inhibitor for PKM2/PDK1. This compound effectively inhibits the proliferation and induces apoptosis in NSCLC cells. It promotes intercellular ROS production and modulates apoptotic proteins, engaging in both mitochondrial and death receptor pathways [1].
价 格：￥电议型 号：T74814产 地：中国大陆
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T72693PKM2 activator 5；PKM2 激活剂5PKM2 activator 5
PKM2 activator 5 is a novel and potent PKM2 activator (AC50: 0.316 ?M) with potential anticancer activity for the study of cancer metabolism-related diseases.
价 格：￥电议型 号：T72693产 地：中国大陆
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T72692PKM2 activator 4；化合物 PKM2 activator 4PKM2 activator 4
PKM2 Activator 4, a chemical compound, functions as an activator of PKM2 with an activation concentration (AC 50) ranging from 1 to 10 μM. It is primarily utilized in cancer research.
价 格：￥电议型 号：T72692产 地：中国大陆
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T67900PKM2 inhibitor G；化合物 PKM2 inhibitor GPKM2 inhibitor G
PKM2 inhibitor G is a inhibitor of pyruvate kinase.
价 格：￥电议型 号：T67900产 地：中国大陆
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T62758PKM2 activator 2；PKM2激活剂2PKM2 activator 2
PKM2 activator 2 is a pyruvate kinase M2 (PKM2) activator with an AC 50 value of 66 nM.PKM2 activator 2 has anti-tumor proliferative properties and attenuates the Warburg effect by normalizing cellular glycolytic metabolism through activation of PKM2.
价 格：￥电议型 号：T62758产 地：中国大陆
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T61504PKM2 activator 3；化合物 PKM2 activator 3PKM2 activator 3
PKM2 activator 3 is a highly potent compound that activates PKM2, with an AC 50 value of 90 nM. It exhibits excellent Caco-2 permeability, a low efflux ratio, and remarkable microsomal stability. PKM2 activator 3 is particularly valuable for anticancer research purposes [1]. (AC 50: the concentration at which 50% enzyme activation occurs.)
价 格：￥电议型 号：T61504产 地：中国大陆
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T4170PKM2-IN-1；化合物PKM2 inhibitorPKM2 inhibitor|||compound 3k；PKM2 inhibitor|||compound 3k
PKM2-IN-1 (compound 3k) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.
价 格：￥电议型 号：T4170产 地：中国大陆
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T39984PKM2-IN-3PKM2-IN-3PKM2-IN-3
PKM2-IN-3 is a potent PKM2 kinase inhibitor, displaying an IC 50 value of 4.1 μM. The compound effectively suppresses PKM2-mediated glycolysis and NLRP3 activation, thereby exerting an anti-neuroinflammatory effect.
价 格：￥电议型 号：T39984产 地：中国大陆
