T7400RRX-001Parasite,RRx-001,RRX 001,Apoptosis,Inhibitor,inhibit,RRX001

RRx-001 is a potent inhibitor ofglucose 6-phosphate dehydrogenase(G6PD) and with potent antimalarial activity

价 格：￥电议型 号：T7400产 地：中国大陆

T8595Practololreceptor,inhibit,arrhythmias,β1-adrenergic,Practolol,Beta Receptor,Adrenergic Receptor,card

Practolol is a selective β-adrenoceptor blocker.

价 格：￥电议型 号：T8595产 地：中国大陆

TN71724,5-Dibromo-1H-Pyrrole-2-Carboxylic Acid

4,5-Dibromo-1H-Pyrrole-2-Carboxylic Acid is a marine derived natural products found in Agelas oroides.

价 格：￥电议型 号：TN7172产 地：中国大陆

T6476Dofetilidecardiovascular,potent,specific,class,antiarrhythmic,orally,Inhibitor,UK68789,UK-68789,Dofe

Dofetilide is a sulfonamide class III antiarrhythmic agent and potassium channel blocker. Dofetilide selectively blocks cardiac ion channels of the rapid component of the delayed rectifier potassium current Ikr. This antiarrhythmic agent prolongs cardiac action potential duration and effective refractory period due to delayed repolarization without affecting conduction velocity. This results in a normal sinus rhythm. Dofetilide is used in the treatment of atrial fibrillation and flutter.

价 格：￥电议型 号：T6476产 地：中国大陆

T9581ARRY-797ARRY 797,ARRY797

ARRY-797 is a potent and selective p38α inhibitor and inhibits LPS-Induced IL-6.

价 格：￥电议型 号：T9581产 地：中国大陆

T59362,3-DIHYDRO-1H-PYRROLO[2,3-B]PYRIDINE2,3 DIHYDRO 1H PYRROLO[2,3 B]PYRIDINE,2,3DIHYDRO1HPYRROLO[2,3B]

价 格：￥电议型 号：T5936产 地：中国大陆

T95712,4,5-Trichloro-7H-pyrrolo[2,3-d]pyrimid2,4,5Trichloro7Hpyrrolo[2,3d]pyrimid,2,4,5 Trichloro 7H pyrr

2,4,5-Trichloro-7H-pyrrolo[2,3-d]pyrimid is a chemical agent.

价 格：￥电议型 号：T9571产 地：中国大陆

T8948Ferrohemeinhibit,Inhibitor,Ferroheme

protoheme used as nutrient fortifier, blood tonic and food additive for iron

价 格：￥电议型 号：T8948产 地：中国大陆

T2518ARRY-380 (analog )Inhibitor,HER1,EGFR,ARRY380 (analog ),Epidermal growth factor receptor,ARRY 380 (a

ARRY-380 is a potent and selective HER2 inhibitor.

价 格：￥电议型 号：T2518产 地：中国大陆

T6438Cefoselis SulfateCefoselis,cephalosporin,Gram-negative,Gram-positive,Bacterial,barrier,FK037,Inhibit

Cefoselis is a widely used beta-lactam antibiotic.

价 格：￥电议型 号：T6438产 地：中国大陆

TWP2911ThymidineThymidine,precursor,synchronizing,inhibit,NSC21548,DNA,NSC-21548,Inhibitor,replication,arre

1. Thymidine overload due to Thymidine phosphorylase deficiency, and mitochondrial toxicity caused by antiviral Thymidine analogues.

价 格：￥电议型 号：TWP2911产 地：中国大陆

T8873BractoppinDNA break,Bractoppin,phosphopeptide,inhibit,DNA/RNA Synthesis,DNA damage,RAD51,G2 arrest,I

Bractoppin is a drug-like inhibitor of phosphopeptide recognition by the human BRCA1 tandem (t)BRCT domain (IC50 = 0.074 μM), which selectively inhibits substrate binding with nanomolar potency in vitro. Structure-activity exploration suggests that Bractoppin engages BRCA1 tBRCT residues recognizing pSer in the consensus motif, pSer-Pro-Thr-Phe, plus an abutting hydrophobic pocket that is distinct in structurally related BRCT domains, conferring selectivity.

价 格：￥电议型 号：T8873产 地：中国大陆

T67758Pumecitinib3Azetidineacetonitrile,3[3amino4(7Hpyrrolo[2,3d]pyrimidin4yl)1Hpyrazol1yl]1[(1methylethyl

Pumecitinib is a Janus kinase (JAK) inhibitor. Pumecitinib exhibits anti-inflammatory activity.

价 格：￥电议型 号：T67758产 地：中国大陆

T12770RR-11a analog

RR-11a analog is an inhibitor of asparaginyl endopeptidase with IC50s of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively.

价 格：￥电议型 号：T12770产 地：中国大陆

TN6848Piperonylic acidformation,virus,natural,inactivator,Cytochrome P450,Piperonylic acid,quasi-irreversi

Piperonylic acid is a natural molecule bearing a methylenedioxy function that closely mimics the structure of trans-cinnamic acid. Piperonylic acid selectively inactivate the CYP73A P450 subpopulation.

价 格：￥电议型 号：TN6848产 地：中国大陆

T7697BIX-01294PRMT1,recurrent,Autophagy,H3K9me3,Inhibitor,Cdkn1a,inhibit,p53,Gadd45a,MLKL,Histone Methylt

BIX-01294 is an G9a Histone Methyltransferase inhibitor(IC50 : 1.9 μM).

价 格：￥电议型 号：T7697产 地：中国大陆

T8375ML-210residue,Ferroptosis,inhibit,peroxidase,ML-210,Covalent,selenocysteine,Glutathione Peroxidase,M

ML-210 is a selective RAS and covalent glutathione peroxidase 4 (GPX4) inhibitor(GPX4, EC50 : 30 nM), with anti-cancer activity

价 格：￥电议型 号：T8375产 地：中国大陆

TN2289Licorice-saponin H2(18β,20α)-Glycyrrhizic acid,inhibit,Inhibitor,triterpene,Licorice-saponin H2,Lico

Licoricesaponin H2 is a natural product

价 格：￥电议型 号：TN2289产 地：中国大陆

T7827Glycyrrhizinic acid, potassium saltGlycyrrhizinic acid, potassium salt

Glycyrrhizinic acid, potassium salt can reduce ventricular arrhythmias caused by veratrol

价 格：￥电议型 号：T7827产 地：中国大陆

T11230ERRα antagonist-1

ERRα antagonist-1 is a selective and high affinity estrogen-related receptor α (ERRα) antagonist. ERRα antagonist-1 inhibits interaction of ERRα with Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, the IC50 values are 170 nM and 180 nM, respectively. ERRα antagonist-1 does not inhibit the interaction of either ERRβ or ERRγ with PGC-1α and PGC-1β coactivator, and also does not inhibit interaction of ERα or ERβ with PGC-1α or SRC-1.

价 格：￥电议型 号：T11230产 地：中国大陆