T8439Clobenpropit dihydrobromideApoptosis,inhibit,Clobenpropit dihydrobromide,histamine H3R,antagonist,in

Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)

价 格：￥电议型 号：T8439产 地：中国大陆

T38163ML-148ML-148,ML 148,selective,Inhibitor,prostaglandin-signaling,15-PGDH,15-Hydroxyprostaglandin dehy

ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM). ML-148 can be used to profile across a panel of related dehydrogenase or reductase enzymes and in studies about prostaglandin-signaling pathways.

价 格：￥电议型 号：T38163产 地：中国大陆

T10889CRTh2 antagonist 2CRTh2 antagonist 2,CRTh-2 antagonist 2

CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia.

价 格：￥电议型 号：T10889产 地：中国大陆

T9975GPR183GPR183 antagonist-1,SAE-14,inhibit,SAE 14,SAE14,HL-60,GPR183,Inhibitor,GPR183 antagonist SAE-1

GPR183 is a chemotactic receptor known for its role in the maturation of B cells, and the endogenous ligand is the oxysterol 7α,25-dihydroxycholesterol (7α,25-OHC). GPR183 can be used in research on inflammatory bowel disease (IBD).

价 格：￥电议型 号：T9975产 地：中国大陆

T10269AHR antagonist 2AHR antagonist 2

AHR antagonist 2 is an antagonist of the aryl hydrocarbon receptor. The IC50s for human AHR and mouse AHR are 0.885 and 2.03 nM, respectively.

价 格：￥电议型 号：T10269产 地：中国大陆

T63812MrgprX2 antagonist-8

MrgprX2 antagonist-8 is an MrgprX2 antagonist that can be used to study inflammatory diseases.

价 格：￥电议型 号：T63812产 地：中国大陆

T5903Sitagliptin Intermediate 2Sitagliptin Intermediate 2

价 格：￥电议型 号：T5903产 地：中国大陆

T101625-HT3 antagonist 35 HT3 antagonist 3,5-HT-3 antagonist 3,5HT3 antagonist 3

5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).

价 格：￥电议型 号：T10162产 地：中国大陆

T11230ERRα antagonist-1

ERRα antagonist-1 is a selective and high affinity estrogen-related receptor α (ERRα) antagonist. ERRα antagonist-1 inhibits interaction of ERRα with Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, the IC50 values are 170 nM and 180 nM, respectively. ERRα antagonist-1 does not inhibit the interaction of either ERRβ or ERRγ with PGC-1α and PGC-1β coactivator, and also does not inhibit interaction of ERα or ERβ with PGC-1α or SRC-1.

价 格：￥电议型 号：T11230产 地：中国大陆

T8649TMBIM6 antagonist-1TMBIM-6 antagonist-1,TMBIM6 antagonist 1,HT1080,SKBR3,TMBIM6 antagonist1,MCF7,Mam

BIA is a bax inhibitor

价 格：￥电议型 号：T8649产 地：中国大陆

TQ0022Capromorelin TartrateInhibitor,Growth hormone secretagogue receptor,GHSR,Capromorelin,inhibit,Caprom

Capromorelin Tartrate is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).

价 格：￥电议型 号：TQ0022产 地：中国大陆

TQ0292GrapiprantRQ 00000007,Inhibitor,Grapiprant,CJ 023423,RQ00000007,Prostaglandin Receptor,AAT 007,inhib

Grapiprant is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM).

价 格：￥电议型 号：TQ0292产 地：中国大陆

T7806Licarbazepinepartial,Licarbazepine,Sodium Channel,Na channels,voltage,Inhibitor,sodium,seizures,stab

Licarbazepine is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial seizures and bipolar disorders.

价 格：￥电议型 号：T7806产 地：中国大陆

T15387GLP-1R Antagonist 1GLP 1R Antagonist 1,GLP1R Antagonist 1

GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).

价 格：￥电议型 号：T15387产 地：中国大陆

T60145CCR6 antagonist 1CCR6antagonist1

CCR6 antagonist 1 is a CCR6 antagonist. CCR6 antagonist 1 inhibits the CCL20/CCR6 axis. CCR6 antagonist 1 can be used in the research of autoimmune-mediated inflammatory diseases, such as inflammatory bowel diseases (IBDs).

价 格：￥电议型 号：T60145产 地：中国大陆

T38622Bcl-xL antagonist 2Bcl xL antagonist 2,BclxL antagonist 2

Bcl-xL antagonist 2 is an effective and selective antagonist of Bcl-xL with an IC50 of 91 nM and a Ki of 65 nM. Bcl-xL antagonist 2 induces apoptosis in cancer cells and can be used in studies about chronic lymphocytic leukemia and non-Hodgkin’s lymphoma.

价 格：￥电议型 号：T38622产 地：中国大陆

TQ0025E7046Inhibitor,E-7046,Prostaglandin Receptor,E7046,E 7046,inhibit

E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.

价 格：￥电议型 号：TQ0025产 地：中国大陆

TP1865LRhodopsin Epitope Tag acetateRhodopsin Epitope Tag acetate

Rhodopsin Epitope Tag acetate is a 9-amino acid peptide representing C terminus of bovine rhodopsin widely used as an epitope tag. A number of anti-rhodopsin antibodies can recognize this epitope.

价 格：￥电议型 号：TP1865L产 地：中国大陆

T61813AMPA receptor antagonist-3

AMPA receptor antagonist-3 is an AMPA receptor antagonist (patent US20070027143A1).

价 格：￥电议型 号：T61813产 地：中国大陆

T62420P2Y2R/GPR17 antagonist 1

P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist. P2Y2R/GPR17 antagonist 1 shows IC50 values of 3.17 ?M and 1.67 ?M against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes.

价 格：￥电议型 号：T62420产 地：中国大陆