T31204Darapladib-impurityDarapladib impurity,Darapladibimpurity

Darapladib-impurity is the impurity of Darapladib. Darapladib inhibits lipoprotein-associated phospholipase A2 (Lp-PLA2)

价 格：￥电议型 号：T31204产 地：中国大陆

T67698WAY-300374WAY300374

WAY-300374 inhibits the p53-MDM2 protein-protein interaction.

价 格：￥电议型 号：T67698产 地：中国大陆

T7848PT-2385Inhibitor,inhibit,Hypoxia-inducible factors,HIF/HIF Prolyl-Hydroxylase,HIF-PH,PT 2385,HIFs,PT

PT-2385 is a selective HIF-2α inhibitor (Kd<50 nM).

价 格：￥电议型 号：T7848产 地：中国大陆

T8439Clobenpropit dihydrobromideApoptosis,inhibit,Clobenpropit dihydrobromide,histamine H3R,antagonist,in

Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)

价 格：￥电议型 号：T8439产 地：中国大陆

TN12955-O-Caffeoylshikimic acidinhibit,5 O Caffeoylshikimic acid,Inhibitor,5OCaffeoylshikimic acid

5-O-Caffeoylshikimic acid shows anti-oxidative activity; it also shows anti-inflammatory activity, the underlying mechanism was associated with downregulation of nuclear factor-κB.

价 格：￥电议型 号：TN1295产 地：中国大陆

PDK04236-METHYL-1H-INDOLE-2-CARBOXYLIC ACID6METHYL1HINDOLE2CARBOXYLICACID

价 格：￥电议型 号：PDK0423产 地：中国大陆

T22849ICI 199,441 hydrochlorideICI 199,441 hydrochloride

ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.

价 格：￥电议型 号：T22849产 地：中国大陆

TN12373-O-Methylgallic acidAnthocyanin,3 O Methylgallic acid,inhibit,3OMethylgallic acid,metabolite,anti-c

3,4-Dihydroxy-5-methoxybenzoic acid reduces cell proliferation in Caco-2 cells(IC50 = 24.1 μM) more effectively than anthocyanins and may offer protection against colon cancer after its formation in the gut. 3,4-Dihydroxy-5-methoxybenzoic acid inhibits transcription factors NF-κB, AP-1, STAT-1, and OCT-1 which are known to be activated in colorectal cancer.

价 格：￥电议型 号：TN1237产 地：中国大陆

T16536Pimonidazole hydrochlorideinhibit,Pimonidazole hydrochloride,Pimonidazole,Inhibitor

Pimonidazole hydrochloride accumulates in hypoxic cells via covalent binding with macromolecules or by forming reductive metabolites after the reduction of its nitro group. It can be used for qualitative and quantitative assessment of tumor hypoxia. Pimonidazole hydrochloride is a novel hypoxia marker for the complementary study of tumor hypoxia and cell proliferation in tumors.

价 格：￥电议型 号：T16536产 地：中国大陆

TN1438beta-Amyrin acetateHMG-CoA,betaAmyrin acetate,LDL,Fungal,inhibit,Inhibitor,arthritic,hemolysis,antif

beta-Amyrin acetate inhibits HMG-CoA Reductase (HMGCR) and sEH activity with IC50 of 3.4 μM. beta-Amyrin acetate has anti-inflammatory, antifungal, antioxidant, and anti-hyperlipidemic activities.

价 格：￥电议型 号：TN1438产 地：中国大陆

TN4871PyrolinPyrolin

Pyrolin has a strong antifungal activity and exerts a potent impact on the ultrastructure of M.fructicola.

价 格：￥电议型 号：TN4871产 地：中国大陆

T22761EIT hydrobromide

EIT hydrobromide is an iNOS inhibitor.

价 格：￥电议型 号：T22761产 地：中国大陆

T9192BIIB068ADME,inhibit,FcγR,Autoimmune,Bruton tyrosine kinase,TNFα,BIIB 068,ROS,Inhibitor,reversible,Bt

BIIB068 is an selective, reversible and orally active BTK inhibitor (IC50 = 1 nM, Kd = 0.3 nM). BIIB068 is 400 times more selective for BTK than other kinases.

价 格：￥电议型 号：T9192产 地：中国大陆

TJS03384-Methylesculetininhibit,4 Methylesculetin,Glutathione Peroxidase,4-Methylesculetin,Inhibitor,4Methy

4-methylesculetin is one of the coumarin derivatives with great anti-oxidant and anti-inflammatory activities.

价 格：￥电议型 号：TJS0338产 地：中国大陆

TQ0015PRN1371inhibit,CSF1R,PRN 1371,Inhibitor,colony stimulating factor 1 receptor,c-Fms,CSF-1R,FGFR,CSF-1

PRN1371 is a specific and potent FGFR1-4 and CSF1R inhibitor (IC50s: 0.6/1.3/4.1/19.3/8.1 nM for FGFR1/2/3/4 and CSF1R).

价 格：￥电议型 号：TQ0015产 地：中国大陆

TN2100PratenseinInhibitor,Nuclear factor-kappaB,Nuclear factor-κB,cognitive,inhibit,BDNF,synapse,Pratensei

Pratensein as a novel transcriptional up-regulator of scavenger receptor class B type I in HepG2 cells.

价 格：￥电议型 号：TN2100产 地：中国大陆

T8595Practololreceptor,inhibit,arrhythmias,β1-adrenergic,Practolol,Beta Receptor,Adrenergic Receptor,card

Practolol is a selective β-adrenoceptor blocker.

价 格：￥电议型 号：T8595产 地：中国大陆

T8796CAN508inhibit,CAN 508,ATP-competitive,Cyclin dependent kinase,esophageal,cells,CDK,CAN508,Inhibitor,

CAN508 is a potent, ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 μM. It is also a competitive inhibitor of Cdk2-cyclin E with respect to ATP, with Ki and IC50 values of 13.3 and 20 μM, respectively.CAN508 exhibits a 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes. Antitumor activity.

价 格：￥电议型 号：T8796产 地：中国大陆

T7741DS-1001binhibit,DS 1001b,Inhibitor,Isocitrate Dehydrogenase (IDH),DS-1001b,DS1001b

DS-1001b is an inhibitor of mutant IDH-1 (Isocitrate Dehydrogenase-1)

价 格：￥电议型 号：T7741产 地：中国大陆

T9041AES-350Histone deacetylases,AES 350,MV4-11,AES-350,Apoptosis,acute myeloid leukemia,AML,Inhibitor,in

AES-350 is a potent and orally active HDAC6 inhibitor(IC50 and a Ki of 0.0244 μM and 0.035 μM, respectively). It is also against HDAC-3, -8, and -11 in an enzymatic activity assay with IC50 values of 0.187 μM, 0.245 μM, and >1μM, respectively. AES-350 triggers apoptosis in AML cells through HDAC inhibition and can be used for acute myeloid leukemia (AML) research.

价 格：￥电议型 号：T9041产 地：中国大陆