T22964Glemanserin

Glemanserin is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.

价 格：￥电议型 号：T22964产 地：中国大陆

T7151GSK2982772inhibit,Receptor-interacting protein kinases,GSK2982772,RIPK,Inhibitor,RIP kinase,GSK 2982

GSK2982772 is an inhibitor of receptor interacting serine/threonine kinase 1 (RIPK1)with IC50 values of 16 nM and 20 nM for human and monkey RIP1, respectively.

价 格：￥电议型 号：T7151产 地：中国大陆

T11299FLT3-IN-4

FLT3-IN-4 is a potent and orally effective Fms-like tyrosine receptor kinase 3 (FLT3;?IC50=7 nM) inhibitor ,for treating acute myelogenous leukemia.

价 格：￥电议型 号：T11299产 地：中国大陆

T7294AramcholInhibitor,inhibit,Aramchol

Aramchol, also known as arachidyl amido cholanoic acid, is a conjugate of arachidic acid and cholic acid. It reduces ex vivo cholesterol crystallization in native human bile and dissolves pre-formed cholesterol crystals in a dose-dependent manner.

价 格：￥电议型 号：T7294产 地：中国大陆

TN12975-O-Methylvisamminolinhibit,Inhibitor,5 O Methylvisamminol,5OMethylvisamminol

5-O-Methylvisamminol is a natural product

价 格：￥电议型 号：TN1297产 地：中国大陆

T22345INCB054329Inhibitor,inhibit,INCB 054329,Epigenetic Reader Domain

INCB054329, a structurally distinct bromodomain and extraterminal domain (BET) inhibitor, inhibits BRD2-BD1, BRD2-BD2, BRD3-BD1, BRD3-BD2, BRD4-BD1, BRD4-BD2, BRDT-BD1 and BRDT-BD2 with IC50 values of 44 nM, 5 nM, 9 nM, 1 nM, 28 nM, 3 nM, 119 nM and 63 nM respectively.

价 格：￥电议型 号：T22345产 地：中国大陆

TN1829KakkalideKakkalide,Inhibitor,inhibit

Kakkalide is a potent lactate dehydrogenase (LDH) inhibitor, it has anti-inflammatory effects.

价 格：￥电议型 号：TN1829产 地：中国大陆

T16929SR2211SR-2211,SR2211

SR2211 is a specific modulator and an inverse agonist of RORγ(IC50 = 320 nM, Ki = 105 nM).

价 格：￥电议型 号：T16929产 地：中国大陆

TP2137Lpp60 c-src (521-533) (phosphorylated) acetatepp60 c src (521 533) (phosphorylated) acetate,pp60 csrc

pp60 c-src (521-533) (phosphorylated) acetate is a regulator of focal adhesion formation and cell spreading. pp60 c-src (521-533) (phosphorylated) acetate also regulates cell motility and is a key component in the signaling pathway triggered by the motogenic hyaluronan receptor RHAMM.

价 格：￥电议型 号：TP2137L产 地：中国大陆

T12433PF-06952229

PF-06952229 is a selective inhibitor of TGFβRI. PF-06952229 can be used in studies about the treatment of solid tumors, specifically metastatic breast cancer.

价 格：￥电议型 号：T12433产 地：中国大陆

TQ0156GW1929GW 1929,GW1929,Peroxisome proliferator-activated receptors,PPAR,inhibit,GW-1929,Inhibitor

GW1929 is a potent PPAR-γ agonist (pKi: 8.84 for human PPAR-γ; pEC50s of 8.56 and 8.27 for human and murine PPAR-γ).

价 格：￥电议型 号：TQ0156产 地：中国大陆

T90604Compound NB-48-0729Compound NB480729,Compound NB 48 0729

价 格：￥电议型 号：T90604产 地：中国大陆

T29231ZLD1039

ZLD1039 is a potent, highly selective, and orally bioavailable EZH2 inhibitor. ZLD1039 shows potent and concentration-dependent inhibition of PRC2 enzymatic activity against EZH2 wild-type as well as Y641F, and A677G mutant enzymes with IC50 values of 5.6, 15, and 4.0?nM, respectively. ZLD1039 inhibits breast tumor growth and metastasis.

价 格：￥电议型 号：T29231产 地：中国大陆

T9788SN32976SN-32976,SN32976

SN32976 is a pan PI3K inhibitor. SN32976 potently inhibited PI3K isoforms and mTOR, displaying preferential activity for PI3Kα and sparing of PI3Kδ.

价 格：￥电议型 号：T9788产 地：中国大陆

TQ0111LDN-192960DYRK,Dual specificity tyrosine regulated kinase,Inhibitor,Dual specificity tyrosine phosph

LDN-192960 is a potent inhibitor of Haspin and DYRK2 (IC50s: 10 nM and 48 nM).

价 格：￥电议型 号：TQ0111产 地：中国大陆

T8472ERK1/2 inhibitor 2ERK-1/2 inhibitor 2,Extracellular signal regulated kinases,Inhibitor,ASTX 029,ERK1

ASTX029 is a selective and orally bioavailable extracellular signal-regulated kinases 1 and 2 (ERK 1/2) inhibitor, with potential antineoplastic activity.

价 格：￥电议型 号：T8472产 地：中国大陆

T9853STING activator Compound 53Inhibitor,HEK293T,STING agonist-12,MPYS,STING agonist12,STING,STING agoni

STING activator Compound 53 based on an oxindole core structure demonstrated robust on-target functional activation of STING (human EC50 185 nM) in immortalised and primary cells and a cytokine induction fingerprint consistent with STING activation.

价 格：￥电议型 号：T9853产 地：中国大陆

T60007WAY-329764WAY329764,WAY 329764

WAY-329764 is an antibacterial agent (extracted from patent RU2371444 C1).

价 格：￥电议型 号：T60007产 地：中国大陆

T9294DL-ValineDL-Valine,DL Valine,DLValine,inhibit,Inhibitor

DL-Valine is 2-amino-3-methylbutanoic acid.It is synthesized in plants via several steps starting from pyruvic acid.

价 格：￥电议型 号：T9294产 地：中国大陆

TP1863LGlucagon (19-29), human acetateGlucagon (1929), human acetate,Glucagon (19 29), human acetate

Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.

价 格：￥电议型 号：TP1863L产 地：中国大陆