T6173BI 25364-[[(7R)-8-环戊基-7-乙基-5,6,7,8-四氢-5-甲基-6-氧代-2-喋啶基]氨基]-3-甲氧基-N-(1-甲基-4-哌啶基)苯甲酰胺

BI2536 is an effective Plk1 inhibitor (IC50: 0.83 nM). It has 4- and 11-fold greater selectivity than Plk2 and Plk3.

价 格：￥电议型 号：T6173产 地：中国大陆

T6169Indirubin靛玉红；Indigopurpurin；NSC 105327；Couroupitine B；Indigo red

Indirubin is a potent cyclin-dependent kinases and GSK-3β inhibitor with IC50 of about 5 uM and 0.6 uM.

价 格：￥电议型 号：T6169产 地：中国大陆

T6078SaracatinibAZD0530；塞卡替尼

Saracatinib (AZD0530) is an effective Src inhibitor (IC50: 2.7 nM), and effective to Lck, Fyn, Lyn, Blk, Fgr and c-Yes.

价 格：￥电议型 号：T6078产 地：中国大陆

T6053Turofexorate Isopropyl妥芬异丙酯；FXR-450；XL335；WAY-362450

Turofexorate Isopropyl (XL335) is a potent, selective, and orally bioavailable FXR agonist with EC50 of 4 nM

价 格：￥电议型 号：T6053产 地：中国大陆

T5S1530Isochlorogenic acid C金银花；异绿原酸C

1. Isochlorogenic acid C has antioxidant activity.

价 格：￥电议型 号：T5S1530产 地：中国大陆

T5S0053CoptisineCoptisin；黄连碱

1. Coptisine treatment increases cell viability based on its reversal effect on the enhanced activity of Indoleamine 2, 3-dioxygenase . 2. Coptisine treats myocardial I/R likely through suppressing myocardial apoptosis and inflammation by inhibiting the R

价 格：￥电议型 号：T5S0053产 地：中国大陆

T59531-Aminobenzotriazole1-氨基苯并三唑；3-Aminobenzotriazole；ABT

1-Aminobenzotriazole (ABT) is a non-specific cytochrome P450 (CYP) inhibitor.

价 格：￥电议型 号：T5953产 地：中国大陆

T5853Rubitecan鲁比特康；9-Nitrocamptothecin；RFS 2000

Rubitecan is a DNA topoisomerase I inhibitor. It inhibits DNA topoisomerase I and increases the fraction of supercoiled DNA in a cell-free assay in a concentration-dependent manner.Rubitecan is a semisynthetic agent related to camptothecin with potent ant

价 格：￥电议型 号：T5853产 地：中国大陆

T5753Flavokawain C黄卡瓦胡椒素 C；卡瓦胡椒素C

Flavokawain C (FKC), a naturally occurring chalcone, which can be isolated from Kava.FKC has the potential to be developed into chemotherapeutic drug for the treatment of colon adenocarcinoma.

价 格：￥电议型 号：T5753产 地：中国大陆

T5653Cinnamyl acetate乙酸桂酯；3-Phenylallyl acetate

价 格：￥电议型 号：T5653产 地：中国大陆

T5538DC661

DC661 is palmitoyl-protein thioesterase 1 (PPT1) inhibitor, inhibits autophagy, and acts as an anti-lysosomal agent. Anti-cancer activity

价 格：￥电议型 号：T5538产 地：中国大陆

T5537IDF-11774

IDF-11774 is a HIF-1 inhibitor.It reduces hif-1α HRE luciferase activity (IC50 = 3.65 μM).

价 格：￥电议型 号：T5537产 地：中国大陆

T5536SJA710-6

SJA710-6 is a small molecule able to selectively differentiate MSCs toward hepatocyte-like cells.

价 格：￥电议型 号：T5536产 地：中国大陆

T5535ERK5-IN-2

ERK5-IN-2 is an orally active, sub-micromolar, selective ERK5 inhibitor with IC50s of 0.82 μM, 3 μM for ERK5 and ERK5 MEF2D, respectively.

价 格：￥电议型 号：T5535产 地：中国大陆

T5534LOC14

LOC14 to be the most potent PDI inhibitor reported to date( EC50 : 500 nM)

价 格：￥电议型 号：T5534产 地：中国大陆

T5533MC180295(rel)-MC180295

MC180295 is a novel potent, highly selective CDK9 inhibitor (IC50: 5 nM), displays >22-fold selectivity over other CDKs.

价 格：￥电议型 号：T5533产 地：中国大陆

T5532BMS-687453

BMS-687453 is a potent and selective PPAR alpha agonist, with an EC(50) of 10 nM for human PPARalpha and approximately 410-fold selectivity vs human PPARgamma in PPAR-GAL4 transactivation assays.

价 格：￥电议型 号：T5532产 地：中国大陆

T5531GSK-4716

GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand

价 格：￥电议型 号：T5531产 地：中国大陆

T5511L-765314

L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the role of α1B receptors in the regulation of blood pressure.

价 格：￥电议型 号：T5511产 地：中国大陆

T54533-Methyltoxoflavin3-methyl toxoflavin

3-methyltoxoflavin is an effective inhibitor of protein disulfide isomerase (PDI) and its IC50 value is 170 nM.

价 格：￥电议型 号：T5453产 地：中国大陆