当前位置：易推广 > 上海陶术生物科技有限公司 > 产品展示
企业档案
会员类型：会员
已获得易推广信誉 等级评定
(0 -40)基础信誉积累，可浏览访问
(41-90)良好信誉积累，可接洽商谈
(91+ )优质信誉积累，可持续信赖
易推广会员：5年
工商认证 【已认证】
最后认证时间：
注册号： 【已认证】
法人代表： 【已认证】
企业类型：生产商 【已认证】
注册资金：人民币万 【已认证】
产品数：86101
参观次数：3605811
自主品牌
已选条件
-
T16810Ruzadolane；卢扎朵仑UP 26-91；卢扎朵仑|||UP 26-91
Ruzadolane (formerly known as UP 26-91) is a 5-hydroxytryptamine receptor antagonist developed as a non-narcotic central analgesic for the treatment of anxiety disorders and pain.
价 格：￥电议型 号：T16810产 地：中国大陆
-
T16791Rottlerin；粗糠柴苦素Mallotoxin|||NSC 56346|||NSC 94525；Mallotoxin|||NSC 56346|||粗糠柴苦素|||NSC 94525
Rottlerin (NSC-56346) is a natural product purified from Mallotus Philippinensis and is a specific PKC inhibitor (IC50: PKCδ of 3-6 μM, PKCα,β,γ of 30-42 μM, PKCε,η,ζ of 80-100 μM). Rottlerin causes apoptosis via caspase 3 activation.
价 格：￥电议型 号：T16791产 地：中国大陆
-
T16783Rolziracetam；罗拉西坦CI-911；罗拉西坦|||CI-911
Rolziracetam (CI-911) is a nootropic drug of the racetam family. It can improve short-term memory in rats and monkeys.
价 格：￥电议型 号：T16783产 地：中国大陆
-
T16774RO-9187；化合物 T16774RO-9187
RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).
价 格：￥电议型 号：T16774产 地：中国大陆
-
T16757Risdiplam；化合物RisdiplamRO7034067|||RG7916；RO7034067|||RG7916
Risdiplam (RO7034067) (RG7916) is orally administered. Risdiplam is a centrally and peripherally distributed SMN2 pre-mRNA splicing modifier which increases survival motor neuron (SMN) protein levels[1].
价 格：￥电议型 号：T16757产 地：中国大陆
-
T16750Rigosertib；瑞格色替ON-01910；ON-01910|||瑞格色替
Rigosertib (ON-01910) is a selective and non-ATP-competitive inhibitor of PLK1 (IC50: 9 nM). Rigosertib is a multi-kinase inhibitor and a selective anti-cancer agent, which induces apoptosis by inhibition of the PI3 kinase/Akt pathway, promotes the phosphorylation of histone H2AX and induces G2/M arrest in the cell cycle.
价 格：￥电议型 号：T16750产 地：中国大陆
-
T16713R121919；化合物R121919NBI30775；NBI30775
R121919 (NBI30775) is a potent small molecule adrenocorticotropic hormone-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity that inhibits the CRF1 receptor, the CRF2 receptor, and the CRF-binding proteins.
价 格：￥电议型 号：T16713产 地：中国大陆
-
T16691Pyrene-amido-PEG4-azide；化合物 T16691Pyrene-amido-PEG4-azide
Pyrene-amido-PEG4-azide is a PEG-based proteolysis targeting chimera (PROTAC) linker utilized for synthesizing PROTACs [1].
价 格：￥电议型 号：T16691产 地：中国大陆
-
T16591Propargyl-PEG1-SS-PEG1-PFP ester；化合物 T16591Propargyl-PEG1-SS-PEG1-PFP ester
Propargyl-PEG1-SS-PEG1-PFP ester is a cleavable linker consisting of a 1-unit polyethylene glycol (PEG) backbone, designed for use in the synthesis of antibody-drug conjugates (ADCs)[1].
价 格：￥电议型 号：T16591产 地：中国大陆
-
T16510PF-915275；化合物PF-915275PF-915275
PF-915275 is an effective and selective inhibitor of human 11β-hydroxysteroid dehydrogenase type 1 (11βHSD1, Ki = 2.3 nM, EC50 = 15 nM in vitro HEK293 cells). The dose-dependent effect of PF-915275 on conversion of cortisone to cortisol in primary human and monkey hepatocytes, with an EC50 of 20 and 100 nM, respectively.
价 格：￥电议型 号：T16510产 地：中国大陆
-
T16506PF-4878691；化合物PF-48786913M-852A；3M-852A
PF-4878691 (3M-852A) is an effective and selective Toll-like receptor 7 agonists modelled. It is used to dissociate its antiviral and inflammatory activities.
价 格：￥电议型 号：T16506产 地：中国大陆
-
T16503PF-4191834；化合物PF-4191834PF-04191834；PF-04191834
PF-4191834 is a noniron chelating and non-redox inhibitor of the 5-Lipoxygenase (5-LOX) with an IC50 of 229 nM. PF-4191834 shows ~300-fold selectivity for 5-LOX over 12-LOX and 15-LOX and displays no activity toward the cyclooxygenase enzymes. PF-4191834
价 格：￥电议型 号：T16503产 地：中国大陆
-
T16491PF-06446846 hydrochloride；化合物PF-06446846盐酸盐PF-06446846 hydrochloride
PF-06446846 hydrochloride, an orally active and highly selective inhibitor, targets Proprotein Convertase Subtilisin/Kexin type 9 (PCSK9) translation by inducing ribosomal stalling at approximately codon 34, effectively suppressing PCSK9 expression.
价 格：￥电议型 号：T16491产 地：中国大陆
-
T16480PF-04991532；化合物 T16480PF-04991532
PF-04991532 is an effective, hepatoselective glucokinase activator. It has EC50s of 80 and 100 nM in human and rat, respectively.
价 格：￥电议型 号：T16480产 地：中国大陆
-
T1643Penciclovir；喷昔洛韦BRL 39123|||VSA 671；喷昔洛韦|||BRL 39123|||VSA 671
Penciclovir (BRL 39123) is a Herpesvirus Nucleoside Analog DNA Polymerase Inhibitor. In HSV infected cells, penciclovir is phosphorylated by viral thymidine kinase and subsequently converted by cellular kinases into the active metabolite, penciclovir triphosphate, which competitively inhibits viral HSV polymerase by blocking deoxyguanosine triphosphate substrate binding. As a result, herpes viral DNA synthesis and replication are selectively inhibited.
价 格：￥电议型 号：T1643产 地：中国大陆
-
T16391ON-013100；化合物ON-013100ON-013100
ON-013100 is an antineoplastic drug. ON-013100 also acts as a mitotic inhibitor that could inhibit Cyclin D1 expression.
价 格：￥电议型 号：T16391产 地：中国大陆
-
T16339Norverapamil hydrochloride；盐酸去甲维拉帕米(±)-Norverapamil hydrochloride|||D591 hydrochloride；(±)-Norverapa
Norverapamil hydrochloride (D591 hydrochloride) ((±)-Norverapamil hydrochloride) is an N-demethylated metabolite of Verapamil and it is an L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor.
价 格：￥电议型 号：T16339产 地：中国大陆
-
T16291NF157；化合物 T16291NF157
NF157 significantly decreases the expression of metalloproteinase (MMP)-3, MMP-13, which can be used in the treatment of osteoarthritis (OA). NF157 is a highly selective nanomolar P2Y11 antagonist (pKi: 7.35). The IC50s are 463 nM, 1811 μM, 170 μM for P2Y11 (Ki=44.3 nM), P2Y1 (Ki=187 μM), P2Y2 (Ki=28.9 μM), respectively.
价 格：￥电议型 号：T16291产 地：中国大陆
-
T16191N-(Azido-PEG3)-N-Fluorescein-PEG3-acid；化合物 T16191N-(Azido-PEG3)-N-Fluorescein-PEG3-acid
N-(Azido-PEG3)-N-Fluorescein-PEG3-acid is a PEGylated PROTAC linker incorporating azide, fluorescein, and carboxylic acid functional groups.
价 格：￥电议型 号：T16191产 地：中国大陆
-
T16162Mutated EGFR-IN-1；AZD9291中间体1Osimertinib analog；Osimertinib analog|||AZD9291中间体1
Mutated EGFR-IN-1 (Osimertinib analog) is a useful intermediate for the inhibitors design for mutated EGFR, such as L858R EGFR, Exonl9 deletion activating mutant, and T790M resistance mutant.
价 格：￥电议型 号：T16162产 地：中国大陆
