T6S0105PeiminineInhibitor,inhibit,Peiminine,Autophagy

1. Peiminine is an effective inhibitor for lung inflammation and pulmonary fibrosis in a rat model of bleomycin-induced lung injury.

价 格：￥电议型 号：T6S0105产 地：中国大陆

T5467SAR125844Inhibitor,SAR125844,c-Met/HGFR,inhibit,SAR 125844,SAR-125844,Apoptosis

SAR125844, a potent and highly selective inhibitor of the MET receptor tyrosine kinase (RTK), for intravenous administration. (IC50 value of 4.2 nmol/L)

价 格：￥电议型 号：T5467产 地：中国大陆

PDK0168Compound PDK0168Compound PDK0168

价 格：￥电议型 号：PDK0168产 地：中国大陆

T17875Pomalidomide-C2-NH2Inhibitor,E3 Ligase Ligand-Linker Conjugates,PomalidomideC2NH2,Pomalidomide-C-2-N

Pomalidomide-C2-NH2 is a synthesized E3 ligase ligand-linker conjugate containing a Pomalidomide-based cereblon ligand and a linker.

价 格：￥电议型 号：T17875产 地：中国大陆

Fr12622Compound Fr12622Compound Fr12622

价 格：￥电议型 号：Fr12622产 地：中国大陆

T9609GRK5-IN-2metabolic,bicyclic,insulin,kinase,inhibit,Inhibitor,disease,pyridine-based,GRK5 IN 2,GRK-5-

GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor. It regulates the expression and/or release of insulin and is useful for the metabolic disease research.

价 格：￥电议型 号：T9609产 地：中国大陆

TN1026Vomicineinhibit,Inhibitor,activity,Vomicine,alkaloid,antidiabetic

Vomicine is a natural product from Strychnos nux-vomica, the S. nux-vomica extracts show antihyperglycemic activity in experimental animals.

价 格：￥电议型 号：TN1026产 地：中国大陆

TN12613-O-Caffeoylquinic acid methyl esterInhibitor,inhibit,3 O Caffeoylquinic acid methyl ester,3OCaffeoy

3-O-Caffeoylquinic acid methyl ester is a natural product from Morus alba L.

价 格：￥电议型 号：TN1261产 地：中国大陆

T60123Chimmitecan

Chimmitecan is a potent inhibitor of topoisomerase I and displays outstanding activity in vitro and in vivo.

价 格：￥电议型 号：T60123产 地：中国大陆

T6635EMD638683inhibit,EMD-638683,EMD638683,Serum and glucocorticoid-regulated kinase,EMD 638683,Inhibitor

EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).

价 格：￥电议型 号：T6635产 地：中国大陆

T7622GabazineInhibitor,Gamma-aminobutyric acid Receptor,Gabazine,γ-Aminobutyric acid Receptor,inhibit,SR

Gabazine is an antagonist of GABAA receptors (Ki : 74-150 nM)

价 格：￥电议型 号：T7622产 地：中国大陆

TP2212La-MSH, amide Acetate(581-05-5 free base)a MSH, amide Acetate(581 05 5 free base),aMSH, amide Acetate

a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities. α-MSH is a post-translational derivative of pro-opiomelanocortin (POMC)

价 格：￥电议型 号：TP2212L产 地：中国大陆

TQ0029ASTX660Inhibitor,inhibit,ASTX-660,ASTX660,IAP,ASTX 660

ASTX660 is an orally bioavailable dual antagonist of cIAP and XIAP.

价 格：￥电议型 号：TQ0029产 地：中国大陆

TN71672,4,5-Tribromoimidazole

2,4,5-Tribromoimidazole is a marine derived natural products found in Hexaplex trunculus.

价 格：￥电议型 号：TN7167产 地：中国大陆

T37082HS271HS271,HS-271

HS271 is a selective, highly potent and orally active IRAK4 inhibitor (IC50= 7.2 μM). HS271 shows excellent enzymatic and cellular activities, as well as excellent pharmacokinetic properties.

价 格：￥电议型 号：T37082产 地：中国大陆

TQ0271Falnidamol

Falnidamol is an orally active, selective EGFR tyrosine kinase inhibitor with an IC50 of 3 nM. Falnidamol displays > 1000-fold lower potency against ErbB2 (IC50=3.4 μM) and a range of other related tyrosine kinases (IC50>10 μM). Falnidamol is a pyrimido-pyrimidine compound and has anti-cancer activity.

价 格：￥电议型 号：TQ0271产 地：中国大陆

T6917OleuropeinPPARγ,olive,PPAR,Peroxisome proliferator-activated receptors,inhibit,Apoptosis,leaves,Oleu

Oleuropein is an antioxidant polyphenol isolated from olive leaf.

价 格：￥电议型 号：T6917产 地：中国大陆

T7295MiridesapGSK 2315698,GSK-2315698,Miridesap,Inhibitor,inhibit

Miridesap is a divalent crosslinker of SAP that causes rapid depletion of circulating SAP via hepatic clearance. It also produces significant reduction of SAP from cerebrospinal fluid and visceral amyloid deposits

价 格：￥电议型 号：T7295产 地：中国大陆

T7604ValrubicinInhibitor,AD 32,AD32,Valrubicin,inhibit,PKC,Antibiotic,Protein kinase C

Valrubicin (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and has antitumor and anti-inflammatory activity.

价 格：￥电议型 号：T7604产 地：中国大陆

TCS0102PulegoneEndogenous Metabolite,Transient receptor potential channels,TRP Channel,Pulegone,Inhibitor,i

1. Pulegone has cytotoxicity followed by regenerative cell proliferation is the MOA for Pulegone-induced urothelial tumors in female rats. 2. Pulegone induces a verapamil-sensitive psychostimulant effect that appears to independ on the opening of L-type calcium channels. 3. Pulegone has negative reinforcing properties and seems to possess anxiolytic-like actions unrelated to the benzodiazepine site of the γ-aminobutyric acid type A (GABAA) receptor.

价 格：￥电议型 号：TCS0102产 地：中国大陆