Fr12622Compound Fr12622Compound Fr12622

价 格：￥电议型 号：Fr12622产 地：中国大陆

T9609GRK5-IN-2metabolic,bicyclic,insulin,kinase,inhibit,Inhibitor,disease,pyridine-based,GRK5 IN 2,GRK-5-

GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor. It regulates the expression and/or release of insulin and is useful for the metabolic disease research.

价 格：￥电议型 号：T9609产 地：中国大陆

TN1026Vomicineinhibit,Inhibitor,activity,Vomicine,alkaloid,antidiabetic

Vomicine is a natural product from Strychnos nux-vomica, the S. nux-vomica extracts show antihyperglycemic activity in experimental animals.

价 格：￥电议型 号：TN1026产 地：中国大陆

TN12613-O-Caffeoylquinic acid methyl esterInhibitor,inhibit,3 O Caffeoylquinic acid methyl ester,3OCaffeoy

3-O-Caffeoylquinic acid methyl ester is a natural product from Morus alba L.

价 格：￥电议型 号：TN1261产 地：中国大陆

T60123Chimmitecan

Chimmitecan is a potent inhibitor of topoisomerase I and displays outstanding activity in vitro and in vivo.

价 格：￥电议型 号：T60123产 地：中国大陆

T6635EMD638683inhibit,EMD-638683,EMD638683,Serum and glucocorticoid-regulated kinase,EMD 638683,Inhibitor

EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).

价 格：￥电议型 号：T6635产 地：中国大陆

T7622GabazineInhibitor,Gamma-aminobutyric acid Receptor,Gabazine,γ-Aminobutyric acid Receptor,inhibit,SR

Gabazine is an antagonist of GABAA receptors (Ki : 74-150 nM)

价 格：￥电议型 号：T7622产 地：中国大陆

TP2212La-MSH, amide Acetate(581-05-5 free base)a MSH, amide Acetate(581 05 5 free base),aMSH, amide Acetate

a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities. α-MSH is a post-translational derivative of pro-opiomelanocortin (POMC)

价 格：￥电议型 号：TP2212L产 地：中国大陆

T67742EX-A5386

EX-A5386 is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.

价 格：￥电议型 号：T67742产 地：中国大陆

TQ0029ASTX660Inhibitor,inhibit,ASTX-660,ASTX660,IAP,ASTX 660

ASTX660 is an orally bioavailable dual antagonist of cIAP and XIAP.

价 格：￥电议型 号：TQ0029产 地：中国大陆

TN71672,4,5-Tribromoimidazole

2,4,5-Tribromoimidazole is a marine derived natural products found in Hexaplex trunculus.

价 格：￥电议型 号：TN7167产 地：中国大陆

T37082HS271HS271,HS-271

HS271 is a selective, highly potent and orally active IRAK4 inhibitor (IC50= 7.2 μM). HS271 shows excellent enzymatic and cellular activities, as well as excellent pharmacokinetic properties.

价 格：￥电议型 号：T37082产 地：中国大陆

TQ0271Falnidamol

Falnidamol is an orally active, selective EGFR tyrosine kinase inhibitor with an IC50 of 3 nM. Falnidamol displays > 1000-fold lower potency against ErbB2 (IC50=3.4 μM) and a range of other related tyrosine kinases (IC50>10 μM). Falnidamol is a pyrimido-pyrimidine compound and has anti-cancer activity.

价 格：￥电议型 号：TQ0271产 地：中国大陆

T6917OleuropeinPPARγ,olive,PPAR,Peroxisome proliferator-activated receptors,inhibit,Apoptosis,leaves,Oleu

Oleuropein is an antioxidant polyphenol isolated from olive leaf.

价 格：￥电议型 号：T6917产 地：中国大陆

TP1086Men 10376 TFA(135306-85-3,free)Men 10376 TFA(135306853,free),Men 10376 TFA(135306 85 3,free)

Men 10376 TFA is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.

价 格：￥电议型 号：TP1086产 地：中国大陆

T7295MiridesapGSK 2315698,GSK-2315698,Miridesap,Inhibitor,inhibit

Miridesap is a divalent crosslinker of SAP that causes rapid depletion of circulating SAP via hepatic clearance. It also produces significant reduction of SAP from cerebrospinal fluid and visceral amyloid deposits

价 格：￥电议型 号：T7295产 地：中国大陆

T7604ValrubicinInhibitor,AD 32,AD32,Valrubicin,inhibit,PKC,Antibiotic,Protein kinase C

Valrubicin (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and has antitumor and anti-inflammatory activity.

价 格：￥电议型 号：T7604产 地：中国大陆

T11178LELN318463 racemate

ELN318463 racemate is the racemate of ELN318463 which is an amyloid precursor protein (APP) selective γ-secretase inhibitor.

价 格：￥电议型 号：T11178L产 地：中国大陆

TCS0102PulegoneEndogenous Metabolite,Transient receptor potential channels,TRP Channel,Pulegone,Inhibitor,i

1. Pulegone has cytotoxicity followed by regenerative cell proliferation is the MOA for Pulegone-induced urothelial tumors in female rats. 2. Pulegone induces a verapamil-sensitive psychostimulant effect that appears to independ on the opening of L-type calcium channels. 3. Pulegone has negative reinforcing properties and seems to possess anxiolytic-like actions unrelated to the benzodiazepine site of the γ-aminobutyric acid type A (GABAA) receptor.

价 格：￥电议型 号：TCS0102产 地：中国大陆

TQ0187SR-3677Inhibitor,Rho-associated protein kinase,Autophagy,SR 3677,Rho-kinase,SR3677,ROCK,ROK,SR-3677,

SR-3677 is an effective and specific inhibitor of ROCK2 (IC50: 3 nM).

价 格：￥电议型 号：TQ0187产 地：中国大陆