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  • T14783Bromo-PEG1-acid；化合物 T14783Bromo-PEG1-acid

    Bromo-PEG1-acid is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

    价 格：￥电议型 号：T14783产 地：中国大陆

  • T14683BMS-983970；化合物 T14683BMS-983970

    BMS-983970 is an oral inhibitor of pan-Notch, and for the treatment of multiplecancers.

    价 格：￥电议型 号：T14683产 地：中国大陆

  • T14672BMS-248360；化合物 T14672BMS-248360

    BMS-248360 is a potent and orally active dual antagonist of both angiotensin II receptor (AT1) and endothelin A (ETA) receptor. With Kis of 10 nM and 1.9 nM for hAT1 and hETA receptor, respectively. BMS-248360 shows hypertensive effects[1].

    价 格：￥电议型 号：T14672产 地：中国大陆

  • T14583Biotin-PEG2-azide；化合物 T14583Biotin-PEG2-azide

    Biotin-PEG2-azide is a PEG-based PROTAC linker can be used in the synthesis of PROTACs.

    价 格：￥电议型 号：T14583产 地：中国大陆

  • T14506BAY 60-6583；化合物BAY 60-6583BAY 60-6583

    BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 receptors.BAY 60-6583 is cardioprotective in a model of myocardial ischemia.The Ki values for BAY 60-6583 binding to mouse, rabbit, and dog A2BAR were 750 nM, 340 nM, and 330 nM, respectively. The Ki values of BAY 60-6583 binding to A2BAR in mice, rabbits and dogs were 750 nM, 340 nM and 330 nM respectively.

    价 格：￥电议型 号：T14506产 地：中国大陆

  • T14483Azido-PEG9-Boc；化合物 T14483Azido-PEG9-Boc

    Azido-PEG9-Boc is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

    价 格：￥电议型 号：T14483产 地：中国大陆

  • T1446Bambuterol hydrochloride；盐酸班布特罗(±)-Bambuterol hydrochloride|||KWD-2183 hydrochloride|||Bambuterol HC

    Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.

    价 格：￥电议型 号：T1446产 地：中国大陆

  • T14383AZD8329；化合物 T14383AZD8329

    AZD8329 is a selectable and potent inhibitor of human recombinant 11β-HSD1 and isolated human adipocyte 11?-HSD1 and is an inhibitor of rat 11β-HSD1 (IC50 - 89nM) and dog recombinant 11β-HSD1. AZD8329 has a higher affinity for 11β-HSD1 than human recombinant 11β-HSD2 and 17 AZD8329 has the ability to reduce the activity of 11β-HSD1 in adipose tissue and liver samples.

    价 格：￥电议型 号：T14383产 地：中国大陆

  • T14378LAZD5582 acetate (1258392-53-8 free base)；化合物AZD5582 acetateAZD5582 acetate (1258392-53-8 free base)

    AZD5582 acetate is an inhibitor of IAPs, which binds to the BIR3 domains cIAP1, cIAP2, and XIAP with IC50s of 15, 21, and 15 nM, respectively. AZD5582 induces apoptosis.

    价 格：￥电议型 号：T14378L产 地：中国大陆

  • T14360AX-15836；化合物AX-15836AX-15836

    AX-15836 is an inhibitor of ERK5 (IC50 : 8 nM).

    价 格：￥电议型 号：T14360产 地：中国大陆

  • T14283amyloid P-IN-1；化合物amyloid P-IN-1amyloid P IN 1|||amyloid P-IN-1|||amyloid PIN1；amyloid P IN 1|||amyl

    amyloid P-IN-1 can be used in studies about diseases with depletion of serum amyloid P components such as Alzheimer´s disease, amyloidosis, osteoarthritis, and type 2 diabetes mellitus.

    价 格：￥电议型 号：T14283产 地：中国大陆

  • T14216AMG 837；化合物 T14216AMG 837

    AMG 837 is a partial GPR40 agonist with an EC50 value of 13 nM, showcasing 85% of the maximal activity displayed by DHA in standard assay conditions, indicating its high potency and selectivity in vitro. This compound excels as a GPR40 agonist with a notable pharmacokinetic profile, effectively stimulating insulin secretion in a glucose-dependent manner in rodents and demonstrating potent insulin secretion stimulation in MIN6 cells, with efficacy comparable to that observed in aequorin Ca2+-flux

    价 格：￥电议型 号：T14216产 地：中国大陆

  • T14215AMG 837 sodium salt；化合物 T14215AMG 837 sodium salt

    AMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. IC50 value: 13 nM (EC50) [1] Target: GPR40 agonist AMG 837 displayed the expected two-fold increase in potency on GPR4 (EC50 = 13 [±7] nM) compared to the racemic compound and its activity crossed over to the rat and mouse forms of GPR40 (EC50 = 23 and 13 nM, respectively). AMG 837 is a highly potent stimulator of insulin secr

    价 格：￥电议型 号：T14215产 地：中国大陆

  • T14183Alkyne-PEG4-maleimide；化合物 T14183Alkyne-PEG4-maleimide

    Alkyne-PEG4-maleimide is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.

    价 格：￥电议型 号：T14183产 地：中国大陆

  • T14144AGN-195183；化合物 T14144AGN-195183

    AGN 195183 is a potent and selective agonist of RARα(Kd=3 nM) with improved binding selectivity relative to AGN 193836; no activity on RARβ/γ. IC50 value: 3 nM (Kd); 200 nM (EC80, RAR Trans.) Target: RARα agonist Compound 4(AGN-195183) inhibited the growth of breast cancer cell lines, and was inactive in an in vivo model of topical irritation. Compound 4 (AGN 195183) is currently in Phase I/IIA clinical trials in cancer patients. Compound 4 and ATRA inhibit growth of the human breast cancer cell

    价 格：￥电议型 号：T14144产 地：中国大陆

  • T14083Abaperidone；阿巴哌酮Abaperidone

    Abaperidone is a potent 5-HT2A receptor and dopamine D2 receptor antagonist with an IC50 of 6.2 for 5-HT2A receptors and 17 nM for dopamine D2 receptors.Abaperidone is a potentially atypical anti-psychotropic compound that reduces basal hsp70 mRNA expression in rat striatum and prefrontal cortex. expression in the striatum and prefrontal cortex of rats.

    价 格：￥电议型 号：T14083产 地：中国大陆

  • T14076A 839977；化合物A 839977A839977|||A-839977；A839977|||A-839977

    A 839977 is a selective P2X7 receptor antagonist with anti-inflammatory and analgesic activity that inhibits BzATP-induced calcium efflux from the P2X7 receptor for the study of renal fibrosis.

    价 格：￥电议型 号：T14076产 地：中国大陆

  • T140555Z-7-Oxozeaenol；化合物5Z-7-OxozeaenolFR148083|||L783279|||LL-Z 1640-2；FR148083|||L783279|||LL-Z 1640-2

    5Z-7-Oxozeaenol (FR148083) is a potent, irreversible and selective inhibitor of transforming growth factor (TGF)-β-activated kinase 1 with IC50 of 8.1 nM for TAK1 and low activity against MEK1 with IC50 of 411 nM, it is also an inhibitor of VEGF-R2 with IC50 of 52 nM.

    价 格：￥电议型 号：T14055产 地：中国大陆

  • T140283,6,9-Trioxaundecanedioic Acid；化合物 T140283,6,9-Trioxaundecanedioic Acid

    369-Trioxaundecanedioic Acid, a PEG-based PROTAC linker, facilitates PROTAC synthesis[1].

    价 格：￥电议型 号：T14028产 地：中国大陆

  • T139830990CL；化合物0990CL0990CL

    0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMP regulation. In the cell model, low concentration of 0990CL could partially restore cAMP level, and high concentration of 0990CL (10μM) began to have negative effects on cell viability.

    价 格：￥电议型 号：T13983产 地：中国大陆

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