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T79367CDK9-IN-27；化合物 CDK9-IN-27CDK9-IN-27
CDK9-IN-27 (Compound 6a), a CDK9 inhibitor with an IC50 of 0.424 μM, induces apoptosis and S-phase cell cycle arrest. It exhibits cytotoxicity against HepG2, HCT-116, and MCF-7 cell lines, with IC50 values ranging from 10.31 to 40.34 μM, rendering it applicable in cancer research [1].
价 格：￥电议型 号：T79367产 地：中国大陆
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T79365TIM-3-IN-2；TIM-3 抑制剂2TIM-3-IN-2
TIM-3-IN-2 is a Tim3 inhibitor that inhibits the binding of TIM-3 to PtdSer, CEACAM1, and Gal-9 and inhibits the action of TIM-3.TIM-3-IN-2 is able to reverse TIM-3-mediated pro-inflammatory cytokine action.
价 格：￥电议型 号：T79365产 地：中国大陆
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T79360COX-2/15-LOX-IN-2；化合物 COX-2/15-LOX-IN-2COX-2/15-LOX-IN-2
COX-2/15-LOX-IN-2 is a potent inhibitor of both COX-2 and 15-LOX, demonstrating IC50 values of 0.065 μM for COX-2 and 1.86 μM for 15-LOX. Additionally, it exhibits significant antioxidant activity [1].
价 格：￥电议型 号：T79360产 地：中国大陆
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T79354CDK9-IN-24；化合物 CDK9-IN-24CDK9-IN-24
CDK9-IN-24 (compound 21a) is a potent and selective inhibitor of CDK9 that exhibits a pronounced inhibitory impact on tumor proliferation. It impedes cell growth and triggers apoptosis via the downregulation of Mcl-1 and c-Myc, rendering it valuable in the study of acute myeloid leukemia [1].
价 格：￥电议型 号：T79354产 地：中国大陆
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T79353P-gp/BCRP-IN-2；化合物 P-gp/BCRP-IN-2P-gp/BCRP-IN-2
P-gp/BCRP-IN-2 (compound 15), an oxadiazole derivative, functions as a dual inhibitor targeting both the ABC transporter P-glycoprotein (IC50: 1.6 nM) and BCRP (IC50: 600 nM). Additionally, it bolsters the anti-proliferative impact of Doxorubicin in the drug-resistant HT29/DX and MDCK-MDR1 human adenocarcinoma colon cancer cell lines [1].
价 格：￥电议型 号：T79353产 地：中国大陆
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T79337IRAK4-IN-28；化合物 IRAK4-IN-28IRAK4-IN-28
IRAK4-IN-28 (compound 42), an orally-active IRAK4 inhibitor (IC50=8.9 nM), exhibits strong binding affinity with a Kd of 0.58 nM for the target enzyme. It is utilized for research purposes in the study of inflammation and autoimmune diseases [1].
价 格：￥电议型 号：T79337产 地：中国大陆
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T79307DNA polymerase-IN-2；化合物 DNA polymerase-IN-2DNA polymerase-IN-2
DNA polymerase-IN-2 (Compd 3c), a coumarin derivative, demonstrates inhibitory activity towards Taq DNA polymerase, with an IC50 value of 48.25 μM, and holds potential for application in value-added disease research [1].
价 格：￥电议型 号：T79307产 地：中国大陆
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T79291MmpL3-IN-2；化合物 MmpL3-IN-2MmpL3-IN-2
MmpL3-IN-2, an inhibitor targeting MmpL3, exhibits low cytotoxicity and moderate metabolic stability, making it suitable for tuberculosis research [1].
价 格：￥电议型 号：T79291产 地：中国大陆
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T79286TRAP1-IN-2；化合物 TRAP1-IN-2TRAP1-IN-2
TRAP1-IN-2, also known as compound 36, is a selective degrader of the TRAP1 client protein that does not affect Hsp90-cytosolic clients. It inhibits oxidative phosphorylation (OXPHOS) and shifts cellular metabolism toward glycolysis. Additionally, TRAP1-IN-2 compromises the stability of the TRAP1 tetramer and disrupts the mitochondrial membrane potential [1].
价 格：￥电议型 号：T79286产 地：中国大陆
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T79276PAD4-IN-2；化合物 PAD4-IN-2PAD4-IN-2
PAD4-IN-2 (compound 5i) is a PAD4 inhibitor with an IC50 value of 1.94 μM, shown to suppress tumor growth in mice through specific inhibition of the PAD4-H3cit-NETs pathway in neutrophils [1].
价 格：￥电议型 号：T79276产 地：中国大陆
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T79259α-Glucosidase-IN-25；化合物 α-Glucosidase-IN-25α-Glucosidase-IN-25
α-Glucosidase-IN-25 (Compound (R)-8k) serves as a competitive inhibitor for α-glucosidase, demonstrating an inhibitory concentration 50 (IC50) of 1.19μM, making it applicable in anti-diabetic research [1].
价 格：￥电议型 号：T79259产 地：中国大陆
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T79240DNA gyrase B-IN-2；化合物 DNA gyrase B-IN-2DNA gyrase B-IN-2
DNA gyrase B-IN-2 (Compound E), a 2-aminobenzothiazole derivative, serves as a potent inhibitor of DNA gyrase B with substantial efficacy against ESKAPE pathogens. The compound exhibits potent nanomolar-range inhibition (IC 50 < 10 nM) and a broad-spectrum antibacterial effect, with minimum inhibitory concentrations below 0.03 μg/mL for most Gram-positive species and between 4–16 μg/mL for Gram-negative species including E. coli, Acinetobacter baumannii, Pseudomonas aeruginosa, and Klebsiella pn
价 格：￥电议型 号：T79240产 地：中国大陆
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T79237α-Glucosidase-IN-27；化合物 α-Glucosidase-IN-27α-Glucosidase-IN-27
α-Glucosidase-IN-27 (compound 8l), an α-glucosidase inhibitor with an IC50 value of 25.78 μM, demonstrates potential for research into type 2 diabetes (D2M) [1].
价 格：￥电议型 号：T79237产 地：中国大陆
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T79222JAK-IN-29；化合物 JAK-IN-29JAK-IN-29
JAK-IN-29 (Compound 3) is a potent inhibitor of Janus kinases (JAK) [1].
价 格：￥电议型 号：T79222产 地：中国大陆
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T79217RSV L-protein-IN-2；化合物 RSV L-protein-IN-2RSV L-protein-IN-2
RSV L-protein-IN-2 (Compound A), a noncompetitive inhibitor of the RSV polymerase (IC50: 4.5 μM), exhibits antiviral activity against long RSV strains (EC50: 1.3 μM) [1].
价 格：￥电议型 号：T79217产 地：中国大陆
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T79210PIKfyve-IN-2；化合物 PIKfyve-IN-2PIKfyve-IN-2
PIKfyve-IN-2 is a potent inhibitor of the PIKfyve kinase, with potential applications in cancer and autoimmune disorder research [1].
价 格：￥电议型 号：T79210产 地：中国大陆
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T79185STAT6-IN-2；化合物 STAT6-IN-2STAT6-IN-2
STAT6-IN-2 (Comp R-84) serves as a STAT6 inhibitor, effectively reducing the secretion of the chemokine eotaxin-3, which is known to induce eosinophil infiltration. This compound is useful in the study of immune diseases [1].
价 格：￥电议型 号：T79185产 地：中国大陆
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T79169CDK7-IN-22；化合物 CDK7-IN-22CDK7-IN-22
CDK7-IN-22 (compound 101) is a selective CDK7 inhibitor that exhibits antitumor activity, demonstrating specificity for CDK7 [1].
价 格：￥电议型 号：T79169产 地：中国大陆
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T79163RET-IN-24；化合物 RET-IN-24RET-IN-24
RET-IN-24 (Compound 26) is a selective inhibitor of RET tyrosine kinase, demonstrating antitumor activity [1].
价 格：￥电议型 号：T79163产 地：中国大陆
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T79145CK1-IN-2；化合物 CK1-IN-2CK1-IN-2
CK1-IN-2 (compound Nr.4) is a potent inhibitor of CK1, exhibiting IC50 values of 123 nM for CK1a, 19.8 nM for CK1d, 26.8 nM for CK1e, and 74.3 nM for p38a [1].
价 格：￥电议型 号：T79145产 地：中国大陆
