T31204Darapladib-impurityDarapladib impurity,Darapladibimpurity

Darapladib-impurity is the impurity of Darapladib. Darapladib inhibits lipoprotein-associated phospholipase A2 (Lp-PLA2)

价 格：￥电议型 号：T31204产 地：中国大陆

T15018CUDC-427

CUDC-427 is an orally bioactive and pan antagonist of inhibitor of apoptosis proteins(IAPs). CUDC-427 can be used in research on cancers.

价 格：￥电议型 号：T15018产 地：中国大陆

TP1559LZiconotide Acetate (107452-89-1 free base)analgesic,non-opioid,Ziconotide Acetate (107452891 free

Ziconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.

价 格：￥电议型 号：TP1559L产 地：中国大陆

T8439Clobenpropit dihydrobromideApoptosis,inhibit,Clobenpropit dihydrobromide,histamine H3R,antagonist,in

Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)

价 格：￥电议型 号：T8439产 地：中国大陆

T15641K777

K777 is a potent, orally active and irreversible inhibitor of cysteine protease. K777 is a potent CYP3A4 inhibitor (IC50= 60 nM). K777 is also a selective CCR4 antagonist featuring the potent chemotaxis inhibition. K777 irreversibly inhibits Cruzain, which is the major cysteine protease of Trypansoma cruzi, and cathepsins B and L. K777 targets cathepsin-mediated cell entry and wxibits a broad-spectrum antiviral activity. K777 inhibits EBOV and SARS-CoV pseudovirus entry with IC50 values of 0.87

价 格：￥电议型 号：T15641产 地：中国大陆

T8331NUN82647NUN82647,Inhibitor,NUN 82647,inhibit,Apoptosis,QBS,NUN-82647

NUN82647 is an Inhibitor of cell cycle at G2 phase, and apoptosis inducer.

价 格：￥电议型 号：T8331产 地：中国大陆

T27371FR-167356

FR-167356 is a specific inhibitor of a3 isoform vacuolar type H?-ATPase with IC50s of 170 nM, 370 nM and 220 nM for osteoclast plasma membranes, renal brush border membranes and macrophage microsomes. FR-167356 reduces bone metastasis of B16-F10 cells.

价 格：￥电议型 号：T27371产 地：中国大陆

T16940STAT5-IN-2STAT-5-IN-2,STAT5IN2,STAT5 IN 2

STAT5-IN-2 is an inhibitor of STAT5 with antileukemic effects (EC50s: 9 μM and 5 μM in K562 and KU812 cells, respectively).

价 格：￥电议型 号：T16940产 地：中国大陆

TN12955-O-Caffeoylshikimic acidinhibit,5 O Caffeoylshikimic acid,Inhibitor,5OCaffeoylshikimic acid

5-O-Caffeoylshikimic acid shows anti-oxidative activity; it also shows anti-inflammatory activity, the underlying mechanism was associated with downregulation of nuclear factor-κB.

价 格：￥电议型 号：TN1295产 地：中国大陆

PDK04236-METHYL-1H-INDOLE-2-CARBOXYLIC ACID6METHYL1HINDOLE2CARBOXYLICACID

价 格：￥电议型 号：PDK0423产 地：中国大陆

TP1881L1Pep 2-8 ammonium salt(1541011-97-5 free base)Pep 2 8 ammonium salt(1541011 97 5 free base),Pep 28 am

Pep 2-8 ammonium salt is Proprotein convertase subtilisin/kexin type 9 (PCSK9) inhibitor. Potent inhibitor of PCSK9 binding to LDL receptor (IC50 = 0.8 μM). Restores LDL uptake in HepG2 cells treated with PCSK9.

价 格：￥电议型 号：TP1881L1产 地：中国大陆

T22849ICI 199,441 hydrochlorideICI 199,441 hydrochloride

ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.

价 格：￥电议型 号：T22849产 地：中国大陆

TQ0150LevcromakalimPotassium Channel,KcsA,Inhibitor,inhibit,BRL38227,BRL-38227,Levcromakalim

Levcromakalim is an activator of the ATP-sensitive K+ channel.

价 格：￥电议型 号：TQ0150产 地：中国大陆

TN12373-O-Methylgallic acidAnthocyanin,3 O Methylgallic acid,inhibit,3OMethylgallic acid,metabolite,anti-c

3,4-Dihydroxy-5-methoxybenzoic acid reduces cell proliferation in Caco-2 cells(IC50 = 24.1 μM) more effectively than anthocyanins and may offer protection against colon cancer after its formation in the gut. 3,4-Dihydroxy-5-methoxybenzoic acid inhibits transcription factors NF-κB, AP-1, STAT-1, and OCT-1 which are known to be activated in colorectal cancer.

价 格：￥电议型 号：TN1237产 地：中国大陆

T11023DHODH-IN-14DHODH IN 14,DHODHIN14

DHODH-IN-14 is an analog of hydroxyfuran pyrimidine A771726. DHODH-IN-14 is a dihydroorotate dehydrogenase (DHODH) inhibitor IC50 0.49 μM mouse liver DHODH. DHODH-IN-14 can be used for rheumatoid arthritis.

价 格：￥电议型 号：T11023产 地：中国大陆

TP1789LMalantide acetate(86555-35-3 free base)Malantide acetate(86555 35 3 free base),Malantide acetate(865

Malantide acetate is a dodecapeptide phosphorylated by cyclic AMP-dependent protein kinase (PKA), and increases PKA activity.Malantide is a synthetic peptide that is phosphorylated by PKA and is used to measure PKA activity in vitro.

价 格：￥电议型 号：TP1789L产 地：中国大陆

T16536Pimonidazole hydrochlorideinhibit,Pimonidazole hydrochloride,Pimonidazole,Inhibitor

Pimonidazole hydrochloride accumulates in hypoxic cells via covalent binding with macromolecules or by forming reductive metabolites after the reduction of its nitro group. It can be used for qualitative and quantitative assessment of tumor hypoxia. Pimonidazole hydrochloride is a novel hypoxia marker for the complementary study of tumor hypoxia and cell proliferation in tumors.

价 格：￥电议型 号：T16536产 地：中国大陆

TN1438beta-Amyrin acetateHMG-CoA,betaAmyrin acetate,LDL,Fungal,inhibit,Inhibitor,arthritic,hemolysis,antif

beta-Amyrin acetate inhibits HMG-CoA Reductase (HMGCR) and sEH activity with IC50 of 3.4 μM. beta-Amyrin acetate has anti-inflammatory, antifungal, antioxidant, and anti-hyperlipidemic activities.

价 格：￥电议型 号：TN1438产 地：中国大陆

T23128PD180970PD-180970,PD180970

PD180970 is an inhibitor of Bcr-Abl with IC50s of 5 nM, 0.8 nM and 50 nM for the autophosphorylation of p210Bcr-Abl, Src and Kit. PD180970 can be used in studies about chronic myelogenous leukemia.

价 格：￥电议型 号：T23128产 地：中国大陆

TN4871PyrolinPyrolin

Pyrolin has a strong antifungal activity and exerts a potent impact on the ultrastructure of M.fructicola.

价 格：￥电议型 号：TN4871产 地：中国大陆