T6131PimasertibN-[(2S)-2,3-二羟基丙基]-3-[(2-氟-4-碘苯基)氨基]-4-吡啶甲酰胺；MSC1936369B；AS703026；SAR 245509

Pimasertib is an orally bioavailable small-molecule inhibitor of MEK1 and MEK2 (MEK1/2) with potential antineoplastic activity.

价 格：￥电议型 号：T6131产 地：中国大陆

T6121TepotinibMSC2156119；EMD-1214063；特泊替尼

Tepotinib is an inhibitor of MET tyrosine kinase with potential antineoplastic activity.

价 格：￥电议型 号：T6121产 地：中国大陆

T6119SotuletinibBLZ945

BLZ945 is an orally active, effective and specific CSF-1R inhibitor (IC50: 1 nM), >1000-fold selective against its closest receptor tyrosine kinase homologs.

价 格：￥电议型 号：T6119产 地：中国大陆

T6117TivantinibARQ 197

Tivantinib is an orally bioavailable small molecule inhibitor of c-Met with potential antineoplastic activity.

价 格：￥电议型 号：T6117产 地：中国大陆

T6111Selisistat司来司他；EX-527；SEN0014196

EX 527 is an effective and specific SIRT1 inhibitor (IC50: 38 nM) and shows >200-fold selectivity against SIRT2/3.

价 格：￥电议型 号：T6111产 地：中国大陆

T6108Ki16425Debio 0719

Ki16425 is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.

价 格：￥电议型 号：T6108产 地：中国大陆

T6087AZD 6482KIN 193；AZD6482

AZD 6482 is a potent and selective p110β inhibitor with IC50 of 0.69 nM and a PI3Kβ inhibitor with IC50 of 10 nM.

价 格：￥电议型 号：T6087产 地：中国大陆

T6070ON-01910N-[2-甲氧基-5-[[[2-(2,4,6-三甲氧基苯基)乙烯基]磺酰]甲基]苯基]甘氨酸钠盐

ON-01910 is a non-ATP-competitive PLK1 inhibitor(IC50 of 9 nM, in a cell-free assay). It shows 30-fold greater selectivity against Plk2 and no activity to Plk3. Rigosertib inhibits PI3K/Akt pathway and activates oxidative stress signals. Rigosertib induce

价 格：￥电议型 号：T6070产 地：中国大陆

T6067PD 123319(S)-(+)-PD 123319；PD123319

PD 123319 is a potent, selective AT2 angiotensin II receptor antagonist.

价 格：￥电议型 号：T6067产 地：中国大陆

T6025Danoprevir丹诺普韦；R7227；ITMN-191；RO5190591；RG7227

Danoprevir is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).

价 格：￥电议型 号：T6025产 地：中国大陆

T6019Volasertib伏拉塞替；BI 6727

Volasertib (BI-6727) is a potent inhibitor of PLK1 (IC50: 0.87 nM), inducing mitotic arrest and apoptosis. It also inhibits PLK2/PLK3 (IC50s: 5/56 nM).

价 格：￥电议型 号：T6019产 地：中国大陆

T6018Zosuquidar trihydrochloride唑喹达三盐酸盐；RS 33295-198 (D06387) 3HCl；Zosuquidar (LY335979) 3HCl；LY-335979 t

Zosuquidar (LY335979) is a potent modulator of P-glycoprotein-mediated multi-drug resistance with Ki of 60 nM. Phase 3.

价 格：￥电议型 号：T6018产 地：中国大陆

T5S2195Sibiricose A5西伯利亚远志糖A5

Sibiricose A5 is a lactate dehydrogenase inhibitor, it displays antidepressant-like, and antioxidant actions. Sibiricose A5 can protect PC12 cells damage induced by P. tenuifolia.

价 格：￥电议型 号：T5S2195产 地：中国大陆

T5S2102LeonurineSCM-198；益母草碱；盐酸益母草碱

Leonurine is an alkaloid that has been found in H. leonuri and with anti-oxidative and anti-inflammatory.

价 格：￥电议型 号：T5S2102产 地：中国大陆

T5S1989ApiinApioside；芹菜苷

1. Apiin is the reducing and stabilizing agent. 2. Apiin has inhibitory activity in-vitro on iNOS expression and nitrite production when added before LPS stimulation in the medium of J774.A1 cells.

价 格：￥电议型 号：T5S1989产 地：中国大陆

T5S1988Isorhamnetin-3-O-glucosideIsorhamnetin-3-O-beta-D-Glucoside；异鼠李素-3-O-葡萄糖苷

Isorhamnetin-3-O-glucoside inhibits the activity of alpha-glucosidase from rat intestine; it exhibits a potent rat lens aldose reductase (RLAR) inhibition in vitro, its IC(50) being 1.4 microM and has inhibitory effects of sorbitol accumulation, suggests

价 格：￥电议型 号：T5S1988产 地：中国大陆

T5S1982Periplocin杠柳毒苷；Periplocoside

1. Periplocin has anti-cancer effects on lung cancer cells, induces apoptosis and inhibits growth of cancer cells by the beta-catenin/Tcf signaling pathway. 2. Periplocin is used for treatment of rheumatoid arthritis, reinforcement of bones and tendons, p

价 格：￥电议型 号：T5S1982产 地：中国大陆

T5S1981alpha-Cyperoneα-香附酮；α-Cyperone；(+)-α-Cyperone

1. Alpha-Cyperone is a promising inhibitor of Hla production by S. aureus and protects lung cells from this bacterium. 2. Alpha-Cyperone significantly inhibited PGE2 production by suppressing the LPS-induced expression of inducible COX-2 at both the mRNA

价 格：￥电议型 号：T5S1981产 地：中国大陆

T5S1963Orcinol gentiobioside苔黑酚龙胆二糖苷；Anacardoside

价 格：￥电议型 号：T5S1963产 地：中国大陆

T5S1959(-)-Asarinin细辛脂素；Sesamin；Asarinin；Fagarol；Episesamin；Pseudocubebin；Eleutheroside B4

1. (-)-Asarinin shows antibacterial activity.

价 格：￥电议型 号：T5S1959产 地：中国大陆