T6425BTZ043 RacemateBenzothiazinone10526038,inhibit,Benzothiazinone-10526038,BTZ043 Racemate,BTZ 10526038

BTZ043 racemate is a decaprenylphosphoryl-β-D-ribose 2´-epimerase (DprE1) inhibitor, used as a new antimycobacterial agent.

价 格：￥电议型 号：T6425产 地：中国大陆

T10960Darbufelone

Darbufelone is a non-competitive dual inhibitor of PGF2α and LTB4. Dabfilon effectively inhibits PGHS-2 with a Ki of 10 μM and IC50s of 0.19 μM and 20 μM for PGHS-2 and PGHS-1.

价 格：￥电议型 号：T10960产 地：中国大陆

T74564-Ethyloctanoic acid4-Ethyloctanoic acid,4Ethyloctanoic acid,inhibit,4 Ethyloctanoic acid,Inhibitor

4-Ethyloctanoic acid is a natural product isolated from Saussurea lappa Clarke,acts as food additive,Industrial perfume,and so on.

价 格：￥电议型 号：T7456产 地：中国大陆

T6951Pramipexole dihydrochloride hydratetransient,Pramipexole dihydrochloride,Pramipexole dihydrochloride

Pramipexole Dihydrochloride is the hydrochloride salt of pramipexole, a benzothiazole derivative. As a nonergot dopamine agonist, pramipexole binds to D2 and D3 dopamine receptors in the striatum and substantia nigra of the brain.

价 格：￥电议型 号：T6951产 地：中国大陆

TN1576Diallyl disulfidecholesterol biosynthesis,squalene monooxygenase,Inhibitor,inhibit,Diallyl disulfide

Diallyl disulfide has antitumor effect, the effect can be enhanced by miR-200b and miR-22.

价 格：￥电议型 号：TN1576产 地：中国大陆

TPL03664-Biphenylcarboxylic acid4 Biphenylcarboxylic acid,4Biphenylcarboxylic acid

价 格：￥电议型 号：TPL0366产 地：中国大陆

T6717Vanillininhibit,Vanillin,Inhibitor,Endogenous Metabolite

Vanillin is a single molecule extracted from vanilla beans and also a popular odor used widely in perfume, food and medicine.Vanillin can reversibly and non-competitively inhibit the cellulase activity at appropriate concentrations and the value of IC50 was estimated to be 30 g/L.Vanillin protects KSC from UVB irradiation and its effects may occur through the suppression of downstream step of MDM2 in UVB irradiation-induced p53 activation. Vanillin also inhibits yeast growth and fermentation.

价 格：￥电议型 号：T6717产 地：中国大陆

T9678ML328ML328,ML-328

ML328 is a potent and selective inhibitor of bacterial AddAB(IC50 = 1.0 μM) and RecBCD(IC50 = 4.8 μM) helicase-nucleases.

价 格：￥电议型 号：T9678产 地：中国大陆

T21861Drinabant

Drinabant is an orally active CB1 receptor antagonist. Drinabant inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R.

价 格：￥电议型 号：T21861产 地：中国大陆

T28036MI-2-2cell proliferation,inhibit,menin-MLL interaction,Epigenetic Reader Domain,Inhibitor,Hoxa9 expr

MI-2-2 is an inhibitor of bivalent protein-protein interaction between menin and MLL with an IC50 of 46 nM. MI-2-2 binds to menin with Kd of 22 nM.

价 格：￥电议型 号：T28036产 地：中国大陆

T39707AS-1763AS1763,AS 1763

AS-1763 is an orally available and selective BTK inhibitor with an IC50 of 0.85 nM.

价 格：￥电议型 号：T39707产 地：中国大陆

T8606n-acetylciprofloxacinnacetylciprofloxacin,n acetylciprofloxacin

n-acetylciprofloxacin is inhibitor of H37Rv.

价 格：￥电议型 号：T8606产 地：中国大陆

TN6775AcetylcytisineAcetylcytisine

Acetylcytisine is a natural product of The herbs of Genista tinctoria L.

价 格：￥电议型 号：TN6775产 地：中国大陆

T7846Aegelineαsyn,Aegeline,yeast,Inhibitor,protein,Sec22p,inhibit,toxicity,Fungal,SNARE

Aegeline is an alkaloidal-amide, isolated from the leaves of Aegle marmelos and have shown antihyperglycemic as well as antidyslipidemic activities in the validated animal models of type 2 diabetes mellitus.

价 格：￥电议型 号：T7846产 地：中国大陆

T8877BonaftonBonafton

Bonafton is an antiviral agent.

价 格：￥电议型 号：T8877产 地：中国大陆

T6940PHA-767491 hydrochloridePHA767491,PHA 767491,inhibit,CAY-10572,Cyclin dependent kinase,CDK,CAY 10572

PHA-767491 is an effective ATP-competitive dual Cdc7/CDK9 inhibitor (IC50: 10/34 nM). It has ~20-fold selectivity against GSK3-β and CDK1/2, 50-fold selectivity against CDK5 and MK2, 100-fold selectivity against CHK2 and PLK1.

价 格：￥电议型 号：T6940产 地：中国大陆

T7117Sapropterin dihydrochloride(6R)-BH4,Sapropterin,Inhibitor,inhibit,Sapropterin dihydrochloride

Sapropterin dihydrochloride is phenylalanine hydroxylase agonist that is approved for the treatment of BH4 responsive PKU.

价 格：￥电议型 号：T7117产 地：中国大陆

TN2260Taxifolin 7-O-rhamnosideInhibitor,Taxifolin 7Orhamnoside,Taxifolin 7 O rhamnoside,inhibit

Taxifolin 7-O-rhamnoside is a natural product from Hypericum japonicum.

价 格：￥电议型 号：TN2260产 地：中国大陆

T6S1572Sauchinoneantioxidant,LPS,Diastereomeric,TNF-α,iNOS,anti-inflammatory,lignan,COX-2,inhibit,Nuclear f

1. Sauchinone is a useful adjunctive treatment for bacterial infection. 2. Sauchinone, an active lignan found in Saururus chinensis, to regulate the activation of HSCs, to prevent liver fibrosis, and to inhibit oxidative stress in vivo and in vitro. 3. Sauchinone diminishes LPS-induced neutrophil activation and acute lung injury. 4. Sauchinone-induced HO-1 expression plays a key role in the vascular protective effects of Sauchinone in HUVEC. 5. Sauchinone protects skin keratinocytes through inhi

价 格：￥电议型 号：T6S1572产 地：中国大陆

T9295BLU-263BLU 263,BLU263

BLU-263 is an investigational, potent, and selective oral small molecule inhibitor of KIT with sub-nanomolar potency against D816V-mutant KIT.

价 格：￥电议型 号：T9295产 地：中国大陆