T9516BinodenosonMRE 0470,imaging,P1 receptor,stress,oxidative,WRC0470,neutrophil,inhibit,radiotracers,Bin

Binodenoson is a potent and selective A2A adenosine receptor agonist (KD=270 nM). Binodenoson is being developed as a short-acting coronary vasodilator as an adjunct to radiotracers for use in myocardial stress imaging[1].

价 格：￥电议型 号：T9516产 地：中国大陆

T12530PPTNPPTN

PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.

价 格：￥电议型 号：T12530产 地：中国大陆

TP2051LCTCE 9908 acetateCTCE 9908 acetate

CTCE 9908 acetate is an antagonist of CXCR4 and inhibits migration in CXCR4-expressing ovarian cancer cells.

价 格：￥电议型 号：TP2051L产 地：中国大陆

TN6708ETHYL 3,5-DIHYDROXYBENZOATEETHYL 3,5 DIHYDROXYBENZOATE,ETHYL 3,5DIHYDROXYBENZOATE

ETHYL 3,5-DIHYDROXYBENZOATE is a natural product. It inhibits human carbonic anhydrase 2.

价 格：￥电议型 号：TN6708产 地：中国大陆

T21818Pregnenolone CarbonitrileCYPs,Cytochrome P450,P4503A,orally,Pregnenolone Carbonitrile,Pregnenolone 1

Pregnenolone Carbonitrile is an activator of rodent-PXR and induces the expression of CYP3A.

价 格：￥电议型 号：T21818产 地：中国大陆

T8933JNJ-63576253 free baseJNJ 63576253 free base,resistant,TRC 253,JNJ63576253,TRC-253,CRPC,JNJ63576253

JNJ-63576253 is a potent and orally active full antagonist of androgen receptor (AR), with IC50s of 37 and 54 nM for F877L mutant AR and wild-type AR in LNCaP cells. JNJ-63576253 can be used for the research of castration-resistant prostate cancer (CRPC).

价 格：￥电议型 号：T8933产 地：中国大陆

T9352hydrocotarnineE3 ligating enzyme,IL-18,NLRP3,E1/E2/E3 Enzyme,hydrocotarnine,inflammasome activation,

hydrocotarnine?is an inhibitor of Cbl.

价 格：￥电议型 号：T9352产 地：中国大陆

Fr14145Compound Fr14145Compound Fr14145

价 格：￥电议型 号：Fr14145产 地：中国大陆

T8684SotorasibAMG 510,Ras,KRAS,covalent,Sotorasib,regression,mutation,Inhibitor,G12C,anti-tumour,inhibit,

AMG-510 is a selective and orally bioavailable KRAS G12C covalent inhibitor.

价 格：￥电议型 号：T8684产 地：中国大陆

T72722,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE2,3,5TRIFLUORO4(TRIFLUOROMETHYL)PYRIDINE,2,3,5 TRIFLUORO

价 格：￥电议型 号：T7272产 地：中国大陆

T12589PI3Kα/mTOR-IN-1PI3Kα/mTORIN1,PI3Kα/mTOR IN 1,PI-3Kα/mTOR-IN-1

PI3Kα/mTOR-IN-1 is a potent dual inhibitor of PI3Kα/mTOR. PI3Kα/mTOR-IN-1 shows an IC50 of 7 nM for PI3Kα in a cell assay, and Kis of 12.5 nM and 10.6 nM for mTOR and PI3Kα in a cell free assay , respectively.

价 格：￥电议型 号：T12589产 地：中国大陆

T6972RS-1RAD51,RS1,RS-1,inhibit,Inhibitor,RS 1,CRISPR/Cas9

RS-1 is a RAD51 activator. RS-1 also increases CRISPR/Cas9-mediated knock-in efficiencies.

价 格：￥电议型 号：T6972产 地：中国大陆

T61112SLF1081851

SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.

价 格：￥电议型 号：T61112产 地：中国大陆

T17005FPR Agonist 43FPR Agonist 43

FPR Agonist 43 is a dual agonist of formyl peptide receptor 1 and formyl peptide receptor 2 (FPR2)/ALX.

价 格：￥电议型 号：T17005产 地：中国大陆

Fr13755Compound Fr13755Compound Fr13755

价 格：￥电议型 号：Fr13755产 地：中国大陆

T9054RO6889678inhibit,Hepatitis B virus,coregulated protein,UDP-glucuronosyltransferase,HB capsid formati

RO6889678 is HBV inhibitor with a complex ADME profile.

价 格：￥电议型 号：T9054产 地：中国大陆

PDK0356Compound PDK0356Compound PDK0356

价 格：￥电议型 号：PDK0356产 地：中国大陆

T9075BDP-13176inhibit,BDP13176,BDP-13176,Inhibitor,BDP 13176

BDP-13176 is a potent?inhibitor of fascin 1(Kd?of 90 nM and an?IC50?of 240 nM). It has potential as an anti-metastatic agent

价 格：￥电议型 号：T9075产 地：中国大陆

T64375UNC?1021UNC?1021

UNC 1021 is a selective L3MBTL3 inhibitor (IC50 = 0.048 μM).

价 格：￥电议型 号：T64375产 地：中国大陆

T12513PNZ5PNZ5,PNZ-5

PNZ5 is a potent and isoxazole-based pan-BET inhibitor, with high selectivity and potency similar to the well-established (+)-JQ1, with a KD of 5.43 nM for BRD4(1).

价 格：￥电议型 号：T12513产 地：中国大陆