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T73118PI3K-IN-28；化合物 PI3K-IN-28PI3K-IN-28
PI3K-IN-28 is a potent PI3K inhibitor demonstrating high efficacy and lower toxicity in MCF-10a models. It exhibits half-maximal inhibitory concentration (IC50, μM) values of 5.8, 2.3, and 7.9. With a selectivity index (SI) of 39, PI3K-IN-28 emerges as a promising lead compound for the optimization of anticancer agents.
价 格：￥电议型 号：T73118产 地：中国大陆
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T73106EGFR-IN-29；化合物 EGFR-IN-29EGFR-IN-29
EGFR-IN-29 is a potent EGFR inhibitor.
价 格：￥电议型 号：T73106产 地：中国大陆
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T73105EGFR-IN-28；化合物 EGFR-IN-28EGFR-IN-28
EGFR-IN-28 is a potent EGFR inhibitor. EGFR-IN-28 has antitumor activity [1] .
价 格：￥电议型 号：T73105产 地：中国大陆
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T73104EGFR-IN-23；化合物 EGFR-IN-23EGFR-IN-23
EGFR-IN-23, identified as compound 8 in WO2021244502A1, is a potent EGFR tyrosine kinase inhibitor (TKI) demonstrating an inhibitory concentration (IC50) of 8.05 nM against the BaF3/EGFR-DEL19/T790M/C797S cell line.
价 格：￥电议型 号：T73104产 地：中国大陆
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T73103EGFR-IN-21；化合物 EGFR-IN-21EGFR-IN-21
EGFR-IN-21, a potent EGFR inhibitor, exhibits an IC50 of 0.38 nM, demonstrating significant antitumor activity.
价 格：￥电议型 号：T73103产 地：中国大陆
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T73101EGFR-IN-25；化合物 EGFR-IN-25EGFR-IN-25
EGFR-IN-25, an efficacious EGFR inhibitor, demonstrates IC50 values of 9 nM for BaF3 cells (EGFR DEL19/T790M/C797S) and 60 nM for A431 cells (WT), respectively.
价 格：￥电议型 号：T73101产 地：中国大陆
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T73073PTP1B-IN-21；化合物 PTP1B-IN-21PTP1B-IN-21
PTP1B-IN-21 is a compound that functions as a selective inhibitor of protein tyrosine phosphatase 1B (PTP1B; IC50=1.56 μM), demonstrating a marked preference over the structurally similar T-cell protein tyrosine phosphatase (TCPTP; IC50>100 μM). This specificity highlights its potential as a critical agent for type 2 diabetes management.
价 格：￥电议型 号：T73073产 地：中国大陆
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T73072PTP1B-IN-20；化合物 PTP1B-IN-20PTP1B-IN-20
PTP1B-IN-20 is a selective PTP1B (protein tyrosine phosphatase 1B) inhibitor, exhibiting an IC50 of 1.05 μM, and demonstrates selectivity over TCPTP (T-cell protein tyrosine phosphatase), which has an IC50 of 78.0 μM. This compound targets a crucial enzyme for the inhibition of type 2 diabetes, distinguishing itself by its preferential action on PTP1B over the closely related TCPTP.
价 格：￥电议型 号：T73072产 地：中国大陆
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T73036hCA IX-IN-2；化合物 hCA IX-IN-2hCA IX-IN-2
hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative activity.
价 格：￥电议型 号：T73036产 地：中国大陆
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T73011HSP90-IN-20；化合物 HSP90-IN-20HSP90-IN-20
HSP90-IN-20, a potent inhibitor of HSP90, exhibits an IC50 of ≤10 μM, indicating its potential application in cancer research.
价 格：￥电议型 号：T73011产 地：中国大陆
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T73007PARP10-IN-2；化合物PARP10-IN-2PARP10-IN-2
PARP10-IN-2 is a potent inhibitor of PARP10, a mono-ADP-ribosyltransferase, with an IC50 value of 3.64 μM for human PARP10.PARP10-IN-2 also inhibited PARP2 and PARP15, with IC50 values of 27 μM and 11 μM, respectively.
价 格：￥电议型 号：T73007产 地：中国大陆
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T73003METTL3-IN-2；化合物 METTL3-IN-2METTL3-IN-2
METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.
价 格：￥电议型 号：T73003产 地：中国大陆
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T72985Masofaniten；化合物 MasofanitenAndrogen receptor-IN-2；Androgen receptor-IN-2
Masofaniten (Androgen receptor-IN-2), a potent, orally active inhibitor of the androgen receptor, demonstrates significant antitumor activity against prostate cancer.
价 格：￥电议型 号：T72985产 地：中国大陆
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T72983eeAChE-IN-2；化合物 eeAChE-IN-2eeAChE-IN-2
eeAChE-IN-2 is a potent inhibitor of eeAChE, exhibiting inhibitory potency with an IC50 of 2 nM.
价 格：￥电议型 号：T72983产 地：中国大陆
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T72894Clathrin-IN-2；化合物 Clathrin-IN-2Clathrin-IN-2
Clathrin-IN-2 is a potent inhibitor of clathrin-mediated endocytosis (CME), demonstrating an IC50 value of 2.3 μM. Additionally, it exhibits inhibitory effects on dynamin I GTPase, with an IC50 of 7.7 μM.
价 格：￥电议型 号：T72894产 地：中国大陆
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T72893AChE/MAO-IN-2；化合物 AChE/MAO-IN-2AChE/MAO-IN-2
Dual AChE-MAO B-IN-5, an indanone derivative, serves as an effective dual inhibitor for AChE and MAO-B, displaying IC50 values of 0.0224 μM for AChE, 0.0412 μM for MAO-B, and 0.1116 μM for MAO-A. Additionally, it exhibits antioxidant properties and inhibits β-amyloid plaque aggregation, making it suitable for Alzheimer’s disease (AD) research.
价 格：￥电议型 号：T72893产 地：中国大陆
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T72888YAP-TEAD-IN-2；化合物 YAP-TEAD-IN-2YAP-TEAD-IN-2
YAP-TEAD-IN-2 (compound 6) serves as a potent inhibitor of the YAP-TEAD protein-protein interaction (PPI), demonstrating an inhibitory concentration 50 (IC50) value of 2.7 nM [1].
价 格：￥电议型 号：T72888产 地：中国大陆
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T72886Akt1&PKA-IN-2；化合物 Akt1&PKA-IN-2Akt1&PKA-IN-2
Akt1&PKA-IN-2 ((R)-29), a compound with specificity towards PKB/AKT and notable selectivity for cyclin-dependent kinase 2 (CDK2), effectively inhibits AKT1, PKAa, and CDK2a with IC50 values of 0.007 ?M, 0.01 ?M, and 0.69 ?M, respectively.
价 格：￥电议型 号：T72886产 地：中国大陆
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T72880PI3K/AKT-IN-2；化合物 PI3K/AKT-IN-2PI3K/AKT-IN-2
PI3K/AKT-IN-2, a dual inhibitor of PI3K and AKT, prevents the epithelial-mesenchymal transition (EMT) and promotes apoptosis. Additionally, it impedes tubulin polymerization.
价 格：￥电议型 号：T72880产 地：中国大陆
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T72874sEH/AChE-IN-2；化合物 sEH/AChE-IN-2sEH/AChE-IN-2
sEH/AChE-IN-2 and acetylcholinesterase ( AChE ). sEH/AChE-IN-2 provides cumulative effects against neuroinflammation and memory impairment. sEH/AChE-IN-2 has the potential for the research of Alzheimer´s disease (AD) [1] .
价 格：￥电议型 号：T72874产 地：中国大陆
