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T15641K777；化合物K777APC-3316；APC-3316
K777 is a potent, orally active and irreversible inhibitor of cysteine protease. K777 is a potent CYP3A4 inhibitor (IC50= 60 nM). K777 is also a selective CCR4 antagonist featuring the potent chemotaxis inhibition. K777 irreversibly inhibits Cruzain, which is the major cysteine protease of Trypansoma cruzi, and cathepsins B and L. K777 targets cathepsin-mediated cell entry and wxibits a broad-spectrum antiviral activity. K777 inhibits EBOV and SARS-CoV pseudovirus entry with IC50 values of 0.87
价 格：￥电议型 号：T15641产 地：中国大陆
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T15640K134；化合物 T15640OPC33509；OPC33509
K134 is an inhibitor of phosphodiesterase 3. The IC50s of K134 for PDE3A, PDE3B, PDE5, PDE2 and PDE4 are 0.1, 0.28, 12.1, >300 and >300 μM, respectively.
价 格：￥电议型 号：T15640产 地：中国大陆
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T1562Rebamipide；瑞巴派特Proamipide|||OPC12759；Proamipide|||OPC12759|||瑞巴派特
Rebamipide (OPC12759) is a quinolinone derivative with anti-ulcer and anti-inflammatory activities. Rebamipide induces cyclooxygenase 2 (COX2) synthesis which results in an increase in endogenous prostaglandin synthesis in the gastric mucosa. This agent also inhibits H. pylori-induced production of tumor necrosis factor (TNF) alpha and subsequent inflammation of the gastric mucosa. In addition, rebamipide scavenges oxygen-derived free radicals that potentially cause mucosal injury, and stimulate
价 格：￥电议型 号：T1562产 地：中国大陆
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T15190L(S,R,S)-AHPC-PEG4-NH2；化合物T15190LVHL Ligand-Linker Conjugates 4|||E3 ligase Ligand-Linker Conjugates
(S,R,S)-AHPC-PEG4-NH2 (VHL Ligand-Linker Conjugates 4) is a synthetic E3 ligase ligand-linker conjugate comprising a VHL ligand based on (S,R,S)-AHPC and a 4-unit PEG linker.
价 格：￥电议型 号：T15190L产 地：中国大陆
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T15190(S,R,S)-AHPC-PEG4-NH2 hydrochloride；化合物 T15190E3 ligase Ligand-Linker Conjugates 7|||VH032-PEG4-NH2
(S, R, S)-AHPC-PEG4-NH2 hydrochloride is a chemically synthesized conjugate consisting of an E3 ligase ligand-linker, incorporating the VHL ligand based on (S, R, S)-AHPC, and a 4-unit PEG linker, which are specifically designed for use in PROTAC technology.
价 格：￥电议型 号：T15190产 地：中国大陆
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T15163DPC-681；化合物 T15163DPH-153893；DPH-153893
DPC-681 is a potent and selective HIV protease inhibitor (IC90s: 4 to 40 nM for wild-type HIV-1).
价 格：￥电议型 号：T15163产 地：中国大陆
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T15142Vebufloxacin；化合物 T15142OPC7241|||Flumenique|||DM8966；OPC7241|||Flumenique|||DM8966
Vebufloxacin (OPC-7251) shows potent antibacterial activity against gram-positive and -negative bacteria, including Staphylococcus aureus and Pseudomonas aeruginosa. It has potent activity characteristically against Propionibacterium acnes.
价 格：￥电议型 号：T15142产 地：中国大陆
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T15012Crolibulin；化合物CrolibulinEPC2407；EPC2407
Crolibulin (EPC2407) is an inhibitor of small molecule tubulin polymerization.
价 格：￥电议型 号：T15012产 地：中国大陆
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T1466Nadifloxacin；那氟沙星OPC7251；OPC7251|||那氟沙星
Nadifloxacin (OPC7251) has been used in trials studying the treatment of Acne Vulgaris.
价 格：￥电议型 号：T1466产 地：中国大陆
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T1447Fenclonine芬克洛宁Fenchlonine|||PCPA|||CP-10188|||芬克洛宁|||4-Chloro-DL-phenylalanine|||DL-4-Chlorophenylal
Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin (5-HYDROXYTRYPTAMINE). Fenclonine(CP-10188) acts pharmacologically to deplete endogenous levels of serotonin.
价 格：￥电议型 号：T1447产 地：中国大陆
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T13877(S,S,S)-AHPC hydrochloride(S,S,S)-AHPC盐酸盐(S,S,S)-VH032-NH2 hydrochloride|||(S,S,S)-AHPC盐酸盐
(S,S,S)-AHPC hydrochloride ((S,S,S)-VH032-NH2 hydrochloride) is a VHL amino building block, is a ligand used as a negative control for (S,R,S)-AHPC. It is the VH032-based VHL ligand used in the recruitment of the VHL protein.
价 格：￥电议型 号：T13877产 地：中国大陆
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T13876(S,R,S)-AHPC-propargyl；化合物 T13876(S,R,S) AHPC propargyl|||VHL ligand 7|||AHPC-propargyl|||VH032-prop
(S,R,S)-AHPC-propargyl is a VHL ligand which is used in "click reaction" for PROTACs.
价 格：￥电议型 号：T13876产 地：中国大陆
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T13813PCSK9 ligand 1；化合物 T13813PCSK9 ligand 1
PCSK9 ligand 1 is a small molecule ligand for proprotein convertase substilisin-like/kexin type 9 (PCSK9) and shows high affinity to PCSK9(Ki of 107 nM).
价 格：￥电议型 号：T13813产 地：中国大陆
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T13812PCA50941；化合物 T13812PCA50941
PCA50941 is a 1,4-dihydropyridine derivative, treatment for cardiovascular disease.
价 格：￥电议型 号：T13812产 地：中国大陆
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T13804OPC-28326；化合物OPC-28326OPC-28326
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of 2040, 285, and 55?nM, respectively.
价 格：￥电议型 号：T13804产 地：中国大陆
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T13671L(S,R,S)-AHPC-Me dihydrochloride；化合物 T13671LVHL ligand 2 dihydrochloride|||E3 ligase Ligand 1 dihydro
(S,R,S)-AHPC-Me dihydrochloride, also known as VHL ligand 2 dihydrochloride, is a chemical compound utilized in the synthesis of ARV-771. ARV-771, a BET PROTAC degrader relying on von Hippel-Landau (VHL) E3 ligase, demonstrates potent degradation of BET protein in castration-resistant prostate cancer (CRPC) cells, with a DC50 of less than 1 nM. This compound serves as the VHL ligand, specifically the (S,R,S)-AHPC-based VHL ligand, that facilitates the recruitment of von Hippel-Lindau (VHL) prote
价 格：￥电议型 号：T13671L产 地：中国大陆
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T13671(S,R,S)-AHPC-Me hydrochloride；化合物(S,R,S)-AHPC-Me hydrochlorideVHL ligand 2 hydrochloride|||E3 ligase
(S,R,S)-AHPC-Me hydrochloride (VHL ligand 2 hydrochloride) is a chemical compound utilized in the synthesis of ARV-771, an exceptionally potent BET protein degrader. This compound selectively degrades BET protein in cells resistant to castration, exhibiting a remarkable DC50 <1 nM. Recognized as VHL ligand 2 hydrochloride, (S,R,S)-AHPC-Me hydrochloride serves as the VHL ligand derived from (S,R,S)-AHPC for the recruitment of von Hippel-Lindau (VHL) protein.
价 格：￥电议型 号：T13671产 地：中国大陆
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T13547LAMP-PCP disodium；AMP-PCP钠盐AMP-PCP disodium
AMP-PCP disodium is an ATP analogue with binding affinity to the N-terminal domain of Hsp90, with a Kd value of 3.8 μM. The binding of AMP-PCP disodium contributes to the formation of an active homodimer of Hsp90.
价 格：￥电议型 号：T13547L产 地：中国大陆
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T13547AMP-PCP；化合物 T13547AMP-PCP
AMP-PCP is an ATP analog and can bind to the Hsp90 N-terminal domain (Kd: 3.8 μM). AMP-PCP binding favors the formation of the active homodimer of Hsp90.
价 格：￥电议型 号：T13547产 地：中国大陆
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T13423L(1S,2R)-2-PCCA；化合物(1S,2R)-2-PCCA(1S,2R)-2-PCCA（Iso-1609563-71-4）；(1S,2R)-2-PCCA（Iso-1609563-71-4）
(1S,2R)-2-PCCA is a novel and potent small molecule GPR88 receptor agonist with an EC50 value of 3 nM in the non-cellular system and 603 nM in the cellular system.
价 格：￥电议型 号：T13423L产 地：中国大陆
