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T4046BX517；化合物BX517PDK1 inhibitor 2|||BX 517|||BX-517；PDK1 inhibitor 2|||BX 517|||BX-517
BX517 (PDK1 inhibitor 2) is a potent and selective inhibitor of PDK1.
价 格：￥电议型 号：T4046产 地：中国大陆
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T40290CDK12-IN-5；CDK12-IN-5CDK12-IN-5；CDK12-IN-5
CDK12-IN-5 is a pyrazolotriazine compound that effectively inhibits CDK12, with an IC50 value of 23.9 nM at a high ATP concentration of 2 mM. However, CDK12-IN-5 does not exhibit inhibitory effects on CDK2/Cyclin E (IC50 = 173 μM) and CDK9/Cyclin T1 (IC50 = 127 μM) at the same high ATP concentration of 2 mM, as stated in WO2021116178A1.
价 格：￥电议型 号：T40290产 地：中国大陆
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T40289CDK12-IN-6CDK12-IN-6CDK12-IN-6
CDK12-IN-6, a pyrazolotriazine compound, is a powerful inhibitor of CDK12. Its inhibitory activity is significant with an IC50 value of 1.19 μM when tested at high ATP concentration (2 mM). Notably, CDK12-IN-6 does not exhibit any inhibitory effect on CDK2/Cyclin E (IC50 >20 μM) and CDK9/Cyclin T1 (IC50 >20 μM) when tested under the same high ATP conditions (2 mM) (WO2021116178A1).
价 格：￥电议型 号：T40289产 地：中国大陆
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T40288CDK12-IN-4CDK12-IN-4CDK12-IN-4
CDK12-IN-4, a pyrazolotriazine compound, exhibits potent inhibition of CDK12 by achieving an IC50 value of 0.641 μM, utilizing high ATP levels (2 mM). Notably, CDK12-IN-4 does not impact CDK2/Cyclin E (IC50 > 20 μM) or CDK9/Cyclin T1 (IC50 > 20 μM) under the influence of high ATP (2 mM) levels (WO2021116178A1).
价 格：￥电议型 号：T40288产 地：中国大陆
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T39752CDK12-IN-2；化合物CDK12-IN-2CDK12 inhibitor 2|||CDK12-IN-2；CDK12 inhibitor 2|||CDK12-IN-2
CDK12-IN-2 (CDK12 inhibitor 2) is an effective and selective inhibitor of CDK12 with an IC50 of 52 nM, >100 μM, >10 μM and 16 μM for CDK12, CDK2, CDK7, and CDK9. CDK12-IN-2 can be used in studies about the function of CDK12.
价 格：￥电议型 号：T39752产 地：中国大陆
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T31540DK-1-166；化合物 T31540DK1-166|||DK 1-166|||DK-1166；DK1-166|||DK 1-166|||DK-1166
DK-1-166 is a inducer of apoptotic cell death in TNBC cell lines without causing cytotoxicity in the normal mammary epithelial cell line.
价 格：￥电议型 号：T31540产 地：中国大陆
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T31539DK-1-150；化合物 T31539DK-1150|||DK 1-150|||DK1-150|||DK 1 150；DK-1150|||DK 1-150|||DK1-150|||DK 1 150
DK-1-150 is an inducer of apoptotic cell death in TNBC cell lines without causing cytotoxicity in the normal mammary epithelial cell line.
价 格：￥电议型 号：T31539产 地：中国大陆
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T24741RS1-PDK1 inhibitor；RS1-PDK1抑制剂RS-1|||RS1|||RS 1；RS-1|||RS1|||RS 1
RS1-PDK1 inhibitor (RS 1) is a selective inhibitor of the protein kinase PDK1 that can be used to treat and prevent disease or disorders.
价 格：￥电议型 号：T24741产 地：中国大陆
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T16450PDK1-IN-RS2；化合物 T16450PDK1-IN-RS2
PDK1-IN-RS2 inhibits the activation of the downstream kinases S6K1 by PDK1. PDK1-IN-RS2 is a mimic of the peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor (Kd: 9 μM).
价 格：￥电议型 号：T16450产 地：中国大陆
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T14990CDK12-IN-3；化合物 T14990CDK12-IN-3
CDK12-IN-3 is a selective CDK12 inhibitor (IC50: 491 nM in an enzymatic assay).
价 格：￥电议型 号：T14990产 地：中国大陆
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T14915CDK12-IN-E9；化合物 T14915CDK12-IN-E9
CDK12-IN-E9 is a potent and selective covalent CDK12 inhibitor and non-covalent CDK9 inhibitor while avoiding ABC transporter-mediated efflux. It has a weak binding ability to CDK7/CyclinH complex (IC50> 1 μM).
价 格：￥电议型 号：T14915产 地：中国大陆
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T14914Cdk1/2 Inhibitor III；Cdk1/2 抑制剂IIICdk1/2 Inhibitor III
Cdk1/2 Inhibitor III is a selective Cdk1/2 inhibitor with an IC50 value of 2.1 μM against CDK1/cyclin B.
价 格：￥电议型 号：T14914产 地：中国大陆
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T12398MP7；PDK1 抑制剂PDK1 inhibitor；PDK1 抑制剂|||PDK1 inhibitor
MP7 (PDK1 inhibitor) is a inhibitor of phosphoinositide-dependent kinase-1 (PDK1).
价 格：￥电议型 号：T12398产 地：中国大陆
