T7017WNK463Ser/Thr Protease,WNK 463,inhibit,WNK463,Serine proteases,Inhibitor,Serine endopeptidases,Threo

WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).

价 格：￥电议型 号：T7017产 地：中国大陆

T6476Dofetilidecardiovascular,potent,specific,class,antiarrhythmic,orally,Inhibitor,UK68789,UK-68789,Dofe

Dofetilide is a sulfonamide class III antiarrhythmic agent and potassium channel blocker. Dofetilide selectively blocks cardiac ion channels of the rapid component of the delayed rectifier potassium current Ikr. This antiarrhythmic agent prolongs cardiac action potential duration and effective refractory period due to delayed repolarization without affecting conduction velocity. This results in a normal sinus rhythm. Dofetilide is used in the treatment of atrial fibrillation and flutter.

价 格：￥电议型 号：T6476产 地：中国大陆

TN1417Azadirachtinpest,inhibit,cytoskeleton,cellular,transduction,signal,insecticides,Apoptosis,Azadiracht

Azadirachtin has antifungal activity, used as an insecticide.

价 格：￥电议型 号：TN1417产 地：中国大陆

T6S1010Allomatrinealkaloid,antinociceptive,κ-opioid,Allomatrine,receptors,inhibit,(+)-Allomatrine,Inhibitor

Allomatrine is a natural product from Sophora alopecuroides L. Allomatrine, when given i.c.v., may stimulate the descending dynorphinergic neuron, resulting in the stimulation of KORs in the spinal cord.

价 格：￥电议型 号：T6S1010产 地：中国大陆

T8458CNQX disodiumIonotropic glutamate receptors,inhibit,Inhibitor,startle,non-NMDA,fear-potentiated,kain

CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.

价 格：￥电议型 号：T8458产 地：中国大陆

T8402Regorafenib HydrochlorideRaf,PDGFR,Raf kinases,inhibit,Inhibitor,RET,Regorafenib Hydrochloride,Vascu

Regorafenib Hydrochloride is a new oral multikinase inhibitor of angiogenic, stromal and oncogenic receptor tyrosine kinases with potent preclinical antitumor activity

价 格：￥电议型 号：T8402产 地：中国大陆

T8418DCLK1-IN-1DCLK1 IN 1,signaling,PDAC,KRAS,cancer,low,ERK,Inhibitor,selective,DCLK1IN1,inhibit,DCLK-1-

DCLK1-IN-1 is a selective and in vivo-compatible chemical probe of the DCLK1 kinase domain .

价 格：￥电议型 号：T8418产 地：中国大陆

TP1606LNLS PKKKRKV acetate(95088-49-6 free base)NLS PKKKRKV acetate(95088 49 6 free base),NLS PKKKRKV ace

NLS PKKKRKV acetate is a peptide derived from the 40 tumor antigen of the great ape virus (SV40 big T antigen), which is a method to enhance the nuclear portal in the research field of gene transfer.

价 格：￥电议型 号：TP1606L产 地：中国大陆

T7703PK11007PK11007,inhibit,MDM-2/p53,Reactive Oxygen Species,Inhibitor,PK 11007,PK-11007

PK11007 is an anti-p53 drug.

价 格：￥电议型 号：T7703产 地：中国大陆

T9040Aurora kinase inhibitor-2inhibit,Aurora-A,Aurora kinase inhibitor2,Aurora Kinase,ATP-competitive,Aur

Aurora Kinase Inhibitor II is a cell-permeable anilinoquinazoline that inhibit the activity of Aurora A (IC50 = 0.39 M).

价 格：￥电议型 号：T9040产 地：中国大陆

T9031MCU-i4C2C12,Inhibitor,mitochondrial,MCU-i-4,Mitochondrial Metabolism,MCU-i4,MCUi4,Ca2+,uptake,inhibi

MCU-i4 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.

价 格：￥电议型 号：T9031产 地：中国大陆

T9177BPAM344Ionotropic glutamate receptors,GluK3a,PAM,iGluR,BPAM344,BPAM 344,Inhibitor,BPAM-344,KAR,GluK1

BPAM344 is a potent positive allosteric modulator (PAM) of the KAR subunits GluK1b, GluK2a, and GluK3a.

价 格：￥电议型 号：T9177产 地：中国大陆

TN71207-keto-deoxycholic acid

7-keto-deoxycholic acid is converted from Lactobacillus and Bifidobacterium with specific condition and from cholic acid in vitro.

价 格：￥电议型 号：TN7120产 地：中国大陆

TN1012LFebrifugine dihydrochlorideInhibitor,Parasite,Febrifugine dihydrochloride,antimalarial,alkaloid,Quin

Febrifugine dihydrochloride is a biochemical with therapeutic activity regarding malaria, cancer, fibrosis and inflammatory diseases.

价 格：￥电议型 号：TN1012L产 地：中国大陆

PDK0380CarbazoleCarbazole

价 格：￥电议型 号：PDK0380产 地：中国大陆

TP1018LUrechistachykinin II acetateUrechistachykinin II acetate

Urechistachykinin II acetate is an invertebrate rapid kinin-related peptide (TRPs) isolated from carotenoid worms, shows antimicrobial activities without a hemolytic effect

价 格：￥电议型 号：TP1018L产 地：中国大陆

T7123AMG-47aInhibitor,signal,kinases,AMG 47a,JAK,Janus kinase,AMG-47a,transduction,Src,VEGFR,cytoplamic,p

AMG-47a is a potent inhibitor of Lck and T cell proliferation. AMG-47a could promote the degradation of the KRAS oncoprotein. AMG-47a selectively reduced the levels of EGFP-KRASG12V protein but did not affect EGFP protein in cells.

价 格：￥电议型 号：T7123产 地：中国大陆

T4074GSK-872translocation,GSK-872,neurological,HMGB1,Receptor-interacting protein kinases,brain,GSK 872,c

GSK872 (GSK2399872A) is an effective and specific RIP3 kinase inhibitor. It binds RIP3 kinase domain with high affinity (IC50: 1.8 nM) and inhibits kinase activity (IC50: 1.3 nM).

价 格：￥电议型 号：T4074产 地：中国大陆

T8118BekanamycinBekanamycin,Gram-negative,inhibit,influx,action,Antibiotic,calcium,Inhibitor,presynaptic,

Bekanamycin is an aminoglycoside antibiotic.

价 格：￥电议型 号：T8118产 地：中国大陆

T6118NVP-HSP990HSP-990,NVP-HSP990,Apoptosis,Heat shock proteins,NVP HSP990,HSP,NVP-HSP-990,HSP 990,Inhibi

NVP-HSP990 (HSP990) is an effective and specific HSP90α/β inhibitor (IC50: 0.6 /0.8 nM).

价 格：￥电议型 号：T6118产 地：中国大陆