TN2079(-)-Pinoresinol()Pinoresinol,( ) Pinoresinol

(-)-Pinoresinol is isolated from the whole plant of Serissa japonica (Thunb.) Thunb.

价 格：￥电议型 号：TN2079产 地：中国大陆

T60146USP8-IN-1USP8inhibitor

USP8-IN-1 is an inhibitor of USP8 with an IC 50 of 1.9 μM. USP8-IN-1 inhibits H1975 cell growth with a GI 50 of 82.04 μM [1].

价 格：￥电议型 号：T60146产 地：中国大陆

TN2100PratenseinInhibitor,Nuclear factor-kappaB,Nuclear factor-κB,cognitive,inhibit,BDNF,synapse,Pratensei

Pratensein as a novel transcriptional up-regulator of scavenger receptor class B type I in HepG2 cells.

价 格：￥电议型 号：TN2100产 地：中国大陆

TP1882L1Orphanin FQ(1-11) acetate(178249-41-7 free base)Orphanin FQ(1 11) acetate(178249 41 7 free base),Orp

Peptide fragment containing amino acids 1-11 of Nociceptin. Potent agonist of the ORL1/KOR-3 receptor (Ki = 55 nM); displays no affinity for opioid receptors, including μ, δ, κ1 and κ3 receptors (Ki >1000 nM). Displays analgesic properties in CD-1 mice.

价 格：￥电议型 号：TP1882L1产 地：中国大陆

T60032BRM/BRG1 ATP Inhibitor-2Epigenetic Reader Domain,Inhibitor,BRM/BRG1 ATP Inhibitor 2,inhibit,BRM/BRG1

BRM/BRG1 ATP Inhibitor-2 is an inhibitor of BRG1/BRM ATPase and can be used in studies about the treatment of BAF-related disorders.

价 格：￥电议型 号：T60032产 地：中国大陆

T8595Practololreceptor,inhibit,arrhythmias,β1-adrenergic,Practolol,Beta Receptor,Adrenergic Receptor,card

Practolol is a selective β-adrenoceptor blocker.

价 格：￥电议型 号：T8595产 地：中国大陆

T8796CAN508inhibit,CAN 508,ATP-competitive,Cyclin dependent kinase,esophageal,cells,CDK,CAN508,Inhibitor,

CAN508 is a potent, ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 μM. It is also a competitive inhibitor of Cdk2-cyclin E with respect to ATP, with Ki and IC50 values of 13.3 and 20 μM, respectively.CAN508 exhibits a 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes. Antitumor activity.

价 格：￥电议型 号：T8796产 地：中国大陆

TQ0283RS102895CC chemokine receptor,CCR,Inhibitor,RS102895,inhibit,RS-102895,RS 102895

RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.

价 格：￥电议型 号：TQ0283产 地：中国大陆

T9041AES-350Histone deacetylases,AES 350,MV4-11,AES-350,Apoptosis,acute myeloid leukemia,AML,Inhibitor,in

AES-350 is a potent and orally active HDAC6 inhibitor(IC50 and a Ki of 0.0244 μM and 0.035 μM, respectively). It is also against HDAC-3, -8, and -11 in an enzymatic activity assay with IC50 values of 0.187 μM, 0.245 μM, and >1μM, respectively. AES-350 triggers apoptosis in AML cells through HDAC inhibition and can be used for acute myeloid leukemia (AML) research.

价 格：￥电议型 号：T9041产 地：中国大陆

T6908NSC 228155Epidermal growth factor receptor,Histone Acetyltransferase,EGFR,HER1,HATs,inhibit,Inhibito

NSC228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and modulate EGFR tyrosine phosphorylation.

价 格：￥电议型 号：T6908产 地：中国大陆

T6924Riviciclib hydrochlorideinhibit,Inhibitor,Riviciclib,CDK,Riviciclib hydrochloride,Cyclin dependent k

P276-00 is a novel CDK1, CDK4 and CDK9 inhibitor with IC50 of 79 nM, 63 nM and 20 nM, respectively. Phase 2/3.

价 格：￥电议型 号：T6924产 地：中国大陆

T8084Dimethyl 4-hydroxyisophthalateDimethyl 4-hydroxyisophthalate,inhibit,Dimethyl 4 hydroxyisophthalate,

Dimetghyl 4-Hydroxyisophthalate is a methyl salicylate analogue, used as a building block in the chemical synthesis.

价 格：￥电议型 号：T8084产 地：中国大陆

T6767TCS7010Aurora Kinase,inhibit,TCS 7010,Apoptosis,TCS-7010,TCS7010,Inhibitor

Aurora A Inhibitor I is a novel, potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM in a cell-free assay. It is 1000-fold more selective for Aurora A than Aurora B.

价 格：￥电议型 号：T6767产 地：中国大陆

Fr14055Compound Fr14055Compound Fr14055

价 格：￥电议型 号：Fr14055产 地：中国大陆

T6443Chloroprocaine hydrochlorideinhibit,Na,K-ATPase,Sodium potassium pump,Chloroprocaine,anesthetic,2-Ch

Chloroprocaine HCl is a local anesthetic during surgical procedures.

价 格：￥电议型 号：T6443产 地：中国大陆

T7596FirocoxibLPS,COX-2,fever,ML1785713,Cyclooxygenase,COX,inhibit,Firocoxib,Inhibitor,anti-inflammatory,

Firocoxib is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 μM), with anti-inflammatory for use in dogs and horses.

价 格：￥电议型 号：T7596产 地：中国大陆

TP1545L1FFAGLDD amine saltFFAGLDD amine salt

FFAGLDD amine salt is MMP9 selective cleavage peptides, which used for cytosolic delivery of Doxorubi-cin (DOX) and achieve temporally and spatially controlled slow drug delivery and release.

价 格：￥电议型 号：TP1545L1产 地：中国大陆

T8222SelpercatinibFVB/NRj mice,RET (WT),inhibit,Inhibitor,RET (G810R),LOXO 292,LOXO292,RET (V804M),Selper

Selpercatinib is a tyrosine kinase inhibitor with antineoplastic properties(IC50 of 14.0 nM, 24.1 nM, and 530.7 nM for RET (WT), RET (V804M) , and RET (G810R), respectively)

价 格：￥电议型 号：T8222产 地：中国大陆

Fr13877Compound Fr13877Compound Fr13877

价 格：￥电议型 号：Fr13877产 地：中国大陆

TN6982Diethyl phthalate

Diethyl phthalate is a endocrine disrupter affecting the apoptotic system in PC12 cells. Diethyl phthalate is widely used in many plastics and personal care products.

价 格：￥电议型 号：TN6982产 地：中国大陆