T6885MarimastatTA-2516,Marimastat,inhibit,Inhibitor,BB 2516,BB-2516,TA 2516,Matrix metalloproteinases,MMP

Marimastat (BB-2516) is a potent, broad spectrum matrix metalloprotease (MMP) inhibitor. MMP-9 (IC50=3 nM), MMP-1 (IC50=5 nM), MMP-2 (IC50=6 nM), MMP-14 (IC50=9 nM)and MMP-7 (IC50=13 nM).

价 格：￥电议型 号：T6885产 地：中国大陆

T9808Tetradecylthioacetic acidPeroxisome proliferator-activated receptors,β-Oxidation,inhibit,fatty acid

Tetradecylthioacetic acid is a synthetic fatty acid with a sulfur substitution in the β-position. This modification renders TTA unable to undergo complete β-oxidation and increases its biological activity, including activation of peroxisome proliferator activated receptors (PPARs) with preference for PPARα.

价 格：￥电议型 号：T9808产 地：中国大陆

TP1563Gap19myocardial,Gap19,cytoplasmic,Cx40/pannexin-1,inhibit,Gap Junction Protein,C-terminus,Gap 19,hem

Gap19 is a peptide that corresponds to a sequence on the cytoplasmic loop (CL) of Cx43.

价 格：￥电议型 号：TP1563产 地：中国大陆

TN2069PicrocrocinInhibitor,Picrocrocin,antiproliferative,SKMEL-2,Apoptosis,malignant,melanoma,cells,human,

Picrocrocin is a natural product

价 格：￥电议型 号：TN2069产 地：中国大陆

T8596Ceefourin 1P-glycoprotein,chemosensitizers,inhibit,efflux,protein,resistance,Ceefourin 1,Ceefourin1,

Ceefourin 1 is a highly selective multidrug resistance protein 4 (MRP4) inhibitor.

价 格：￥电议型 号：T8596产 地：中国大陆

T6815HS-1371HS-1371,Inhibitor,Receptor-interacting protein kinases,RIPK,inhibit,HS 1371,RIP kinase,HS1371

HS-1371 is a novel kinase inhibitor of receptor-interacting protein kinase 3 (RIP3) with an IC50 of 20.8 nM.

价 格：￥电议型 号：T6815产 地：中国大陆

T9228Propionylpromazine hydrochloridePropiopromazine,Propionylpromazine,DRD2,Dopamine Receptor,Parkinson,

Propionylpromazine hydrochloride is a dopamine receptor D2 (DRD2) antagonist.

价 格：￥电议型 号：T9228产 地：中国大陆

TJS0328Nordalberginpromyelocytic,Inhibitor,coumarin,HL-60,cells,leukemia,differentiation,Nordalbergin,inhib

价 格：￥电议型 号：TJS0328产 地：中国大陆

T17881(S,R,S)-AHPC-C10-NH2PROTAC,(S,R,S) AHPC C10 NH2,Inhibitor,(S,R,S)AHPCC10NH2,E3 Ligase Ligand-Linker

(S,R,S)-AHPC-C10-NH2 is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker used for BET-Targeted PROTAC.

价 格：￥电议型 号：T17881产 地：中国大陆

T8217Enzalutamide carboxylic acidprostate,Enzalutamide carboxylic acid,metastatic,MDV3100 carboxylic acid

Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .

价 格：￥电议型 号：T8217产 地：中国大陆

T6883SamotolisibInhibitor,mTOR,LY-3023414,Phosphoinositide 3-kinase,DNA-dependent protein kinase,inhibit,

LY3023414 is an oral ATP competitive inhibitor of the class I PI3K isoforms, DNA-PK, and mTOR. LY3023414 has been used in trials studying the treatment of Neoplasm, Solid Tumor, COLON CANCER, BREAST CANCER, and Advanced Cancer, among others.

价 格：￥电议型 号：T6883产 地：中国大陆

TN1637EurycomalactoneDNA double-strand,Eurycomalactone,NF-κB,protein synthesis,Inhibitor,Nuclear factor-ka

Eurycomalactone is a natural product isolated from Eurycoma longifolia Jack., acts as a potent NF-κB inhibitor( IC50 of 0.5 μM). Eurycomalactone inhibits protein synthesis, depletes cyclin D1, but does not affect TNFα-induced degradation of IκBα or the phosphorylation of IKKα/β and IκBα.

价 格：￥电议型 号：TN1637产 地：中国大陆

TN6737(25R)-Spirost-4-ene-3,12-dionenatural product,neutrophil,mast cells,histamine,Inhibitor,(25R)Spirost

(25R)-Spirost-4-ene-3,12-dione is a natural product.

价 格：￥电议型 号：TN6737产 地：中国大陆

T8505SC-236SC-236,gastric,PPAR,cancer,ischemia,Liver,inhibit,allodynia,Inhibitor,fibrogenesis,neuroprotec

Sc 236 is an orally active and selective inhibitor of COX-2 (IC50 of 0.005 μM and 17.8 μM for COX-2 and COX-1, respectively).

价 格：￥电议型 号：T8505产 地：中国大陆

TP1053LProtein Kinase C 19-31 acetateProtein Kinase C 19 31 acetate,Protein Kinase C 1931 acetate

Protein Kinase C 19-31 acetate, a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate peptide for testing the protein kinase C activity.

价 格：￥电议型 号：TP1053L产 地：中国大陆

TN1968N-?Feruloyloctopaminecarcinoma,N-?Feruloyloctopamine,inhibit,Protein kinase B,MAPK,PKB,Inhibitor,Hep

N-Feruloyloctopamine is a natural product.

价 格：￥电议型 号：TN1968产 地：中国大陆

T7395LanifibranorInhibitor,IVA 337,Lanifibranor,inhibit,PPAR,Peroxisome proliferator-activated receptors,

Lanifibranor is an agonist of peroxisome proliferator-activated receptors (PPARs) with EC50 values of 1,537, 866, and 206 nM for human recombinant PPARα, PPARβ, and PPARγ, respectively, for transactivation activity

价 格：￥电议型 号：T7395产 地：中国大陆

T1986Atopaxarplatelets,Atopaxar,receptor-1,signaling,PAR-1,inhibit,E-5555,Inhibitor,receptor,Protease Act

Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute Coronary Syndrome.

价 格：￥电议型 号：T1986产 地：中国大陆

T7353RSV604virus,Respiratory syncytial virus,A 60444,respiratory,protein,inhibit,RSV,syncytial,A-60444,In

RSV-604 is an inhibitor of respiratory syncytial virus (RSV) that binds to RSV nucleoprotein (Kd = 1.31 μM)

价 格：￥电议型 号：T7353产 地：中国大陆

TQ0067GSK484 hydrochlorideGSK484 hydrochloride,GSK 484,Protein Arginine Deiminase,GSK-484,GSK-484 hydrochl

GSK484 hydrochloride (GTPL8577) is a specifc and reversible peptidyl arginine deiminase 4 (PAD4) inhibitor. It demonstrates high-affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium.

价 格：￥电议型 号：TQ0067产 地：中国大陆