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T69598Isoproterenol-d7 HCl；化合物 Isoproterenol-d7 HClIsoproterenol-d7 HCl
Isoproterenol-d7 is intended for use as an internal standard for the quantification of isoproterenol by GC- or LC-MS. Isoproterenol is an agonist of β1- and β2-adrenergic receptors (β1- and β2-ARs; Kis = 224 and 458 nM, respectively). It is selective for β1- and β2-ARs over β3-ARs (Ki = 1,570 nM). Isoproterenol inhibits contractions in isolated field-stimulated rat vas deferens (EC50 = 45.6 nM). In vivo, isoproterenol (0.33 mg/kg) decreases blood pressure and increases water intake in nephrectom
价 格：￥电议型 号：T69598产 地：中国大陆
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T69597Befiperide HCl；化合物 Befiperide HClBefiperide HCl
Befiperide, also known as DU-29325, is a substituted piperazine that has agonist activity at serotonin1 receptors.
价 格：￥电议型 号：T69597产 地：中国大陆
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T69579Dothiepin HCl；化合物 Dothiepin HClDothiepin HCl
Dothiepin HCl is a Tricyclic antidepressant (TCA), acting as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also having other activities including antihistamine, antiadrenergic, antiserotonergic, anticholinergic, and sodium channel-blocking effects.
价 格：￥电议型 号：T69579产 地：中国大陆
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T6957PRT-060318；化合物PRT-060318P142-76|||PRT318|||PRT-060318 2HCl；P142-76|||PRT318|||PRT-060318 2HCl
PRT-060318 (P142-76) is a novel selective inhibitor of the Syk tyrosine kinase, as an approach to HIT treatment.
价 格：￥电议型 号：T6957产 地：中国大陆
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T69557ABI-231 HCl；化合物 ABI-231 HClABI-231 HCl
ABI-231 is a potent, orally bioavailable tubulin inhibitor that interacts with the colchicine binding site and is currently undergoing clinical trials for prostate cancer. ABI-231, has an average IC50 = 5.2 nM against panels of melanoma and prostate cancer cell lines, is orally bioavailable, and strongly suppress melanoma tumors in vivo. ABI-231 holds great promise as a new generation of orally available tubulin inhibitor.
价 格：￥电议型 号：T69557产 地：中国大陆
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T6955Propafenone hydrochloride；盐酸普罗帕酮Propafenone HCl|||Arythmol|||SA-79 (hydrochloride)|||Rytmonorm|||Ryt
Propafenone hydrochloride (Arythmol8) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial and ventricular arrhythmias.
价 格：￥电议型 号：T6955产 地：中国大陆
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T69549Ethybenztropine HCl；化合物 Ethybenztropine HClEthybenztropine HCl
Ethybenztropine HCl is an anticholinergic which is used as an antiparkinsonian agent. Ethybenztropine may also act as a dopamine reuptake inhibitor.
价 格：￥电议型 号：T69549产 地：中国大陆
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T69537Difelikefalin HCl；化合物 Difelikefalin HClDifelikefalin HCl
Difelikefalin HCl is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin HCl is selective for KOR over the μ-opioid receptor (MOR; EC50 = >1 ?M in a transactivation assay). It reduces acetic acid-induced writhing, as well as scratching behavior induced by the KOR antagonist GNTI, in mice (ED50s = 0.07
价 格：￥电议型 号：T69537产 地：中国大陆
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T69517Bexotegrast HCl；化合物 Bexotegrast HClBexotegrast HCl
Bexotegrast, also known as PLN-74809, is a small-molecule, dual selective inhibitor of αVβ1 / αVβ6 for idiopathic pulmonary fibrosis (IPF) and primary sclerosing cholangitis (PSC). These integrins cause upstream activation of TGF-β1 in actively fibrotic tissue. Inhibition of these integrins will block TGF-β1 activation, thereby preventing the growth of fibrotic tissue within the lung and bile ducts.
价 格：￥电议型 号：T69517产 地：中国大陆
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T6951Pramipexole dihydrochloride hydrate普拉克索盐酸盐水合物Pramipexole 2HCl Monohydrate|||普拉克索盐酸盐水合物|||Mirapex|||普
Pramipexole dihydrochloride hydrate (Mirapex) is the hydrochloride salt of pramipexole, a benzothiazole derivative. As a nonergot dopamine agonist, pramipexole binds to D2 and D3 dopamine receptors in the striatum and substantia nigra of the brain.
价 格：￥电议型 号：T6951产 地：中国大陆
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T69498DBPR112 HCl；化合物 DBPR112 HClDBPR112 HCl
DBPR112 is a potent EGFR inhibitor (IC50=487 nM) as a Clinical Candidate for the Treatment of Non-Small Cell Lung Cancer. DBPR112), DBPR112not only displayed a potent inhibitory activity against EGFRL858R/T790M double mutations but also exhibited tenfold potency better than the third-generation inhibitor, osimertinib,against EGFR and HER2 exon 20 insertion mutations. Overall, pharmacokinetic improvement through lead-to-candidateoptimization yielded fourfold oral AUC better that afatinib along wi
价 格：￥电议型 号：T69498产 地：中国大陆
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T69493Berubicin HCl；化合物 Berubicin HClBerubicin HCl
Berubicin hydrochloride is the hydrochloride salt of the anthracycline derivative berubicin with potential antineoplastic activity. Berubicin intercalates into DNA and interrupts topoisomerase II activity, resulting in the inhibition of DNA replication and repair, and RNA and protein synthesis. Unlike other anthracycline derivatives, this agent crosses the blood-brain barrier (BBB).
价 格：￥电议型 号：T69493产 地：中国大陆
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T69429Y27632 HCl hydrate；化合物 Y27632 HCl hydrateY27632 HCl hydrate
Y27632 is a selective ROCK inhibitor, which inhibits ET-1-induced increases in natriuretic peptide production, cell size, protein synthesis, and myofibrillar organization. Y27632 prevents dimethylnitrosamine-induced hepatic fibrosis in rats, increases apoptosis and disrupts the actin cortical mat in embryonic avian corneal epithelium, affects initial heart myofibrillogenesis in cultured chick blastoderm, promotes the proliferation and cell cycle progression of cultured astrocyte from spinal cord
价 格：￥电议型 号：T69429产 地：中国大陆
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T69422Flupirtine HCl；化合物 Flupirtine HClFlupirtine HCl
Flupirtine HCl is the salt form of Flupirtine, also known as W-2964, an aminopyridine that functions as a centrally acting non-opioid analgesic. It first became available in Europe in 1984, and is sold mainly under the names Katadolon, Trancolong, Awegal, Efiret, Trancopal Dolo, and Metanor. Like nefopam, it is unique among analgesics in that it is a non-opioid, non-NSAID, non-steroidal centrally acting analgesic. Flupirtine is a selective neuronal potassium channel opener that also has NMDA re
价 格：￥电议型 号：T69422产 地：中国大陆
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T6940PHA-767491 hydrochloride；化合物PHA767491 HClCAY10572|||PHA-767491|||PHA767491 HCl|||CAY-10572 hydrochlo
PHA-767491 hydrochloride (CAY-10572 hydrochloride) is an effective ATP-competitive dual Cdc7/CDK9 inhibitor (IC50: 10/34 nM). It has ~20-fold selectivity against GSK3-β and CDK1/2, 50-fold selectivity against CDK5 and MK2, 100-fold selectivity against CHK2 and PLK1.
价 格：￥电议型 号：T6940产 地：中国大陆
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T69355Butaclamol HCl；化合物 Butaclamol HClButaclamol HCl
Butaclamol, also known as AY-23,028, is a typical antipsychotic which was never marketed. Sold as the hydrochloride salt for use in research, the compound acts as a dopamine receptor antagonist.
价 格：￥电议型 号：T69355产 地：中国大陆
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T69354Enzastaurin 2HCl；化合物 Enzastaurin 2HClEnzastaurin 2HCl
Enzastaurin 2HCl, also known as DB-102 and LY317615, is a synthetic macrocyclic bisindolemaleimide with potential antineoplastic activity. Binding to the ATP-binding site, Enzastaurin 2HCl selectively inhibits protein kinase C beta, an enzyme involved in the induction of vascular endothelial growth factor (VEGF)-stimulated neo-angiogenesis. This agent may decrease tumor blood supply and so tumor burden.
价 格：￥电议型 号：T69354产 地：中国大陆
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T69350Ethionamide HCl；化合物 Ethionamide HClEthionamide HCl
Ethionamide HCl is the salt form of Ethionamide, a second-line antitubercular agent that inhibits mycolic acid synthesis. Ethionamide is a nicotinamide derivative, with antibacterial activity, used to treat tuberculosis. Although the exact mechanism of action of ethionamide is unknown, it may inhibit the synthesis of mycolic acid, a saturated fatty acid found in the bacterial cell wall, thereby inhibiting bacterial cell wall synthesis. This eventually leads to bacterial cell wall disruption and
价 格：￥电议型 号：T69350产 地：中国大陆
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T69318Tazolol HCl；化合物 Tazolol HClTazolol HCl
Tazolol HCl is a selective beta1-agonist, coronartherapeutic agent, and cardiotonic agent.
价 格：￥电议型 号：T69318产 地：中国大陆
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T6930Pazopanib Hydrochloride；盐酸帕唑帕尼GW786034|||Pazopanib HCl|||GW786034 HCl|||Votrient HCl|||Armala；GW7860
Pazopanib Hydrochloride (Votrient HCl) is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FGFR, c-Kit and c-Fms with IC50 of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM in cell-free assays, respectively.
价 格：￥电议型 号：T6930产 地：中国大陆
