您好，欢迎来到易推广！ 请登录 免费注册

上海陶术生物科技有限公司 主营产品：生物试剂,实验服务等

当前位置：易推广 > 上海陶术生物科技有限公司 > 产品展示

企业档案

会员类型：会员

已获得易推广信誉   等级评定
139成长值

(0 -40)基础信誉积累，可浏览访问

(41-90)良好信誉积累，可接洽商谈

(91+  )优质信誉积累，可持续信赖

易推广会员：5年

工商认证 【已认证】

最后认证时间：

注册号： 【已认证】

法人代表： 【已认证】

企业类型：生产商 【已认证】

注册资金：人民币万 【已认证】

产品数：86101

参观次数：3886442

手机网站：http://m.yituig.com/c135739/

旗舰版地址：http://tsbiochem.app17.com

自主品牌

自主品牌

已选条件

  • T72943eIF4A3-IN-17；化合物 eIF4A3-IN-17eIF4A3-IN-17

    eIF4A3-IN-17, a silvestrol analogue, disrupts the assembly of the eIF4F translation complex, exhibiting EC50 values of 0.9, 15, and 1.8 nM for myc-LUC, tub-LUC, and growth inhibition of MBA-MB-231 cells, respectively. This compound holds potential for research in human cancer pathogenesis [1].

    价 格：￥电议型 号：T72943产 地：中国大陆

  • T72931TRK/ALK-IN-1；化合物 TRK/ALK-IN-1TRK/ALK-IN-1

    TRK/ALK-IN-1 is a potent dual inhibitor of TRK and ALK, exhibiting good correlation between its enzymatic inhibition and anti-proliferative activities, with IC50 values of 2.2 nM for TRKA, 9.3 nM for ALK WT, and 38 nM for ALK L1196M. It holds potential for cancer research applications.

    价 格：￥电议型 号：T72931产 地：中国大陆

  • T72928CDK4/6-IN-15；化合物 CDK4/6-IN-15CDK4/6-IN-15

    CDK4/6-IN-15, an orally active and selective inhibitor of CDK4/6, effectively halts the growth of cancer cells by arresting the cell cycle at the G1 phase and inhibiting the phosphorylation of the retinoblastoma tumor suppressor protein (Rb) at S780, as well as suppressing E2 factor (E2F)-regulated gene expression.

    价 格：￥电议型 号：T72928产 地：中国大陆

  • T72924VEGFR-3-IN-1；VEGFR-3抑制剂1VEGFR-3-IN-1

    VEGFR-3-IN-1 is a novel potent and selective VEGFR3 inhibitor with an IC50 of 110.4 nM.VEGFR-3-IN-1 possesses antitumor activity, inactivates the VEGFR3 signaling pathway, and inhibits the proliferation and migration of VEGF-C-induced human dermal lymphatic endothelial cells (HDLEC), MDA-MB-231 and MDA-MB-436 cells. MB-436 cells and inhibited the proliferation and migration of human dermal lymphatic endothelial cells (HDLEC), MDA-MB-231 and MDA-MB-436 cells.

    价 格：￥电议型 号：T72924产 地：中国大陆

  • T72922TNKS1/2-IN-1；化合物 TNKS1/2-IN-1TNKS1/2-IN-1

    TNKS1/2-IN-1 is a potent inhibitor of tankyrase (TNKS1/2), exhibiting pIC50 values between 7.1-8.2. It is utilized in research targeting cancer, fibrosis, and other hyperproliferative diseases.

    价 格：￥电议型 号：T72922产 地：中国大陆

  • T72919PKCiota-IN-1；化合物 PKCiota-IN-1PKCiota-IN-1

    PKCiota-IN-1 is a potent inhibitor of PKCiota (PKC-ι), exhibiting an IC50 of 2.7 nM. Additionally, it displays inhibitory activity against PKC-α and PKC-ε, with IC50 values of 45 nM and 450 nM, respectively.

    价 格：￥电议型 号：T72919产 地：中国大陆

  • T72910APOBEC3G-IN-1；APOBEC3G 抑制剂1APOBEC3G-IN-1

    APOBEC3G-IN-1 (MN136.0185) is a targeted APOBEC3G inhibitor with anti-HIV activity for the study of infectious diseases and cancer.

    价 格：￥电议型 号：T72910产 地：中国大陆

  • T72892AChE/MAO-IN-1；化合物 AChE/MAO-IN-1AChE/MAO-IN-1

    AChE/MAO-IN-1 is a potent inhibitor of human acetylcholinesterase (AChE), monoamine oxidase A (MAO-A), and monoamine oxidase B (MAO-B), demonstrating inhibitory concentrations (IC50) of 0.0248 μM, 0.0409 μM, and 0.1108 μM against AChE, MAO-A, and MAO-B, respectively.

    价 格：￥电议型 号：T72892产 地：中国大陆

  • T72885Akt1&PKA-IN-1；化合物 Akt1&PKA-IN-1Akt1&PKA-IN-1

    Akt1&PKA-IN-1 is a potent dual inhibitor targeting Akt and PKA, exhibiting IC50 values of 0.11 μM for Akt, 0.03 μM for PKAα, and 9.8 μM for CDK2. Notably, it demonstrates selectivity for cyclin-dependent kinase 2 (CDK2).

    价 格：￥电议型 号：T72885产 地：中国大陆

  • T72877p53-HDM2-IN-1；化合物 p53-HDM2-IN-1p53-HDM2-IN-1

    p53-HDM2-IN-1 is a potent inhibitor of the p53-HDM2 protein-protein interaction, demonstrating an inhibitory concentration (IC 50) of 0.103 μM. This compound has significant applications in cancer research.

    价 格：￥电议型 号：T72877产 地：中国大陆

  • T72872HDAC/BET-IN-1；化合物 HDAC/BET-IN-1HDAC/BET-IN-1

    HDAC/BET-IN-1 is a chemical compound exhibiting submicromolar inhibitory activity against HDAC1 and HDAC6, with IC50 values of 0.163 μM and 0.067 μM, respectively, and against BRD4, with a Ki of 0.076 μM. Additionally, it possesses potent antileukemia activity.

    价 格：￥电议型 号：T72872产 地：中国大陆

  • T7285911β-HSD1-IN-10；化合物 11β-HSD1-IN-1011β-HSD1-IN-10

    11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 ?M for humans, is suitable for research into obesity, hyperglycemia, and cognitive impairment.

    价 格：￥电议型 号：T72859产 地：中国大陆

  • T72844EGFR/CDK2-IN-1；化合物 EGFR/CDK2-IN-1EGFR/CDK2-IN-1

    EGFR/CDK2-IN-1, an inhibitor of both EGFR and CDK2, demonstrates effective cytotoxicity towards MCF7 and HepG2 cells, suggesting its potential application in cancer research.

    价 格：￥电议型 号：T72844产 地：中国大陆

  • T72841PBRM1-BD2-IN-1；化合物 PBRM1-BD2-IN-1PBRM1-BD2-IN-1

    PBRM1-BD2-IN-1 is a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, displaying binding affinity and inhibitory efficacy with Kd and IC50 values of 0.7 μM and 0.2 μM, respectively. This compound is utilized in cancer research.

    价 格：￥电议型 号：T72841产 地：中国大陆

  • T72839SHP2/HDAC-IN-1；化合物 SHP2/HDAC-IN-1SHP2/HDAC-IN-1

    SHP2/HDAC-IN-1, a dual allosteric inhibitor targeting SHP2 and HDAC, exhibits potent inhibitory effects with IC 50 values of 20.4 nM (SHP2) and 25.3 nM (HDAC1), respectively. This compound activates T cells, enhances antigen presentation, and promotes cytokine secretion, facilitating efficient antitumor immunity. It holds potential for cancer immunotherapy research.

    价 格：￥电议型 号：T72839产 地：中国大陆

  • T72836SHP2/CDK4-IN-1；化合物 SHP2/CDK4-IN-1SHP2/CDK4-IN-1

    SHP2/CDK4-IN-1 (compound 10) is a dual inhibitor targeting SHP2 and CDK4, exhibiting oral activity and high potency with IC50 values of 4.3 nM for SHP2 and 18.2 nM for CDK4. It effectively induces G0/G1 arrest, inhibiting the proliferation of TNBC cell lines, and demonstrates significant antitumor efficacy in the EMT6 syngeneic mouse model. This compound is valuable for research into triple-negative breast cancer (TNBC) [1].

    价 格：￥电议型 号：T72836产 地：中国大陆

  • T72832MDM2-p53-IN-16；化合物 MDM2-p53-IN-16MDM2-p53-IN-16

    MDM2-p53-IN-16 is a potent inhibitor of the MDM2-p53 complex, exhibiting an IC 50 value of 4.3 nM for the dissociation of the human p53/MDM2 complex. It effectively reactivates p53, leading to apoptosis and cell-cycle arrest in Glioblastoma Multiforme (GBM) cells, positioning it as a valuable agent for cancer research.

    价 格：￥电议型 号：T72832产 地：中国大陆

  • T72827Nrf2/HO-1-IN-1；化合物 Nrf2/HO-1-IN-1Nrf2/HO-1-IN-1

    Nrf2/HO-1-IN-1 is a potent Nrf2/HO-1 pathway inhibitor, with an IC 50 value of 0.38 μM for NO . Nrf2/HO-1-IN-1 can significantly reduce the level of ROS in cells. Nrf2/HO-1-IN-1 can be used for researching anti-inflammatory [1] .

    价 格：￥电议型 号：T72827产 地：中国大陆

  • T72824RAGE/SERT-IN-1；化合物 RAGE/SERT-IN-1RAGE/SERT-IN-1

    RAGE/SERT-IN-1 is a potent, orally active inhibitor of advanced glycation end products (RAGE) and serotonin transporter (SERT), with IC50 values of 8.26 μM and 31.09 nM, respectively. It demonstrates a significant neuroprotective effect against Aβ25-35-induced neuronal damage and alleviates depressive behavior in mice. RAGE/SERT-IN-1 is useful for research on the comorbidity of Alzheimer´s disease and depression [1].

    价 格：￥电议型 号：T72824产 地：中国大陆

  • T72815CBP/p300-IN-10；化合物 CBP/p300-IN-10CBP/p300-IN-10

    CBP/p300-IN-10, a potent inhibitor targeting histone acetyltransferase enzymes EP300 and CREBBP, exhibits IC50 values of 26 nM and 39 nM, respectively. This compound shows potential for anticancer research applications.

    价 格：￥电议型 号：T72815产 地：中国大陆

136373839404142434445101下一页共101页

展台首页| 公司简介| 供应产品| 产品目录| 公司动态| 荣誉证书| 招聘信息| 技术中心| 联系我们| 会员管理

易推广  设计制作，未经允许翻录必究.Copyright(C) 2009 http://www.yituig.com, All rights reserved.

以上信息由企业自行提供，信息内容的真实性、准确性和合法性由相关企业负责，易推广对此不承担任何责任.   总访问量：3886442

中国彩虹热线

快速导航

返回顶部
在线咨询

提交