Fr13587Compound Fr13587Compound Fr13587

7-Chloro-4-(piperazin-1-yl)quinolone is an important scaffold in medicinal chemistry. It exhibited either alone or as hybrid with other active pharmacophores diverse pharmacological profiles. 7-Chloro-4-(piperazin-1-yl)quinolone is a potent sirtuin inhibitor and also inhibits the serotonin uptake ( IC 50 of 50 μM). 7-Chloro-4-(piperazin-1-yl)quinolone exhibits antimalarial activity on D10 and K1 strains of P. falciparum with IC 50 s of 1.18 μM and 0.97 μM, respectively [1].

价 格：￥电议型 号：Fr13587产 地：中国大陆

T38387Compound C108Compound C108,Compound C-108

Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2). Compound C108 can be used in studies about breast tumors and esophageal squamous cell carcinoma.

价 格：￥电议型 号：T38387产 地：中国大陆

T90604Compound NB-48-0729Compound NB480729,Compound NB 48 0729

价 格：￥电议型 号：T90604产 地：中国大陆

PDK0035Compound PDK0035Compound PDK0035

价 格：￥电议型 号：PDK0035产 地：中国大陆

T9853STING activator Compound 53Inhibitor,HEK293T,STING agonist-12,MPYS,STING agonist12,STING,STING agoni

STING activator Compound 53 based on an oxindole core structure demonstrated robust on-target functional activation of STING (human EC50 185 nM) in immortalised and primary cells and a cytokine induction fingerprint consistent with STING activation.

价 格：￥电议型 号：T9853产 地：中国大陆

T8745Compound 23Inhibitor,Raf,A375,HT-29,Compound 23,inhibit,BRAF-V600E,ubiquitin-proteasome system,antic

Compound 23 selectively induces degradation of BRAF-V600E but not wildtype BRAF.

价 格：￥电议型 号：T8745产 地：中国大陆

T7958Methyl arachidateLTA4H,natural,Methyl arachidate,Aminopeptidase,inhibit,Inhibitor,compound,Methyl ei

Methyl Icosanoate is an esterified form of arachidic acid

价 格：￥电议型 号：T7958产 地：中国大陆

T6146Dorsomorphin dihydrochloride6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶；Dorsomorphin (Compound C) 2

Dorsomorphin is a potent, selective and ATP-competitive AMPK inhibitor (Ki: 109 nM) and does not exhibit significant activity on structurally related kinases.

价 格：￥电议型 号：T6146产 地：中国大陆

T4170PKM2-IN-1PKM2 inhibitor；compound 3k

PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.

价 格：￥电议型 号：T4170产 地：中国大陆

T3971CASINPirl1-related Compound 2

CASIN is a specific inhibitor of GTPase Cdc42 (IC50: 2 uM).

价 格：￥电议型 号：T3971产 地：中国大陆

T3964Glutaminase C-IN-1Compound 968；Glutaminase Inhibitor Compound 968

Glutaminase C-IN-1 is a Glutaminase C allosteric inhibitor.

价 格：￥电议型 号：T3964产 地：中国大陆

T3811Ginsenoside C-K20(S)-人参皂苷 C-K；人参皂苷 C-K；Ginsenoside compound K；Ginsenoside K

Ginsenoside C-K is a bacterial metabolite of G-Rb1 exhibiting anti-inflammatory effects by reducing iNOS and COX-2.

价 格：￥电议型 号：T3811产 地：中国大陆

T3587NOD-IN-1Compound 4

NOD-IN-1 is a potent mixed inhibitor of nucleotide-binding oligomerization domain (NOD)-like receptors.

价 格：￥电议型 号：T3587产 地：中国大陆

T3586Compound 4012-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one

Compound 401 is a synthetic DNA-PK inhibitor (IC50 = 0.28 μM) that also targets mTOR but not PI3K.

价 格：￥电议型 号：T3586产 地：中国大陆

T35398MINA53 inhibitor (Compound 10)

MINA53 inhibitor (Compound 10) is an inhibitor of MINA53.

价 格：￥电议型 号：T35398产 地：中国大陆

T28001MDK-6983Compound 6k；MDK 6983；Autophagy inhibitor 6k；MDK6983

MDK-6983 is a autophagy inhibitor. MDK-6983 disrupts the dynamics of actin cytoskeleton in human melanoma cells, affecting processes essential for the maintenance and expansion of tumours such as cell adhesion, motility, proliferation, vesicular transport

价 格：￥电议型 号：T28001产 地：中国大陆

T27635IsoxepacOlopatadine USP Related Compound C

Isoxepac is a non-steroidal anti-antiphlogistic agent and analgesic.

价 格：￥电议型 号：T27635产 地：中国大陆

T2503PAC-1PAC1；Procaspase activating compound 1

PAC-1 has been used in trials studying the treatment of Lymphoma, Melanoma, Solid Tumors, Breast Cancer, and Thoracic Cancers, among others.

价 格：￥电议型 号：T2503产 地：中国大陆

T226783,5-Bis(4-nitrophenoxy)benzoic acid3,5-二(4-硝基苯氧基)苯甲酸；Compound W

The compound is an inhibitor of γ-secretase. It also causes a decrease in the released levels of Aβ42 and notch-1 Aβ-like peptide 25 (Nβ25).

价 格：￥电议型 号：T22678产 地：中国大陆

T21000PiBPittsburgh Compound-B；6-OH-BTA-1；2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇

PiB is a standard for analysis of 11C-PiB. 11C-PiB is a β-amyloid PET imaging tracer for Alzheimer´s disease diagnosis.

价 格：￥电议型 号：T21000产 地：中国大陆