T12513PNZ5PNZ5,PNZ-5

PNZ5 is a potent and isoxazole-based pan-BET inhibitor, with high selectivity and potency similar to the well-established (+)-JQ1, with a KD of 5.43 nM for BRD4(1).

价 格：￥电议型 号：T12513产 地：中国大陆

T74735-Bromoindole5 Bromoindole,5Bromoindole

5-bromoindole is a potential inhibitor of glycogen synthase kinase 3 (GSK-3)and an important pharmaceutical chemical intermediate

价 格：￥电议型 号：T7473产 地：中国大陆

T6654SaponinsSaponins,Inhibitor,Fungal,inhibit,Bacterial

Sapogenins glycosides are a mixture of triterpene and steroid saponins isolated from medicinal plants such as Aesculus hippocastanum L., Hedera helix L. and Ruscus aculeatus L., which are claimed to be effective for the treatment/prevention of venous insufficiency.

价 格：￥电议型 号：T6654产 地：中国大陆

T7007UNC2025Inhibitor,inhibit,FLT3,leukemia,CD135,Fms like tyrosine kinase 3,acute,Cluster of differentia

UNC-2025（ IC50 of 0.74 nM and 0.8 nM） is a potent and orally bioavailable dual MER/FLT3 inhibitor. UNC-2025 is about 20-fold selectivity higher than Axl and Tyro3.

价 格：￥电议型 号：T7007产 地：中国大陆

T60148MSC-4106MSC4106

MSC-4106 is an orally active and potent inhibitor of YAP/TAZ-TEAD. MSC-4106 inhibits TEAD1 or TEAD3 auto-palmitoylation and exhibits inhibitory effect on NCI-H226 tumor xenograft model [1].

价 格：￥电议型 号：T60148产 地：中国大陆

TQ0059Ilorasertibanti-tumor,H1299,Platelet-derived growth factor receptor,Inhibitor,ABT 348,antiproliferat

Ilorasertib (ABT-348) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora A/Aurora B/Aurora C (IC50s: 120 nM/7 nM/1 nM). It also suppresses RET tyrosine kinase, PDGFRβ, and Flt1 (IC50s: 7 nM, 3 nM, and 32 nM).

价 格：￥电议型 号：TQ0059产 地：中国大陆

TN3849Dihydrodehydrodiconiferyl alcoholDihydrodehydrodiconiferyl alcohol

Dihydrodehydrodiconiferyl alcohol is the methanolic extract of Liriodendron tulipifera[1].

价 格：￥电议型 号：TN3849产 地：中国大陆

T9004TM2-115TM2 115,TM2115

TM2-115 is a inhibitor of malaria parasite histone methyltransferases that results in rapid and irreversible parasite death [1].

价 格：￥电议型 号：T9004产 地：中国大陆

TN6772Malabaricone Clipid metabolism,Inhibitor,sphingomyelin synthase,SMS 1,diet,obesity,inhibit,Malabaric

Malabaricone C is a bioactive chemical.

价 格：￥电议型 号：TN6772产 地：中国大陆

T11190EMT inhibitor-1EMT inhibitor1,EMT inhibitor 1

EMT inhibitor-1 is an inhibitor of Hippo, Wnt signaling and TGF- macrophages (TGF-) with antitumor activity.

价 格：￥电议型 号：T11190产 地：中国大陆

T6437CefoperazoneCefoperazone,inhibit,Inhibitor,Antibiotic,Bacterial

Cefoperazone binds to and inactivates penicillin-binding proteins (PBPs) located on the inner membrane of the bacterial cell wall. PBPs are enzymes involved in the terminal stages of assembling the bacterial cell wall and in reshaping the cell wall during growth and division. Inactivation of PBPs interferes with the cross-linkage of peptidoglycan chains necessary for bacterial cell wall strength and rigidity. It can inhibit rMrp2-mediated [3H]E217βG uptake (IC50: 199 μM).

价 格：￥电议型 号：T6437产 地：中国大陆

T4448NADPNADP

价 格：￥电议型 号：T4448产 地：中国大陆

T60187RP-6685RP6685

RP-6685 is a potent, selective and orally active DNA polymerase theta (Polθ) inhibitor with an IC 50 value of 5.8 nM in PicoGreen assay. RP-6685 shows antitumor efficacy in mouse tumor xenograft model [1].

价 格：￥电议型 号：T60187产 地：中国大陆

T8973HS-1793HIF-1α,Inhibitor,MCF-7,HS 1793,breast cancer,inhibit,ERK,HCT116,resveratrol,VEGF,Apoptosis,HS

HS-1793, a resveratrol analogue, downregulates the expression of hypoxia-induced HIF-1 and VEGF and inhibits tumor growth of human breast cancer cells in a nude mouse xenograft model

价 格：￥电议型 号：T8973产 地：中国大陆

T8580Bupranololnon-selective,competitive,Adrenergic Receptor,Bupranolol,Inhibitor,intrinsic,sympathomimet

Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.

价 格：￥电议型 号：T8580产 地：中国大陆

T27969M7594_0037

M7594_0037 is an inhibitor of Human peptide deformylase (HsPDF) and can be used in studies about anticancer.

价 格：￥电议型 号：T27969产 地：中国大陆

T76922,4-DPDCollagen formation,Diethyl ester,Chick-embryo calvaria,2,4DPD,inhibit,Inhibitor,Prolyl hydrox

2,4-DPD is competitive inhibitor of the oxygen-sensing enzyme HIF-α prolyl hydroxylase (HIF-PH)

价 格：￥电议型 号：T7692产 地：中国大陆

T8173Delafloxacin meglumineWQ3034,inhibit,ABT492,ABT-492,Delafloxacin meglumine,Inhibitor,RX3341,RX-3341,

Delafloxacin meglumine is a broad-spectrum fluoroquinolone antibiotic

价 格：￥电议型 号：T8173产 地：中国大陆

T9597H2S Donor 5aEndogenous Metabolite,H2S donor,biological systems,H2S Donor 5a,cysteine-activated,Inhib

H2S Donor 5a is a H2S donor that could mimic the slow and continuous H(2)S generation process.

价 格：￥电议型 号：T9597产 地：中国大陆

T67728α-Glucosidase-IN-23αGlucosidaseIN23

α-Glucosidase-IN-23 is an orally active α-Glucosidase inhibitor. α-Glucosidase-IN-23 can decrease blood glucose by α-glucosidase inhibition (IC50= 4.48 μM).

价 格：￥电议型 号：T67728产 地：中国大陆