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T79786H4R antagonist 2；化合物 H4R antagonist 2H4R antagonist 2
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid arthritis [1] (page 68).
价 格：￥电议型 号：T79786产 地：中国大陆
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T79782FPR1 antagonist 2；化合物 FPR1 antagonist 2FPR1 antagonist 2
Compound 25b, an FPR1 antagonist, exhibits potent inhibition of the formyl peptide receptor 1 with an IC50 of 70 nM. It concurrently hampers cell proliferation and triggers apoptosis, diminishing cell growth and migration, yet paradoxically augments angiogenesis [1].
价 格：￥电议型 号：T79782产 地：中国大陆
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T79781FPR1 antagonist 1；化合物 FPR1 antagonist 1FPR1 antagonist 1
Compound 24a, an FPR1 antagonist, demonstrates potent inhibition of the formyl peptide receptor 1 (FPR1) with an IC50 value of 25 nM. It impedes cell proliferation and promotes apoptosis, thereby inhibiting cell growth. This compound also attenuates cell migration and concurrently promotes angiogenesis [1].
价 格：￥电议型 号：T79781产 地：中国大陆
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T79772RARα antagonist 1；化合物 RARα antagonist 1RARα antagonist 1
Compound 21, an orally active and selective RARα antagonist, exhibits a potent inhibition of the retinoic acid receptor α with an IC50 of 4.6 nM [1].
价 格：￥电议型 号：T79772产 地：中国大陆
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T796845-HT6R antagonist 1；化合物 5-HT6R antagonist 15-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability but also reverses MK-801-induced memory impairments in rats, suggesting its utility in Alzheimer´s disease (AD) research [1].
价 格：￥电议型 号：T79684产 地：中国大陆
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T79575ET receptor antagonist 3；化合物 ET receptor antagonist 3ET receptor antagonist 3
"ET receptor antagonist 3 (compound 17d) is an orally active ET receptor antagonist with an IC50 of 0.26 nM, utilized for pulmonary arterial hypertension (PAH) research. This compound demonstrates efficacy in mitigating monocrotaline-induced PAH in a rat model [1]."
价 格：￥电议型 号：T79575产 地：中国大陆
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T79574ET receptor antagonist 2；化合物 ET receptor antagonist 2ET receptor antagonist 2
ET Receptor Antagonist 2 (Compound 16j) is an orally active ET receptor antagonist with an IC50 of 0.22 nM, suitable for pulmonary arterial hypertension (PAH) research. It has been shown to mitigate monocrotaline-induced PAH in a rat model [1].
价 格：￥电议型 号：T79574产 地：中国大陆
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T79573ET receptor antagonist 1；化合物 ET receptor antagonist 1ET receptor antagonist 1
ET Receptor Antagonist 1 (compound 16h), with an IC50 value of 0.18 nM, is an orally active agent that can be utilized for pulmonary arterial hypertension (PAH) research. It has demonstrated efficacy in mitigating monocrotaline-induced PAH in a rat model [1].
价 格：￥电议型 号：T79573产 地：中国大陆
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T79464RORγ antagonist 1；化合物 RORγ antagonist 1RORγ antagonist 1
RORγ antagonist 1 (compound 22), a potent derivative of betulinic acid, acts as an antagonist to RORγ with a dissociation constant (K D) of 0.18 μM. It demonstrates anti-proliferative effects in the HPAF-II pancreatic cancer xenograft model, inhibits the RAS/MAPK and AKT/mTORC1 signaling pathways, and triggers caspase-dependent apoptosis in pancreatic cancer cells [1].
价 格：￥电议型 号：T79464产 地：中国大陆
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T79431Mu opioid receptor antagonist 7；化合物 Mu opioid receptor antagonist 7Mu opioid receptor antagonist 7
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting ?-opioid receptor (?OR) antagonist with an inhibitory concentration (IC50) of 29 ± 3.0 nM. It is valuable for pain and opioid use disorder research [1].
价 格：￥电议型 号：T79431产 地：中国大陆
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T79418BLT2 antagonist-1；化合物 BLT2 antagonist-1BLT2 antagonist-1
BLT2 antagonist-1 (compound 15b) is a selective inhibitor of the BLT2 receptor, impeding the chemotaxis of CHO-BLT2 cells at an IC50 of 224 nM, while not affecting CHO-BLT1 cell chemotaxis. It blocks the interaction between LTB4 and the BLT2 receptor with a K_i of 132 nM and may serve as a research tool for inflammatory airway diseases, including asthma and chronic obstructive pulmonary disease [1].
价 格：￥电议型 号：T79418产 地：中国大陆
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T79375NMDA receptor antagonist 8；化合物 NMDA receptor antagonist 8NMDA receptor antagonist 8
Compound (R)-10a, an NMDA receptor antagonist, exhibits selectivity for the GluN2B subunit, possessing a Ki of 265 nM and an IC50 of 62 nM. This compound is utilized in research pertaining to neurodegenerative diseases [1].
价 格：￥电议型 号：T79375产 地：中国大陆
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T79374NMDA receptor antagonist 7；化合物 NMDA receptor antagonist 7NMDA receptor antagonist 7
Compound (S)-10a, a GluN2B subunit-selective NMDA receptor antagonist, exhibits a K i of 93 nM and an IC 50 of 72 nM. It is potentially useful for research into neurodegenerative diseases [1].
价 格：￥电议型 号：T79374产 地：中国大陆
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T79273NMDA receptor antagonist 6；化合物 NMDA receptor antagonist 6NMDA receptor antagonist 6
NMDA Receptor Antagonist 6 (Compound 13b) functions as an antagonist at the glycine-binding site of the NMDA receptor and demonstrates cytoneuroprotective efficacy. It safeguards PC12 cells from NMDA-induced damage and apoptosis [1].
价 格：￥电议型 号：T79273产 地：中国大陆
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T79184FKBP51F67V-selective antagonist Ligand2；化合物 FKBP51F67V-selective antagonist Ligand2FKBP51F67V-select
FKBP51F67V-selective antagonist Ligand2 (example 3-3), a potent ligand, selectively binds to the FKBP51 F67V variant, with no affinity for wild-type FKBP51 or FKBP52 [1]. It effectively reverses the anxiogenic phenotype resulting from FKBP51 F67V overexpression in the amygdala.
价 格：￥电议型 号：T79184产 地：中国大陆
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T79115P2X3 antagonist 38；化合物 P2X3 antagonist 38P2X3 antagonist 38
Compound 38, also known as Compound 4, is a potent, orally active P2X3 antagonist that demonstrates inhibitory activity with IC50 values of 0.132 ?M, 0.165 ?M, and 0.421 ?M against human (hP2X3), rat (rP2X3), and guinea pig (gpP2X3) P2X3 receptors, respectively [1].
价 格：￥电议型 号：T79115产 地：中国大陆
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T79071HPK1 antagonist-1；化合物 HPK1 antagonist-1HPK1 antagonist-1
HPK1 antagonist-1 (I-792) is an inhibitor targeting HPK1, with potential applications in cancer and immune disease research [1].
价 格：￥电议型 号：T79071产 地：中国大陆
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T79027A1/A3 AR antagonist 3；化合物 A1/A3 AR antagonist 3A1/A3 AR antagonist 3
A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in the research of chronic heart diseases [1].
价 格：￥电议型 号：T79027产 地：中国大陆
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T79023CaSR antagonist-1；化合物 CaSR antagonist-1CaSR antagonist-1
CaSR Antagonist-1 is a potent inhibitor of the calcium-sensing receptor (CaSR) with an inhibitory concentration (IC50) of 50 nM, suitable for the investigation of diseases related to dysregulated bone or mineral homeostasis, including osteoporosis [1].
价 格：￥电议型 号：T79023产 地：中国大陆
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T78779D3R/MOR antagonist 2；化合物 D3R/MOR antagonist 2D3R/MOR antagonist 2
Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR partial agonism and may reduce opioid-misuse liability through D3R antagonism [1].
价 格：￥电议型 号：T78779产 地：中国大陆
