T6635EMD638683inhibit,EMD-638683,EMD638683,Serum and glucocorticoid-regulated kinase,EMD 638683,Inhibitor

EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).

价 格：￥电议型 号：T6635产 地：中国大陆

TP2212La-MSH, amide Acetate(581-05-5 free base)a MSH, amide Acetate(581 05 5 free base),aMSH, amide Acetate

a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities. α-MSH is a post-translational derivative of pro-opiomelanocortin (POMC)

价 格：￥电议型 号：TP2212L产 地：中国大陆

T67742EX-A5386

EX-A5386 is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.

价 格：￥电议型 号：T67742产 地：中国大陆

TN71672,4,5-Tribromoimidazole

2,4,5-Tribromoimidazole is a marine derived natural products found in Hexaplex trunculus.

价 格：￥电议型 号：TN7167产 地：中国大陆

TP1086Men 10376 TFA(135306-85-3,free)Men 10376 TFA(135306853,free),Men 10376 TFA(135306 85 3,free)

Men 10376 TFA is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.

价 格：￥电议型 号：TP1086产 地：中国大陆

T7295MiridesapGSK 2315698,GSK-2315698,Miridesap,Inhibitor,inhibit

Miridesap is a divalent crosslinker of SAP that causes rapid depletion of circulating SAP via hepatic clearance. It also produces significant reduction of SAP from cerebrospinal fluid and visceral amyloid deposits

价 格：￥电议型 号：T7295产 地：中国大陆

Fr14534Compound Fr14534Compound Fr14534

价 格：￥电议型 号：Fr14534产 地：中国大陆

T9459GR103545Inhibitor,Opioid Receptor,imaging,GR103545,inhibit,κ-OR,GR 103545,κ-opioid receptor,GR-10354

(R)-(-)-GR103545 fumarate is a chemical compound.

价 格：￥电议型 号：T9459产 地：中国大陆

T9306EST64454 Maleic acid saltEST-64454 Maleic acid salt,EST64454 Maleic acid salt

EST64454 Maleic acid salt is a compound.

价 格：￥电议型 号：T9306产 地：中国大陆

T30577BRD0418

BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.

价 格：￥电议型 号：T30577产 地：中国大陆

T9753LEI110HepG2 cells,inhibit,thiol hydrolases,LEI110,Inhibitor,LEI-110,lipolysis,Phospholipase,LEI 110

LEI110 is a potent Phospholipase A2, group XVI (PLA2G16) inhibitor with an Ki value of 20 nM. LEI110 is a selective pan-inhibitor of the HRASLS family of thiol hydrolases (i.e., PLA2G16, HRASLS2, RARRES3 and iNAT).

价 格：￥电议型 号：T9753产 地：中国大陆

T9519EliapixantInhibitor,chronic,Eliapixant,cough,refractory,BAY-1817080,P2X Receptor,BAY1817080,P2X3,inh

Eliapixant (BAY 1817080) is a potent and selective P2X3 receptor antagonist, with an IC50 of 8 nM. Eliapixant can be used for the research of refractory chronic cough.

价 格：￥电议型 号：T9519产 地：中国大陆

T7529Yamogenintriacylglyceride,Inhibitor,fatty acid synthesis,Diastereomer,Yamogenin,Liver X receptor,LXR

Yamogenin is a diastereomer of diosgenin, which we have identified as the compound responsible for the anti-hyperlipidemic effect of fenugreek.

价 格：￥电议型 号：T7529产 地：中国大陆

T7303LIXIVAPTANVPA 985,LIXIVAPTAN,VPA985,inhibit,Inhibitor,Vasopressin Receptor

Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)

价 格：￥电议型 号：T7303产 地：中国大陆

T8435YM90Kanticonvulsant,AMPA,Inhibitor,ischemia,inhibit,neuroprotective,Ionotropic glutamate receptors,Y

YM90K hydrochloride is an antagonist of AMPA receptor.

价 格：￥电议型 号：T8435产 地：中国大陆

T8485THIQmutant,MC Receptor,inhibit,THIQ,melanocortin,affinity,activity,erectile,selective,eliciting,Mela

THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).

价 格：￥电议型 号：T8485产 地：中国大陆

T6885MarimastatTA-2516,Marimastat,inhibit,Inhibitor,BB 2516,BB-2516,TA 2516,Matrix metalloproteinases,MMP

Marimastat (BB-2516) is a potent, broad spectrum matrix metalloprotease (MMP) inhibitor. MMP-9 (IC50=3 nM), MMP-1 (IC50=5 nM), MMP-2 (IC50=6 nM), MMP-14 (IC50=9 nM)and MMP-7 (IC50=13 nM).

价 格：￥电议型 号：T6885产 地：中国大陆

T8556Z-Gly-Gly-Arg-AMC TFA (66216-78-2 free base)Z Gly Gly Arg AMC TFA (66216 78 2 free base),ZGlyGlyArgA

Z-Gly-Gly-Arg-AMC is a thrombin-specific fluorogenic substrate for testing of thrombin generation in PRP and platelet-poor plasma (PPP).

价 格：￥电议型 号：T8556产 地：中国大陆

T6S1579MonotropeinMonotropein,Inhibitor,inhibit

1. Monotropein has antinociceptive action. 2. Monotropein has anti-apoptosis and anti-catabolic activity in chondrocytes. 3. Monotropein has anti-inflammatory action by inhibition of the expressions of inflammatory mediators via NF-κB inactivation, and support its possible therapeutic role in colitis. 4. Monotrope ininhibit the expressions of inducible nitric oxide synthase (iNOS), cyclooxygenase-2 (COX-2), tumor necrosis factor-α (TNF-α), and interleukin-1β (IL-1β) mRNA in LPS-induced RAW 264.7

价 格：￥电议型 号：T6S1579产 地：中国大陆

TP1045LOrexin B, rat, mouse AcetateOrexin B, rat, mouse Acetate

Orexin B, rat, mouse Acetate is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.

价 格：￥电议型 号：TP1045L产 地：中国大陆