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T74754FXR antagonist 2；化合物 FXR antagonist 2FXR antagonist 2
Compound A-26, also known as FXR antagonist 2, is a diarylamide derivative that functions as a moderate FXR antagonist. It is utilized in researching hyperlipidemia and type 2 diabetes [1].
价 格：￥电议型 号：T74754产 地：中国大陆
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T74606A2A/A3u00A0AR antagonist-1；化合物 A2A/A3u00A0AR antagonist-1A2A/A3u00A0AR antagonist-1
Compound 23, designated as A2A/A3 AR antagonist-1, is a dual fluorescent ligand targeting A2A and A3 adenosine receptors (AR), exhibiting dissociation constants (Ki) of 90 nM for hA2A AR and 31.8 nM for hA3 AR, respectively [1].
价 格：￥电议型 号：T74606产 地：中国大陆
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T74538Galectin-3 antagonist 2；化合物 Galectin-3 antagonist 2Galectin-3 antagonist 2
Galectin-3, a β-galactoside-specific carbohydrate recognition protein (lectin), facilitates the migration of B-cell precursor acute lymphoblastic leukemia (BCP-ALL) cells and demonstrates resistance to pharmaceutical interventions.
价 格：￥电议型 号：T74538产 地：中国大陆
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T74350Neuropeptide Y Y1u00A0receptor antagonist 1；化合物 Neuropeptide Y Y1u00A0receptor antagonist 1Neuropept
Neuropeptide Y Y1 receptor antagonist 1 (compound 39), a fluorescent probe, serves as a powerful antagonist against the neuropeptide Y Y1 receptor (Y1R), exhibiting a K? value of 0.19 nM [1]. It should be stored in conditions shielded from light.
价 格：￥电议型 号：T74350产 地：中国大陆
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T74266Protease-Activated Receptor-1 antagonistu00A02；化合物 Protease-Activated Receptor-1 antagonistu00A02Pro
Protease-Activated Receptor-1 Antagonist 2 is an orally active antagonist of protease-activated receptor-1 (PAR-1), demonstrating significant potency with an IC 50 of 7 nM. It exhibits favorable pharmacokinetic characteristics, making it valuable in cardiovascular disease (CVD) research, including studies on atherosclerosis and restenosis [1].
价 格：￥电议型 号：T74266产 地：中国大陆
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T7347CU-CPT-8m；化合物CU-CPT-8mTLR8-specific antagonist；TLR8-specific antagonist
CU-CPT-8m (TLR8-specific antagonist) is an toll-like receptor 8 (TLR8) antagonist (IC50 : 67 nM)
价 格：￥电议型 号：T7347产 地：中国大陆
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T7302CU-CPT9b；化合物CU-CPT9bCU-CPT-9b|||TLR8-specific antagonist 1；CU-CPT-9b|||TLR8-specific antagonist 1
CU-CPT9b (TLR8-specific antagonist 1) is an antagonist of toll-like receptor 8 (TLR8; Kd = 21 nM). It inhibits activation of NF- B induced by the TLR8 agonist R-848 in TLR8-overexpressing HEK-Blue cells with an IC50 value of 0.7 nM.
价 格：￥电议型 号：T7302产 地：中国大陆
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T72626A2AR-antagonist-1；化合物 A2AR-antagonist-1A2AR-antagonist-1
A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability in mouse liver microsomes (t1/2 = 86.1 min). Additionally, it activates T cells by inhibiting immunosuppressive molecules (LAG-3 and TIM-3) and promoting expression of effector molecules (GZMB, IFNG, and IL-2) [1].
价 格：￥电议型 号：T72626产 地：中国大陆
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T72625LTB4 antagonist 1；化合物 LTB4 antagonist 1LTB4 antagonist 1
LTB4 Antagonist 1, a carboxamide-acid derivative, potently inhibits Leukotriene B4 (LTB4) activity with an IC50 value of 288 nM and exhibits notable anti-inflammatory properties [1].
价 格：￥电议型 号：T72625产 地：中国大陆
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T72621GCGR antagonist 2；化合物 GCGR antagonist 2GCGR antagonist 2
GCGR Antagonist 2, a Furan-2-carbohydrazide, serves as an orally active antagonist of the glucagon receptor. It exhibits affinity for the human glucagon receptor (hGluR) with a dissociation constant (Kd) of 2.3 nM and demonstrates inhibitory activity against the rat receptor with a half-maximal inhibitory concentration (IC50) of 0.43 nM. Additionally, this compound effectively prevents glucagon-stimulated glycogenolysis.
价 格：￥电议型 号：T72621产 地：中国大陆
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T72606AT1R antagonist 1；化合物 AT1R antagonist 1AT1R antagonist 1
AT1R Antagonist 1 (compound 10) serves as a potent, selective ligand for AT1R with considerable affinity, demonstrated by a K i value of 8.5 nM [1].
价 格：￥电议型 号：T72606产 地：中国大陆
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T72588A3AR antagonist 2；化合物 A3AR antagonist 2A3AR antagonist 2
A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.
价 格：￥电议型 号：T72588产 地：中国大陆
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T72536GPR84 antagonist 2；化合物 GPR84 antagonist 2GPR84 antagonist 2
GPR84 Antagonist 2, a potent and selective GPR84 antagonist (IC 50 = 8.95 nM), demonstrates oral activity and significantly enhances potency in calcium mobilization assays. It effectively inhibits neutrophil and macrophage chemotaxis following GPR84 activation, highlighting its research potential for ulcerative colitis.
价 格：￥电议型 号：T72536产 地：中国大陆
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T72492GnRH-R antagonist 1；化合物 GnRH-R antagonist 1GnRH-R antagonist 1
GnRH-R antagonist 1 (Compound 21a), is an orally active, membrane-permeable agent with a high binding affinity (IC50=0.57 nM) and potent in vitro antagonistic efficacy (IC50=2.18 nM). It is utilized in research focused on advanced prostate cancer and the prevention of premature LH surges [1].
价 格：￥电议型 号：T72492产 地：中国大陆
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T72473NOD1/2 antagonist-1；化合物 NOD1/2 antagonist-1NOD1/2 antagonist-1
NOD1/2 Antagonist-1 is a potent dual inhibitor of nucleotide-binding oligomerization domain-like receptors 1 and 2 (NOD1/2), displaying inhibitory concentrations (IC50) of 1.13 μM for NOD1 and 0.77 μM for NOD2. It exhibits an acceptable half-life (T1/2) of 67.6 minutes. Additionally, NOD1/2 Antagonist-1 enhances the antitumor efficiency of Paclitaxel (PTX).
价 格：￥电议型 号：T72473产 地：中国大陆
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T72410Sortilin antagonist 1；化合物 Sortilin antagonist 1Sortilin antagonist 1
Sortilin Antagonist 1, a potent sortilin antagonist, exhibits an inhibition constant (IC50) of 20 nM against Neurotensin (NTS) binding to sortilin. Neurotensin acts as a sortilin ligand. This compound is utilized in neurological disease research.
价 格：￥电议型 号：T72410产 地：中国大陆
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T72224NK1 receptor antagonist 2；化合物 NK1 receptor antagonist 2NK1 receptor antagonist 2
NK1 Receptor Antagonist 2, a compound targeting the NK1 receptor, holds potential for tinnitus and hearing loss research.
价 格：￥电议型 号：T72224产 地：中国大陆
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T72198P2X7 receptor antagonist-3；化合物 P2X7 receptor antagonist-3P2X7 receptor antagonist-3
P2X7 receptor antagonist-3 is a powerful inhibitor of the P2X7 receptor, exhibiting IC50 values of 4.2 nM in humans and 6.8 nM in rats, indicating its high potency in both species.
价 格：￥电议型 号：T72198产 地：中国大陆
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T72091ADRA1D receptor antagonist 1 free base；化合物 ADRA1D receptor antagonist 1 free baseADRA1D receptor ant
ADRA1D receptor antagonist 1 (free base) antagonist ( K i =1.6 nM). ADRA1D receptor antagonist 1 (free base) dose-dependently inhibits bladder contraction with an IC 30 value of 15 nM. ADRA1D receptor antagonist 1 (free base) can be used in studies of overactive bladder disorders such as urinary urgency, frequency and incontinence.
价 格：￥电议型 号：T72091产 地：中国大陆
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T71515RhlR Antagonist E22；化合物 RhlR Antagonist E22RhlR Antagonist E22
RhlR antagonist E22 is a quorum sensing modulator as an RhlR antagonist.
价 格：￥电议型 号：T71515产 地：中国大陆
