PDK0113Compound PDK0113Compound PDK0113

价 格：￥电议型 号：PDK0113产 地：中国大陆

T7945SU14813c-Kit,Inhibitor,VEGFR,Vascular endothelial growth factor receptor,SU 14813,PDGFR,CD117,Platel

SU14813 is a multi-receptor tyrosine kinase inhibitor with potent antiangiogenesis and antitumor activity (IC50s of 50, 2, 4, 15 nM for VEGFR2, VEGFR1, PDGFRβ and KIT).

价 格：￥电议型 号：T7945产 地：中国大陆

T4030ML213CID-3111211

ML213 is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM, respectively.

价 格：￥电议型 号：T4030产 地：中国大陆

T12571PSI-6206 13CD3PSI-6206 13CD3,RO-2433 13CD3,GS-331007 13CD3

PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.

价 格：￥电议型 号：T12571产 地：美洲

T79900Cbl-b-IN-13；化合物 Cbl-b-IN-13Cbl-b-IN-13

Cbl-b-IN-13 (Example 520) is a potent Cbl-b inhibitor exhibiting an IC50 of less than 100 nM and is capable of activating T-cells [1].

价 格：￥电议型 号：T79900产 地：中国大陆

T79481Chitin synthase inhibitor 13；化合物 Chitin synthase inhibitor 13Chitin synthase inhibitor 13

Chitin Synthase Inhibitor 13 (compound 12g), a non-competitive antagonist of chitin synthase, demonstrates broad-spectrum antifungal activity and has an inhibition concentration (IC50) of 106.7 μM [1].

价 格：￥电议型 号：T79481产 地：中国大陆

T79187CT1113；化合物 CT1113CT1113

CT1113, a potent inhibitor of both USP28 and USP25, effectively reduces MYC levels in vivo and demonstrates anti-tumor efficacy in a mouse pancreatic cancer CDX model [1].

价 格：￥电议型 号：T79187产 地：中国大陆

T72029CDK8-IN-13；化合物CDK8-IN-13CDK8-IN-13

CDK8-IN-13 is a CDK8 inhibitor (IC50: 51.9 nM) with potent, selective and oral activity. CDK8-IN-13 induces apoptosis and reduces the expression of p-STAT1 S727 and p-STAT5 S726. CDK8-IN-13 exhibits anti-tumour activity.

价 格：￥电议型 号：T72029产 地：中国大陆

T68537CEP-14513；化合物 CEP-14513CEP-14513

CEP-14513 is a potent ALK inhibitor. CEP-14513 displayed potent ALK inhibitory activity in both in vitro enzymatic assay (IC50 = 5 nM) and cell-based assays of ALK tyrosine phosphorylation (IC50 = 30 nM).

价 格：￥电议型 号：T68537产 地：中国大陆

T6801CeMMEC13；化合物CeMMEC13CeMMEC13

CeMMEC13 is an isoquinolinone that selectively inhibits the second bromodomain of TAF1 (IC50 = 2.1 μM).

价 格：￥电议型 号：T6801产 地：中国大陆

T64482Urea-13C；化合物 Urea-13CUrea-13C

Urea-13C is a useful organic compound for research related to life sciences. The catalog number is T64482 and the CAS number is 58069-82-2.

价 格：￥电议型 号：T64482产 地：中国大陆

T63885c-Met-IN-13；化合物 c-Met-IN-13c-Met-IN-13

c-Met-IN-13 is a potent inhibitor of c-Met (IC50: 2.43 nM). c-Met-IN-13 exhibits anti-proliferative effects in a concentration-dependent and time-dependent manner. c-Met-IN-13 exhibits significant cytotoxicity against cancer cells. c-Met-IN-13 has shown therapeutic potential against cancer.

价 格：￥电议型 号：T63885产 地：中国大陆

T63519Cap-dependent endonuclease-IN-13；化合物 Cap-dependent endonuclease-IN-13Cap-dependent endonuclease-IN-1

Cap-dependent endonuclease-IN-13 is a potent inhibitor of cap-dependent endonuclease (CEN) and shows research potential against influenza virus infection (influenza A only).

价 格：￥电议型 号：T63519产 地：中国大陆

T62919CDK9-IN-13；化合物 CDK9-IN-13CDK9-IN-13

CDK9-IN-13 is a potent and selective CDK inhibitor (IC50<3 nM). CDK9-IN-13 has a very short half-life in rodents.

价 格：￥电议型 号：T62919产 地：中国大陆

T62759CDK7-IN-13；化合物 CDK7-IN-13CDK7-IN-13

CDK7-IN-13 is a pyrimidine-derived compound that is a potent inhibitor of CDK7. CDK7-IN-13 has the potential to be investigated in a variety of cancers (particularly those with dysregulated transcription).

价 格：￥电议型 号：T62759产 地：中国大陆

T62605CDK4/6-IN-13；化合物 CDK4/6-IN-13CDK4/6-IN-13

Compounds 10B and 10C, functioning as cdk4/6 inhibitors, demonstrated low nanomolar activity, optimal antiproliferative effects, excellent metabolic properties, and acceptable pharmacokinetics targeting cdk4/6.

价 格：￥电议型 号：T62605产 地：中国大陆

T624793CPLro-IN-1；化合物 3CPLro-IN-13CPLro-IN-1

3CPLro-IN-1 (compound A17) is a potent, orally active inhibitor of SARS-CoV-2 3CLpro (IC50: 5.65 μM). 3-Chymotrypsin-like cysteine protease (3CLpro), a protein essential for viral replication, is an attractive drug target against COVID-19. Antitumor agent-51

价 格：￥电议型 号：T62479产 地：中国大陆

T61952Carbonic anhydrase inhibitor 13；化合物 Carbonic anhydrase inhibitor 13Carbonic anhydrase inhibitor 13

Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).

价 格：￥电议型 号：T61952产 地：中国大陆

T61714COX-2-IN-13；化合物 COX-2-IN-13COX-2-IN-13

COX-2-IN-13 (compound 13e) is a highly potent and selective inhibitor of COX-2, demonstrating a remarkable IC50 value of 0.98 μM. It exhibits strong anti-inflammatory activity and has shown favorable results in vivo acute toxicity studies [1].

价 格：￥电议型 号：T61714产 地：中国大陆

T61589c-Fms-IN-13；化合物c-Fms-IN-13c-Fms-IN-13

c-Fms-IN-13 (compound 14) is a potent FMS kinase inhibitor (IC50= 17 nM). c-Fms-IN-13 is an anti-inflammatory agent.

价 格：￥电议型 号：T61589产 地：中国大陆