T31204Darapladib-impurityDarapladib impurity,Darapladibimpurity

Darapladib-impurity is the impurity of Darapladib. Darapladib inhibits lipoprotein-associated phospholipase A2 (Lp-PLA2)

价 格：￥电议型 号：T31204产 地：中国大陆

T67698WAY-300374WAY300374

WAY-300374 inhibits the p53-MDM2 protein-protein interaction.

价 格：￥电议型 号：T67698产 地：中国大陆

T7848PT-2385Inhibitor,inhibit,Hypoxia-inducible factors,HIF/HIF Prolyl-Hydroxylase,HIF-PH,PT 2385,HIFs,PT

PT-2385 is a selective HIF-2α inhibitor (Kd<50 nM).

价 格：￥电议型 号：T7848产 地：中国大陆

T15018CUDC-427

CUDC-427 is an orally bioactive and pan antagonist of inhibitor of apoptosis proteins(IAPs). CUDC-427 can be used in research on cancers.

价 格：￥电议型 号：T15018产 地：中国大陆

TP1559LZiconotide Acetate (107452-89-1 free base)analgesic,non-opioid,Ziconotide Acetate (107452891 free

Ziconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.

价 格：￥电议型 号：TP1559L产 地：中国大陆

T8439Clobenpropit dihydrobromideApoptosis,inhibit,Clobenpropit dihydrobromide,histamine H3R,antagonist,in

Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)

价 格：￥电议型 号：T8439产 地：中国大陆

T15641K777

K777 is a potent, orally active and irreversible inhibitor of cysteine protease. K777 is a potent CYP3A4 inhibitor (IC50= 60 nM). K777 is also a selective CCR4 antagonist featuring the potent chemotaxis inhibition. K777 irreversibly inhibits Cruzain, which is the major cysteine protease of Trypansoma cruzi, and cathepsins B and L. K777 targets cathepsin-mediated cell entry and wxibits a broad-spectrum antiviral activity. K777 inhibits EBOV and SARS-CoV pseudovirus entry with IC50 values of 0.87

价 格：￥电议型 号：T15641产 地：中国大陆

T8331NUN82647NUN82647,Inhibitor,NUN 82647,inhibit,Apoptosis,QBS,NUN-82647

NUN82647 is an Inhibitor of cell cycle at G2 phase, and apoptosis inducer.

价 格：￥电议型 号：T8331产 地：中国大陆

T9840AtaquimasAtaquimas

Ataquimast inhibits IL-5 secretion along with that of TNF-a, IL-4 and GM-CSF from human cells.

价 格：￥电议型 号：T9840产 地：中国大陆

T16940STAT5-IN-2STAT-5-IN-2,STAT5IN2,STAT5 IN 2

STAT5-IN-2 is an inhibitor of STAT5 with antileukemic effects (EC50s: 9 μM and 5 μM in K562 and KU812 cells, respectively).

价 格：￥电议型 号：T16940产 地：中国大陆

PDK04236-METHYL-1H-INDOLE-2-CARBOXYLIC ACID6METHYL1HINDOLE2CARBOXYLICACID

价 格：￥电议型 号：PDK0423产 地：中国大陆

TP1881L1Pep 2-8 ammonium salt(1541011-97-5 free base)Pep 2 8 ammonium salt(1541011 97 5 free base),Pep 28 am

Pep 2-8 ammonium salt is Proprotein convertase subtilisin/kexin type 9 (PCSK9) inhibitor. Potent inhibitor of PCSK9 binding to LDL receptor (IC50 = 0.8 μM). Restores LDL uptake in HepG2 cells treated with PCSK9.

价 格：￥电议型 号：TP1881L1产 地：中国大陆

T22849ICI 199,441 hydrochlorideICI 199,441 hydrochloride

ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.

价 格：￥电议型 号：T22849产 地：中国大陆

T11023DHODH-IN-14DHODH IN 14,DHODHIN14

DHODH-IN-14 is an analog of hydroxyfuran pyrimidine A771726. DHODH-IN-14 is a dihydroorotate dehydrogenase (DHODH) inhibitor IC50 0.49 μM mouse liver DHODH. DHODH-IN-14 can be used for rheumatoid arthritis.

价 格：￥电议型 号：T11023产 地：中国大陆

TN1438beta-Amyrin acetateHMG-CoA,betaAmyrin acetate,LDL,Fungal,inhibit,Inhibitor,arthritic,hemolysis,antif

beta-Amyrin acetate inhibits HMG-CoA Reductase (HMGCR) and sEH activity with IC50 of 3.4 μM. beta-Amyrin acetate has anti-inflammatory, antifungal, antioxidant, and anti-hyperlipidemic activities.

价 格：￥电议型 号：TN1438产 地：中国大陆

TN4871PyrolinPyrolin

Pyrolin has a strong antifungal activity and exerts a potent impact on the ultrastructure of M.fructicola.

价 格：￥电议型 号：TN4871产 地：中国大陆

TP1898HS024selective,melanocortin,intake,Inhibitor,Melanocortin Receptor,MC Receptor,HS-024,food,HS024,inh

Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.

价 格：￥电议型 号：TP1898产 地：中国大陆

TN1768IriflophenoneInhibitor,MCF-7,proliferation,Iriflophenone,cells,T-47D,inhibit

Iriflophenone?stimulates cells proliferation in?MCF-7 and T-47D human breast cancer.

价 格：￥电议型 号：TN1768产 地：中国大陆

TJS03384-Methylesculetininhibit,4 Methylesculetin,Glutathione Peroxidase,4-Methylesculetin,Inhibitor,4Methy

4-methylesculetin is one of the coumarin derivatives with great anti-oxidant and anti-inflammatory activities.

价 格：￥电议型 号：TJS0338产 地：中国大陆

T9645CU-115

CU-115 is a selective and potent TLR8 antagonist with IC50 of 1.04 ?M and =>50 ?M for TLR8 and TLR7, respectively. CU-115 decreases production of TNF-α and IL-1β activated by R-848 in THP-1 cells.

价 格：￥电议型 号：T9645产 地：中国大陆