T6445CilomilastCilomilast,asthma,immunomodulatory,obstructive,Inhibitor,Phosphodiesterase (PDE),inhibit,P

Cilomilast is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity. Phase 3.

价 格：￥电议型 号：T6445产 地：中国大陆

PDK0140Compound PDK0140Compound PDK0140

价 格：￥电议型 号：PDK0140产 地：中国大陆

T7761Pomalidomide-C2-NH2 hydrochloridePomalidomideC2NH2 hydrochloride,inhibit,Inhibitor,Pomalidomide-C-2-

Pomalidomide-C2-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conjugate. Pomalidomide-C2-NH2 hydrochloride incorporates the Pomalidomide based cereblon ligand and a linker used in PROTAC technology.

价 格：￥电议型 号：T7761产 地：中国大陆

T8081LC3-mHTT-IN-AN1Autophagosome-tethering compounds,LC3mHTTINAN1,Autophagy,LC3 mHTT IN AN1,ATTECs,Inhib

LC3-mHTT-IN-AN1 is a mHTT-LC3 linker compound that interacts with both mutant huntingtin protein (mHTT) and LC3B. LC3-mHTT-IN-AN1 targeted mHTT to autophagosomes reduces the levels of mHTT in an allele-selective manner in cultured Huntington disease (HD) mouse neurons.

价 格：￥电议型 号：T8081产 地：中国大陆

T407281-Bromo-6-chlorohexane

1-Bromo-6-chlorohexane is used as PROTAC linker.

价 格：￥电议型 号：T40728产 地：中国大陆

T86022-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE2 CHLOROMETHYL 1,1 DIOXO 1,2

2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).

价 格：￥电议型 号：T8602产 地：中国大陆

TQ0012AZ3451AZ 3451,inhibit,Protease Activated Receptor (PAR),AZ-3451,AZ3451,Thrombin receptors,Inhibitor

AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).

价 格：￥电议型 号：TQ0012产 地：中国大陆

T89084-Chloro-2’-bromoacetophenone4 Chloro 2’ bromoacetophenone,4Chloro2’bromoacetophenone

4-Chloro-2´-bromoacetophenone against glycogen synthase kinase-3 (GSK-3beta).

价 格：￥电议型 号：T8908产 地：中国大陆

T86348-Bromotheophylline8-Bromotheophylline,Inhibitor,8 Bromotheophylline,inhibit,8Bromotheophylline

Bromotheophylline is the active moiety of pamabrom, a mixture of 2-amino-2-methyl-propanol and bromotheophylline. From this mixture, bromotheophylline acts as a weak diuretic that has been used along with some analgesics to relieve the symptoms of premenstrual syndrome

价 格：￥电议型 号：T8634产 地：中国大陆

T9756AZD-9574PPAR,Peroxisome proliferator-activated receptors,breast cancer,inhibit,AZD-9574,HRR,HRR-defi

AZD-9574 is a selective inhibitor of PARP1 at the sites of SSBs. AZD-9574 exhibits anti-cancer activities and can be used in studies about HRD+ breast cancer and advanced solid malignancies.

价 格：￥电议型 号：T9756产 地：中国大陆

TN13438-GeranyloxypsoralenCYPs,Cytochrome P450,8Geranyloxypsoralen,inhibit,8-Geranyloxypsoralen,Inhibitor,

8-Geranyloxypsoralen inhibits α2-secretase (BACE1) activity in non-competitive manner, with the IC(50) values <25.0 μM, it can induce vasorelaxation on rat arterial tissues. 8-Geranyloxypsoralen possesses nematicidal activities, the median lethal concentrations (LC(50)) is 188.3 mg/ L against B. xylophilus and is 117.5 mg/L against P. redivivus.

价 格：￥电议型 号：TN1343产 地：中国大陆

TQ0312SphingomyelinSphingomyelin

Sphingomyelin is a natural sphingolipid that existed in animal cell membranes. It implicates the regulation of transmembrane signaling.

价 格：￥电议型 号：TQ0312产 地：中国大陆

T8386Esomeprazole Magnesium trihydrateinhibit,K+-ATPase,Esomeprazole magnesium,antioxidant,Proton Pump,(S

Esomeprazole Magnesium trihydrate is a proton pump inhibitor indicated for the short-term treatment of gastroesophageal reflux disease in patients with a history of erosive esophagitis.Esomeprazole magnesium trihydrate acts as an exosome inhibitor by blocking the exosome release via the inhibition of V-H+-ATPases

价 格：￥电议型 号：T8386产 地：中国大陆

T9214ELOVL6-IN-1ELOVL6IN1,noncompetitive,orally,palmitoyl-CoA,potent,malonyl-CoA,ELOVL-6-IN-1,Inhibitor,s

ELOVL6-IN-1 is a potent, orally active and selective ELOVL6 inhibitor. ELOVL6-IN-1 dose-dependently inhibits mouse ELOVL6 activities, with an IC50 value of 0.350 μM. ELOVL6-IN-1 inhibits ELOVL6 in a noncompetitive manner for malonyl-CoA (Ki=994 nM) and palmitoyl-CoA[1].

价 格：￥电议型 号：T9214产 地：中国大陆

T8109d-Neomenthold Neomenthol,dNeomenthol

d-Neomenthol is a natural product.

价 格：￥电议型 号：T8109产 地：中国大陆

T8919Homo SildenafilInhibitor,Phosphodiesterase (PDE),Homo Sildenafil,inhibit

Homo Sildenafil is an analog of Sildenafil, It acts as a phosphodiesterase inhibitor.

价 格：￥电议型 号：T8919产 地：中国大陆

T7378BRD9539Histone Methyltransferase,chromatin,PRC2,BRD9539,G9a,senescent,BRD-9539,BRD 9539,inhibit,H3K9

BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 μM

价 格：￥电议型 号：T7378产 地：中国大陆

T61301Chromenone 1

Chromenone 1 is a potent potentiator of osteogenic bone morphogenetic protein (BMP). Chromenone 1 induces a pronounced, kinase-independent, negative TGFβ feedback that enhances nuclear BMP-Smad signaling outputs.

价 格：￥电议型 号：T61301产 地：中国大陆

T6832Fatostatin hydrobromideGolgi,ob/ob,inhibit,Fatostatin hydrobromide,prostate,SREBP-mediated,cancer,mi

Fatostatin ia an inhibitor of sterol regulatory element binding protein (SREBP). It impairs the activation of SREBP-1 and SREBP-2.

价 格：￥电议型 号：T6832产 地：中国大陆

T9825CORT-108297 EnantiomerCORT108297 Enantiomer,CORT 108297 Enantiomer

CORT-108297 Enantiomer is an enantiomer of CORT-108297 which is an antagonist of the Glucocorticoid Receptor.

价 格：￥电议型 号：T9825产 地：中国大陆