T6681STF-083010STF 083010,STF-083010,Inositol requiring enzyme 1,Inhibitor,inhibit,IRE1

STF-083010 is a selective inhibitor of the IRE1α endonuclease.

价 格：￥电议型 号：T6681产 地：中国大陆

T21302LUNC 569 hydrochlorideUNC 569 hydrochloride

UNC 569 hydrochloride is a reversible and ATP-competitive inhibitor of Mer with an IC50 of 2.9 nM and a Ki of 4.3 nM. UNC 569 hydrochloride inhibits Axl and Tyro3 with IC50s of 37 nM and 48 nM, respectively. UNC 569 hydrochloride can be used in studies about acute lymphoblastic leukemia and atypical teratoid/rhabdoid tumors.

价 格：￥电议型 号：T21302L产 地：中国大陆

TQ0317R1530antitumor,Inhibitor,Fibroblast growth factor receptor,mitosis,FGFR,angiogenesis,R1530,VEGFR,ant

R1530 is a multikinase inhibitor with antineoplastic and antiangiogenesis activities.

价 格：￥电议型 号：TQ0317产 地：中国大陆

TQ0282Avosentaninhibit,SPP 301,Inhibitor,Avosentan,SPP301,Endothelin Receptor

Avosentan (Ro 67-0565) is an effective and selective antagonist of the endothelin receptor (ETA receptor).

价 格：￥电议型 号：TQ0282产 地：中国大陆

T30544BMS-919373

BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.

价 格：￥电议型 号：T30544产 地：中国大陆

TP1304CompstatinComplement System,Inhibitor,Compstatin,inhibit

Compstatin, a cyclic tridecapeptide, which was originally discovered from phage-display libraries, is a highly potent and selective C3 inhibitor.

价 格：￥电议型 号：TP1304产 地：中国大陆

T7359CAY10471 RacemateCAY 10471,CAY10471,TM30089,Inhibitor,CAY-10471,TM 30089,TM-30089,CAY10471 Racemate,

CAY 10471 is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the human CRTH2/DP2, DP1, and TP receptors( Ki values of 0.6, 1200, and >10,000 nM,respectively)

价 格：￥电议型 号：T7359产 地：中国大陆

T30677LC15AlkOPP Tetrabutylamine salt(946615-44-7 Free base)

C15AlkOPP Tetrabutylamine salt is a “clickable” alkyne-modified analogs of the lipid substrates farnesyl diphosphate (FPP).

价 格：￥电议型 号：T30677L产 地：中国大陆

T9588JI130JI130,JI-130

JI130 is able to impair the ability of Hes1 to repress transcription. JI130 treatment significantly reduced tumor volume in a murine pancreatic tumor xenograft model.

价 格：￥电议型 号：T9588产 地：中国大陆

Fr213071,2,3,4-Tetrahydro-6-quinolinecarboxylic Acid

价 格：￥电议型 号：Fr21307产 地：中国大陆

T62530N-Arachidonyldopamine

N-Arachidonyldopamine is a potent and selective endogenous CB1 receptor agonist (Ki= 250 nM). N-Arachidonyldopamine is also a potent and selective TRPV1 agonist (EC50= ~ 50 nM).

价 格：￥电议型 号：T62530产 地：中国大陆

T6336AmonafideNafidimide；Quinamed；AS1413；NSC308847,AS1413；氨萘非特

Amonafide(AS1413) produces protein-associated DNA-strand breaks through a topoisomerase II-mediated reaction, but does not produce topoisomerase I-mediated DNA cleavage.

价 格：￥电议型 号：T6336产 地：中国大陆

T6331Allitinib tosylateAST-1306 TsOH；AST-6；Allitinib；AST-1306 (TsOH)；AST-1306；艾力替尼

AST-1306 is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of 0.5 nM and 3 nM, respectively.

价 格：￥电议型 号：T6331产 地：中国大陆

T6330LinperlisibPI3Kδ-IN-2

PI3Kδ-IN-2 is a potent and selective inhibitor of PI3Kδ

价 格：￥电议型 号：T6330产 地：中国大陆

T6309AZ960AZ 960

AZ 960 is an effective ATP competitive JAK2 inhibitor (IC50/Ki: <3 nM and0.45 nM).

价 格：￥电议型 号：T6309产 地：中国大陆

T6308StatticSTAT3 Inhibitor V

Stattic is a small molecule inhibitor of STAT3. It selectively inhibits STAT3 activation, dimerization, and nuclear translocation (IC50: 5.1 μM).

价 格：￥电议型 号：T6308产 地：中国大陆

T6307Lubiprostone芦比前列酮；鲁比前列酮；RU-0211；SPI-0211

Lubiprostone, an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.

价 格：￥电议型 号：T6307产 地：中国大陆

T6306ErteberelLY500307

LY500307 is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.

价 格：￥电议型 号：T6306产 地：中国大陆

T6305SNX2112SNX 2112；PF 04928473；SNX-2112

SNX-2112 is an orally active Hsp90 inhibitor, with a Kd of 16 nM.

价 格：￥电议型 号：T6305产 地：中国大陆

T6304AT7867

AT7867 is a potent ATP-competitive inhibitor of Akt1/2/3 and p70S6K/PKA with IC50 of 32 nM/17 nM/47 nM and 85 nM/20 nM, respectively; little activity outside the AGC kinase family.

价 格：￥电议型 号：T6304产 地：中国大陆