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T1613Hydralazine hydrochloride；盐酸肼屈嗪Hydralazine HCl|||Apresoline；Hydralazine HCl|||Apresoline|||盐酸肼屈嗪
Hydralazine hydrochloride (Apresoline) is the hydrochloride salt of hydralazine, a phthalazine derivative with antihypertensive and potential antineoplastic activities. Hydralazine alters intracellular calcium release and interferes with smooth muscle cell calcium influx, resulting in arterial vasodilatation. This agent also inhibits the phosphorylation of myosin protein and chelation of trace metals required for smooth muscle contraction, resulting in an increase in heart rate, stroke volume, a
价 格：￥电议型 号：T1613产 地：中国大陆
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T16129MPI_5a；化合物MPI_5aMPI_5a
MPI_5a is an effective and selective inhibitor of HDAC6 (IC50=36 nM). MPI_5a weakly inhibits other HDAC isoforms and it also inhibits acyl-tubulin accumulation in cells (IC50: 210 nM).
价 格：￥电议型 号：T16129产 地：中国大陆
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T16128MP-A08；化合物MP-A08MP-A08
MP-A08 is a highly selective ATP competitive inhibitor of sphingosine kinase (SPHK1) that targets both SphK1 and SphK2 (Ki: 6.9 ± 0.8 μM and 27 ± 3 μM, respectively).
价 格：￥电议型 号：T16128产 地：中国大陆
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T16127Moricizine；莫雷西嗪Moracizine；Moracizine|||莫雷西嗪
Moricizine is an antiarrhythmia agent which is used primarily for ventricular rhythm disturbances.
价 格：￥电议型 号：T16127产 地：中国大陆
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T16126Monepantel；化合物 MonepantelAAD1566|||PPL-1；AAD1566|||PPL-1
Monepantel (AAD1566) is an organic anthelmintic and nicotinic acetylcholine receptor antagonist from roundworms and esophagostomies that is widely used for de-worming in agriculture and livestock.
价 格：￥电议型 号：T16126产 地：中国大陆
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T16125MMV390048；化合物MMV390048MMV390048
MMV390048 is an antimalarial agent and is a representative of a new chemical class of Plasmodium PI4K inhibitor (Kdapp=0.3 μM). MMV390048 binds to the ATP binding site of Plasmodium PI4K and does not bind to other P. falciparum and human kinases apart from human PIP4K2C, thus alleviating potential kinase-mediated safety concerns.
价 格：￥电议型 号：T16125产 地：中国大陆
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T16124MMP13-IN-3；化合物MMP13-IN-3MMP13-IN-3
MMP13-IN-3 is >1000 selective over other MMPs. MMP13-IN-3 is an effective, selective, and orally active MMP-13 inhibitor (IC50=1 nM) for the potential treatment of osteoarthritis.
价 格：￥电议型 号：T16124产 地：中国大陆
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T16123MMG-11；化合物 T16123MMG-11
MMG-11 inhibits both TLR2/1 and TLR2/6 signaling (IC50s: 1.7 μM for Pam3CSK4-induced hTLR2/1 and 5.7 μM for Pam2CSK4-induced hTLR2/6 responses). MMG-11 is an effective and selective human TLR2 antagonist with low cytotoxicity.
价 格：￥电议型 号：T16123产 地：中国大陆
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T16122MMAF sodium；化合物 T16122Monomethylauristatin F sodium；Monomethylauristatin F sodium
MMAF sodium is widely used as a cytotoxic component of antibody-drug conjugates (ADCs) such as Vorsetuzumab mafodotin and SGN-CD19A. MMAF sodium is an effective tubulin polymerization inhibitor and is used as an antitumor agent.
价 格：￥电议型 号：T16122产 地：中国大陆
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T16121MMAF Hydrochloride；化合物 T16121Monomethylauristatin F Hydrochloride；Monomethylauristatin F Hydrochlori
MMAF Hydrochloride is widely used as a cytotoxic component of antibody-drug conjugates (ADCs) such as Vorsetuzumab mafodotin and SGN-CD19A. MMAF Hydrochloride is an effective tubulin polymerization inhibitor and is used as an antitumor compound.
价 格：￥电议型 号：T16121产 地：中国大陆
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T16120MLT-748；化合物 T16120MLT-748
MLT-748 is an effective, selective, and allosteric MALT1 inhibitor. It binds MALT1 in the allosteric Trp580 pocket (IC50: 5 nM).
价 格：￥电议型 号：T16120产 地：中国大陆
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T1612Neostigmine methyl sulfate；甲硫酸新斯的明Normastigmin|||Hodostin|||Syntostigmin；Normastigmin|||甲基硫酸新斯的明|||甲
Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase, can not cross the blood-brain barrier, used in the treatment of myasthenia gravis.
价 格：￥电议型 号：T1612产 地：中国大陆
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T16119MLT-747；化合物 T16119MLT-747
MLT-747 is an effective and allosteric inhibitor of MALT1. It binds MALT1 in the allosteric Trp580 pocket (IC50: 14 nM).
价 格：￥电议型 号：T16119产 地：中国大陆
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T16118MLS0315771；化合物MLS0315771MLS0315771
MLS0315771 is an effective and biologically active competitive phosphomannose isomerase (MPI) inhibitor (IC50: ~1 μM and a Ki: 1.4 μM).
价 格：￥电议型 号：T16118产 地：中国大陆
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T16117Pevonedistat hydrochloride化合物 T16117MLN4924 hydrochloride
Pevonedistat hydrochloride is an effective and selective inhibitor of NEDD8-activating enzyme (IC50: 4.7 nM).
价 格：￥电议型 号：T16117产 地：中国大陆
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T16116MLN-4760；化合物MLN-4760MLN-4760
MLN-4760 is an angiotensin-converting (ACE2) inhibitor(human ACE2;IC50=0.44 nM). It also has excellent selectivity (>5000-fold) versus related enzymes including human testicular ACE (IC50, >100 μM) and bovine carboxypeptidase A (CPDA; IC50, 27 μM).
价 格：￥电议型 号：T16116产 地：中国大陆
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T16115MLi-2；化合物MLi-2MLi-2
MLi-2 is a structurally novel, highly potent, and selective LRRK2 kinase inhibitor with central nervous system activity. MLi-2 exhibits exceptional potency in a purified LRRK2 kinase assay in vitro (IC50 = 0.76 nM), a cellular assay monitoring dephosphorylation of LRRK2 pSer935 LRRK2 (IC50 = 1.4 nM), and a radioligand competition binding assay (IC50 = 3.4 nM).
价 格：￥电议型 号：T16115产 地：中国大陆
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T16114Pavinetant；化合物 PavinetantMLE-4901|||AZD4901|||AZD2624；MLE-4901|||AZD4901|||AZD2624
Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.
价 格：￥电议型 号：T16114产 地：中国大陆
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T16113ML753286；化合物 T16113ML753286
ML753286 has high permeability and low to medium clearance in rodent and human liver S9 fractions. ML753286 is an orally active and selective inhibitor of BCRP (IC50: 0.6 μM). It is also stable in plasma across species.
价 格：￥电议型 号：T16113产 地：中国大陆
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T16112ML67-33化合物 T16112ML-67-33|||ML6733|||ML67 33
ML67-33 rapidly and reversibly affects K2P2.1 (TREK-1) (EC50s: 36.3 μM and 9.7 μM in cell-free and HEK293 cells, respectively). ML67-33 is a selective activator of temperature- and mechano-sensitive K2P channels.
价 格：￥电议型 号：T16112产 地：中国大陆
