T8796CAN508inhibit,CAN 508,ATP-competitive,Cyclin dependent kinase,esophageal,cells,CDK,CAN508,Inhibitor,

CAN508 is a potent, ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 μM. It is also a competitive inhibitor of Cdk2-cyclin E with respect to ATP, with Ki and IC50 values of 13.3 and 20 μM, respectively.CAN508 exhibits a 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes. Antitumor activity.

价 格：￥电议型 号：T8796产 地：中国大陆

TQ0283RS102895CC chemokine receptor,CCR,Inhibitor,RS102895,inhibit,RS-102895,RS 102895

RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.

价 格：￥电议型 号：TQ0283产 地：中国大陆

T9041AES-350Histone deacetylases,AES 350,MV4-11,AES-350,Apoptosis,acute myeloid leukemia,AML,Inhibitor,in

AES-350 is a potent and orally active HDAC6 inhibitor(IC50 and a Ki of 0.0244 μM and 0.035 μM, respectively). It is also against HDAC-3, -8, and -11 in an enzymatic activity assay with IC50 values of 0.187 μM, 0.245 μM, and >1μM, respectively. AES-350 triggers apoptosis in AML cells through HDAC inhibition and can be used for acute myeloid leukemia (AML) research.

价 格：￥电议型 号：T9041产 地：中国大陆

T61518TAK-653

TAK-653, an AMPA receptor potentiator with minimal agonistic activity, produces an antidepressant-like effect with a favorable safety profile in rats.

价 格：￥电议型 号：T61518产 地：中国大陆

T6908NSC 228155Epidermal growth factor receptor,Histone Acetyltransferase,EGFR,HER1,HATs,inhibit,Inhibito

NSC228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and modulate EGFR tyrosine phosphorylation.

价 格：￥电议型 号：T6908产 地：中国大陆

T14526Bemesetron

Bemesetron is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.

价 格：￥电议型 号：T14526产 地：中国大陆

T7815LAOD9604 acetate(221231-10-3 free base)AOD9604 acetate(221231103 free base),AOD-9604 acetate(221231-1

AOD9604 acetate is a potential anti-obesity peptide based on the human growth hormone.

价 格：￥电议型 号：T7815L产 地：中国大陆

Fr14055Compound Fr14055Compound Fr14055

价 格：￥电议型 号：Fr14055产 地：中国大陆

T75283,7-dimethylocta-2,6-dienyl 5,9,13-trimethyltetradeca-4,8,12-enoate3,7dimethylocta2,6dienyl 5,9,13tr

3,7-dimethylocta-2,6-dienyl 5,9,13-trimethyltetradeca-4,8,12-enoate is a chemical compound

价 格：￥电议型 号：T7528产 地：中国大陆

T7596FirocoxibLPS,COX-2,fever,ML1785713,Cyclooxygenase,COX,inhibit,Firocoxib,Inhibitor,anti-inflammatory,

Firocoxib is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 μM), with anti-inflammatory for use in dogs and horses.

价 格：￥电议型 号：T7596产 地：中国大陆

T60057WAY-388657WAY 388657,WAY388657

WAY-388657 is a Notum Pectinacetylesterase inhibitor with IC50 < 0.025 μM.

价 格：￥电议型 号：T60057产 地：中国大陆

TP1545L1FFAGLDD amine saltFFAGLDD amine salt

FFAGLDD amine salt is MMP9 selective cleavage peptides, which used for cytosolic delivery of Doxorubi-cin (DOX) and achieve temporally and spatially controlled slow drug delivery and release.

价 格：￥电议型 号：TP1545L1产 地：中国大陆

T40652Meclizine

Meclizine (Meclozine) shows antihistamine activity and reversibly inhibits the interaction of histamine at the H1 receptors . Meclizine is a member of the piperazine class of H1 antagonists. Meclizine is an effective anti-motion sickness agent. Meclizine crosses the blood–brain barrier. Meclizine is an agonist ligand for mouse constitutive androstane receptor (CAR) and an inverse agonist for Human CAR. Meclizine can be used for the research of polyQ toxicity disorders, such as Huntington´s

价 格：￥电议型 号：T40652产 地：中国大陆

T6507Gabapentin hydrochlorideInhibitor,Gabapentin hydrochloride,Gabapentin,Calcium Channel,Ca channels,in

Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.

价 格：￥电议型 号：T6507产 地：中国大陆

T38163ML-148ML-148,ML 148,selective,Inhibitor,prostaglandin-signaling,15-PGDH,15-Hydroxyprostaglandin dehy

ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM). ML-148 can be used to profile across a panel of related dehydrogenase or reductase enzymes and in studies about prostaglandin-signaling pathways.

价 格：￥电议型 号：T38163产 地：中国大陆

T6648Rotundine5-hydroxytryptamine Receptor,Inhibitor,Dopamine Receptor,Rotundine,5-HT Receptor,inhibit,Se

Rotundine (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.

价 格：￥电议型 号：T6648产 地：中国大陆

T60199NCRW0005-F05NCRW0005F05

NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 value of 0.21 μM. NCRW0005-F05 can be used to research diabetes, obesity and Parkinson´s disease [1].

价 格：￥电议型 号：T60199产 地：中国大陆

T17239VU0155069

VU0155069 strongly inhibits the invasive migration of several cancer cell lines in transwell assays. VU0155069 is a selective phospholipase D1 inhibitor (IC50: 46 nM in vitro).

价 格：￥电议型 号：T17239产 地：中国大陆

T60072ZL0590non-KAc binding site,ZL0590,ZL-0590,BRD4 BD1,Inhibitor,acute airway inflammation,inhibit,Epige

ZL0590 is an effective and selective inhibitor of BD1-BRD4 (IC50 = 90 nM) with anti-inflammatory activities.

价 格：￥电议型 号：T60072产 地：中国大陆

T22900L-701252

L-701252 is a potent antagonist of glycine site NMDA receptor with an IC50 of 420 nM. L-701252 provides a small degree of neuroprotection in global cerebral ischaemia.

价 格：￥电议型 号：T22900产 地：中国大陆