TN1121EvocarpineEvocarpine,Ca2+,HL-60,inhibit,antimycobacterial,Inhibitor,leukaemia,Bacterial,Apoptosis,In

Evocarpine shows antimycobacterial, and vasorelaxant effects, it can inhibit Ca2+ influx through voltage-dependent calcium channels.

价 格：￥电议型 号：TN1121产 地：中国大陆

TQ0062NastorazepideZ360,CCK Receptor,Cholecystokinin Receptor,Inhibitor,Z 360,Nastorazepide,inhibit

Nastorazepide is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity.

价 格：￥电议型 号：TQ0062产 地：中国大陆

T9609GRK5-IN-2metabolic,bicyclic,insulin,kinase,inhibit,Inhibitor,disease,pyridine-based,GRK5 IN 2,GRK-5-

GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor. It regulates the expression and/or release of insulin and is useful for the metabolic disease research.

价 格：￥电议型 号：T9609产 地：中国大陆

T60123Chimmitecan

Chimmitecan is a potent inhibitor of topoisomerase I and displays outstanding activity in vitro and in vivo.

价 格：￥电议型 号：T60123产 地：中国大陆

TQ0029ASTX660Inhibitor,inhibit,ASTX-660,ASTX660,IAP,ASTX 660

ASTX660 is an orally bioavailable dual antagonist of cIAP and XIAP.

价 格：￥电议型 号：TQ0029产 地：中国大陆

T7604ValrubicinInhibitor,AD 32,AD32,Valrubicin,inhibit,PKC,Antibiotic,Protein kinase C

Valrubicin (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and has antitumor and anti-inflammatory activity.

价 格：￥电议型 号：T7604产 地：中国大陆

T60147BAY-091BAY091

BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.

价 格：￥电议型 号：T60147产 地：中国大陆

T20600KaolinKaolin

Kaolin is a clay dominated by minerals of the kaolinite family. Kaolin increased the sensitivity of this method for monitoring hemophilia therapy.

价 格：￥电议型 号：T20600产 地：中国大陆

T60202MMRi62

MMRi62, a ferroptosis inducer targeting MDM2-MDM4 (negative regulators of tumor suppressor p53). MMRi62 shows a P53-independent pro-apoptotic activity against pancreatic ductal adenocarcinoma (PDAC) cells and induce autophagy. MMRi62 inducesferroptosis, resulting in a increase of reactive oxygen and lysosomal degradation of ferritin heavy chain (FTH1). MMRi62 also leads to proteasomal degradation of mutant p53, also inhibits orthotopic xenograft PDAC mouse model in vivo with high frequency mutat

价 格：￥电议型 号：T60202产 地：中国大陆

T7409360A360A,Telomerase,inhibit,Inhibitor,G-quadruplex

360A is a stabilizing G-Quadruplex ligand, and also inhibits telomerase activity for telomerase in TRAP-G4 assay(IC50 : 300 nM).

价 格：￥电议型 号：T7409产 地：中国大陆

TJS0328Nordalberginpromyelocytic,Inhibitor,coumarin,HL-60,cells,leukemia,differentiation,Nordalbergin,inhib

价 格：￥电议型 号：TJS0328产 地：中国大陆

T6068MK-5108MK 5108,VX689,Aurora Kinase,VX 689,inhibit,Autophagy,MK-5108,Inhibitor

MK-5108 is a highly potent and specific Aurora-A kinase inhibitor with an IC50 value of 0.064 nM.

价 格：￥电议型 号：T6068产 地：中国大陆

T5362Y06036inhibit,Epigenetic Reader Domain,Inhibitor,Y-06036,Y 06036,Y06036

Y06036, a potent and selective BET inhibitor, can bind to the BRD4(1) bromodomain (Kd: 82 nM).

价 格：￥电议型 号：T5362产 地：中国大陆

T6588Mitoxantroneleukaemia,NSC301739,PKC,MCF-7,NSC 301739,lymphocytes,Topoisomerase,Mitoxantrone,HL60 cel

Mitoxantrone is an anthracenedione antibiotic with antineoplastic activity. Mitoxantrone intercalates into and crosslinks DNA, thereby disrupting DNA and RNA replication. This agent also binds to topoisomerase II, resulting in DNA strand breaks and inhibition of DNA repair. Mitoxantrone is less cardiotoxic compared to doxorubicin.

价 格：￥电议型 号：T6588产 地：中国大陆

T60052BMS-905BMS905,BMS 905

BMS-905 is a potent dual inhibitors of TLR7 and TLR8 with good selectivity against TLR9 and other family members. BMS-905 can be used in studies about the treatment of diseases such as psoriasis, arthritis, and lupus.

价 格：￥电议型 号：T60052产 地：中国大陆

T10874CP-060CP060,CP 060

CP-?060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.

价 格：￥电议型 号：T10874产 地：中国大陆

TP1760LAMARA peptide acetate(163560-19-8 free base)AMARA peptide acetate(163560 19 8 free base),AMARA pep

AMARA peptide acetate is a substrate for SIK and AMPK.AMARA peptide is a minimal substrate of several members of the protein kinases family. It consists of the phosphorylation site for AMP-activated Protein Kinase (AMPK).

价 格：￥电议型 号：TP1760L产 地：中国大陆

T60128N,N-Didesethyl Sunitinib HydrochlorideN,NDidesethylSunitinibHydrochloride

N,N-Didesethyl Sunitinib Hydrochloride is a potent AMPK inhibitor with IC50 of 393 nM and 141 nM for AMPKα1 and AMPK2,respectively.

价 格：￥电议型 号：T60128产 地：中国大陆

T36010p38 MAPK Inhibitorp-38 MAPK Inhibitor,p38 MAPK Inhibitor

p38 MAPK inhibitor is a potent inhibitor of p38 MAP kinase (IC50 = 35 nM). It inhibits senescence induced by the oncogene RAS.

价 格：￥电议型 号：T36010产 地：中国大陆

T7353RSV604virus,Respiratory syncytial virus,A 60444,respiratory,protein,inhibit,RSV,syncytial,A-60444,In

RSV-604 is an inhibitor of respiratory syncytial virus (RSV) that binds to RSV nucleoprotein (Kd = 1.31 μM)

价 格：￥电议型 号：T7353产 地：中国大陆