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  • T78934c-Met-IN-18；化合物 c-Met-IN-18c-Met-IN-18

    C-Met-IN-18, an ATP-competitive type-III inhibitor, targets both wild-type (WT) and D1228V mutant c-MET with IC50 values of 0.013 ?M and 0.20 ?M, respectively. It is utilized in research pertaining to c-MET-driven cancers [1].

    价 格：￥电议型 号：T78934产 地：中国大陆

  • T78932hDHODH-IN-12；化合物 hDHODH-IN-12hDHODH-IN-12

    hDHODH-IN-12 is a potent inhibitor of dihydroorotate dehydrogenase (DHODH), exhibiting an inhibitory concentration (IC50) of 0.421 μM. As the rate-limiting enzyme in the de novo synthesis of pyrimidines, critical for DNA/RNA synthesis, DHODH is localized within the inner membrane of human mitochondria. hDHODH-IN-12 is applicable in lung cancer research [1].

    价 格：￥电议型 号：T78932产 地：中国大陆

  • T78930T3SS-IN-1；化合物 T3SS-IN-1T3SS-IN-1

    T3SS-IN-1 (compound B9) is a potent type III secretion system (T3SS) inhibitor that also suppresses hpa1 promoter activity and harpin protein expression, without impacting bacterial growth [1].

    价 格：￥电议型 号：T78930产 地：中国大陆

  • T78921FAP-IN-1；化合物 FAP-IN-1FAP-IN-1

    FAP-IN-1 is a fibroblast activation protein (FAP) inhibitor, exhibiting an IC50 of 3.3 nM, and is utilized for cancer research [1].

    价 格：￥电议型 号：T78921产 地：中国大陆

  • T78913AKT-IN-18；化合物 AKT-IN-18AKT-IN-18

    AKT-IN-18, an Akt inhibitor, demonstrates an IC50 value of 69.45 μM in A549 cells, effectively impeding Akt activity. It promotes apoptosis and is suitable for use in non-small cell lung cancer research [1].

    价 格：￥电议型 号：T78913产 地：中国大陆

  • T78899Laccase-IN-1；化合物 Laccase-IN-1Laccase-IN-1

    Laccase-IN-1 (compound 4b) is an orally active laccase inhibitor, demonstrating an IC50 of 11.3 μM. It exhibits both protective and curative effects against B. dothidea infections in apple fruits. The compound increases cell membrane permeability, disrupts mycelial surface morphology, alters cell ultrastructure, and decreases the ergosterol and exopolysaccharide levels in B. dothidea [1].

    价 格：￥电议型 号：T78899产 地：中国大陆

  • T78889Lysyl hydroxylase 2-IN-1；化合物 Lysyl hydroxylase 2-IN-1Lysyl hydroxylase 2-IN-1

    "Lysyl Hydroxylase 2-IN-1 (compound 12) is a selective inhibitor of lysyl hydroxylase 2 (LH2) with an IC50 of approximately 300 nM and demonstrates specificity for LH2 over LH1 and LH3 [1]."

    价 格：￥电议型 号：T78889产 地：中国大陆

  • T78882NF-κB-IN-12；化合物 NF-κB-IN-12NF-κB-IN-12

    NF-κB-IN-12 (compound 3h) serves as a potent inhibitor of NF-κB, exhibiting an IC50 value of 1.02 μM. It is applicable for research in acute lung injury [1].

    价 格：￥电议型 号：T78882产 地：中国大陆

  • T7888Enpp-1-IN-1；化合物Enpp-1-IN-1Enpp-1-IN-1

    Enpp-1-IN-1 is an inhibitor of Ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp-1)

    价 格：￥电议型 号：T7888产 地：中国大陆

  • T78868TWIK-1/TREK-1-IN-1；化合物 TWIK-1/TREK-1-IN-1TWIK-1/TREK-1-IN-1

    Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers and TWIK-1/TREK-1 heterodimers, both significant for its role as an antidepressant target. Furthermore, TWIK-1/TREK-1-IN-3, a related compound, selectively inhibits these channels with IC50 values of 9.36 μM for TREK-1 homodimers and 14.6 μM for TWIK-1/TREK-1 heterodimers, demonstrating antidepressant-like effects [1].

    价 格：￥电议型 号：T78868产 地：中国大陆

  • T78858cGAS-IN-1；化合物 cGAS-IN-1cGAS-IN-1

    cGAS-IN-1 (compound C20), a flavonoid that acts as a Cyclic GMP-AMP Synthase (cGAS) inhibitor, demonstrates IC50 values of 2.28 μM for human cGAS and 1.44 μM for mouse cGAS. By inhibiting the abnormal activation of cGAS linked to numerous immune-mediated inflammatory diseases, cGAS-IN-1 possesses potential anti-inflammatory properties [1].

    价 格：￥电议型 号：T78858产 地：中国大陆

  • T78845FGFR1/VEGFR2-IN-1；化合物 FGFR1/VEGFR2-IN-1FGFR1/VEGFR2-IN-1

    FGFR1/VEGFR2-IN-1 (compound 2b) is an inhibitor of both FGFR1 and VEGFR2, applicable in cancer research [1].

    价 格：￥电议型 号：T78845产 地：中国大陆

  • T78843MET/PDGFRA-IN-1；化合物 MET/PDGFRA-IN-1MET/PDGFRA-IN-1

    MET/PDGFRA-IN-1 (compound 8c) serves as an inhibitor of MET and PDGFRA proteins, displaying an IC50 of 36 μM against MET. It impedes MET phosphorylation, thereby promoting apoptosis, and curtails the proliferation of various MET-positive cell lines, with IC50 values of 15.3 μM for AsPc-1, 19.0 μM for EBC-1, 22.0 μM for MKN-45, 25.6 μM for Mia-Paca-2, 21.0 μM for HT-29, and 31.5 μM for K562 [1].

    价 格：￥电议型 号：T78843产 地：中国大陆

  • T78839HDAC6-IN-19；化合物 HDAC6-IN-19HDAC6-IN-19

    HDAC6-IN-19 (Compound 14g), an HDAC6 inhibitor with an IC50 of 2.68 nM, additionally inhibits HDAC1, HDAC2, and HDAC3, with IC50 values of 61.6 nM, 98.7 nM, and 103 nM, respectively. This compound effectively suppresses the proliferation of various cancer cell lines, such as leukemia, colon cancer, melanoma, and breast cancer [1].

    价 格：￥电议型 号：T78839产 地：中国大陆

  • T78838Akt/NF-κB/MAPK-IN-1；化合物 Akt/NF-κB/MAPK-IN-1Akt/NF-κB/MAPK-IN-1

    Akt/NF-κB/MAPK-IN-1 (compound 2m) serves as a potent, orally active inhibitor targeting NO with an IC50 of 7.70 μM and demonstrates low toxicity. This compound exerts anti-inflammatory effects by impeding the Akt/NF-κB and MAPK signaling pathways [1].

    价 格：￥电议型 号：T78838产 地：中国大陆

  • T78835Phosphatase-IN-1；Phosphatase 抑制剂 1Phosphatase-IN-1

    Phosphatase-IN-1 (compound II-8), a propranolol derivative, acts as an inhibitor of phosphatidate phosphatase (Pah). It binds to MoPah1 with an affinity constant of 19.8 μM, demonstrating growth inhibition of plant pathogens and anti-fungal properties. Notably, Phosphatase-IN-1 exhibits no toxicity towards rice seedlings and wheat heads [1].

    价 格：￥电议型 号：T78835产 地：中国大陆

  • T78829JNK2-IN-1；化合物 JNK2-IN-1JNK2-IN-1

    JNK2-IN-1 (Compound J27), a selective JNK2 inhibitor with a dissociation constant (Kd) of 79.2 ?M, exhibits anti-inflammatory effects by attenuating TNF-α and IL-6 secretion via inhibition of the NF-κB/MAPK pathway. It effectively mitigates symptoms associated with LPS-induced acute lung injury (ALI) and sepsis [1].

    价 格：￥电议型 号：T78829产 地：中国大陆

  • T78828AChE/BChE-IN-15；化合物 AChE/BChE-IN-15AChE/BChE-IN-15

    AChE/BChE-IN-15 (Compound 6d) serves as an inhibitor for both acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), presenting inhibition constants (IC50) of 20 nM for AChE and 220 nM for BChE. It interacts with the catalytic anionic site (CAS) and the peripheral anionic site (PAS) within the enzymes´ active sites. AChE/BChE-IN-15 is applicable in Alzheimer’s disease research [1].

    价 格：￥电议型 号：T78828产 地：中国大陆

  • T78823Quorum Sensing-IN-3；Quorum Sensing抑制剂1QS-IN-1；QS-IN-1

    Quorum Sensing-IN-3 (QS-IN-1) is a compound with inhibitory effects on bacterial community sensing, which inhibits the exchange of information between bacteria and inhibits biofilm formation.

    价 格：￥电议型 号：T78823产 地：中国大陆

  • T78813CDK2/Bcl2-IN-1；化合物 CDK2/Bcl2-IN-1CDK2/Bcl2-IN-1

    CDK2/Bcl2-IN-1 (compound 1) is a saponin-based inhibitor of CDK-2 (IC50=117.6 nM) that exhibits potent cytotoxic effects on cancer cells. Additionally, it inhibits Bcl-2 and promotes apoptosis in A549 lung cancer cells [1].

    价 格：￥电议型 号：T78813产 地：中国大陆

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