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T76960Verpasep caltespen；化合物 Verpasep caltespenVerpasep caltespen
Verpasep caltespen (HspE7), a recombinant fusion protein, originates from the Mycobacterium bovis Calmette-Guérin heat shock protein 65 (Hsp65) and is covalently bonded at its C-terminal end to the E7 protein of HPV16. This compound has applications in researching both precancerous and cancerous lesions linked to the human papillomavirus (HPV) [1] [2].
价 格：￥电议型 号：T76960产 地：中国大陆
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T76156Sphingomyelin phosphodiesterase；化合物 Sphingomyelin phosphodiesteraseSphingomyelin phosphodiesterase
Sphingomyelin phosphodiesterase, a hydrolase, plays a crucial role in sphingomyelin metabolism by catalyzing the conversion of sphingomyelin into phosphocholine and ceramide. Furthermore, it is instrumental in cellular differentiation, immune and inflammatory responses, as well as intracellular cholesterol trafficking and metabolism [1] [2].
价 格：￥电议型 号：T76156产 地：中国大陆
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T73708Sp-cAMPS triethylamine；化合物 Sp-cAMPS triethylamineSp-cAMPS triethylamine
Sp-cAMPS triethylamine, a cAMP analog, serves as a potent activator of cAMP-dependent PKA I and II and acts as a competitive inhibitor of phosphodiesterase (PDE3A) with a K i of 47.6 ?M. Additionally, it binds the PDE10 GAF domain with an EC 50 of 40 μM [1] [2] [3].
价 格：￥电议型 号：T73708产 地：中国大陆
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T72138Mitochondrial respiration-IN-2；化合物 Mitochondrial respiration-IN-2Mitochondrial respiration-IN-2
Mitochondrial respiration-IN-2, a fluorine derivative of Virginiamycin M1, inhibits the mitochondrial translation of glioblastoma stem cells [1].
价 格：￥电议型 号：T72138产 地：中国大陆
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T72137Mitochondrial respiration-IN-3；化合物 Mitochondrial respiration-IN-3Mitochondrial respiration-IN-3
Mitochondrial respiration-IN-3, a fluorine derivative of Dalfopristin, possesses cell membrane permeability and exhibits the capability to inhibit mitochondrial translation in glioblastoma stem cells. This compound is utilized in cancer research [1].
价 格：￥电议型 号：T72137产 地：中国大陆
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T71664Mespirenone；美螺利酮Mespirenone
Mespirenone is a spironolactone derivative and aldosterone antagonist with diuretic effects.
价 格：￥电议型 号：T71664产 地：中国大陆
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T71130Spectramide；化合物 SpectramideSpectramide
Spectramide is a dopamine D-2 receptor antagonist.
价 格：￥电议型 号：T71130产 地：中国大陆
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T70814Alnespirone；化合物 AlnespironeAlnespirone
Alnespirone, also known as S-20499, is a selective 5-HT1A receptor full agonist of the azapirone chemical class. It has both antidepressant and anxiolytic effects.
价 格：￥电议型 号：T70814产 地：中国大陆
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T70666Alnespirone hydrochloride；化合物 Alnespirone hydrochlorideAlnespirone hydrochloride
Alnespirone hydrochloride is a selective 5-HT1A receptor full agonist of the azapirone chemical class. It has both antidepressant and anxiolytic effects.
价 格：￥电议型 号：T70666产 地：中国大陆
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T69712Icapamespib HCl；化合物 Icapamespib HClIcapamespib HCl
Icapamespib, also known as PU-HZ 151, is a heat shock protein 90 (HSP90) inhibitor. PU-HZ151 showed EC50 of 5 nM in the FP assay as compared to 11 nM for PU-H71 and a logD of 2.37 as compared to 1.21 for PU-H71. PU-HZ151 and radiolabeled PU-HZ151 showed selectivity for epichaperomes over the individual chaperome members. Icapamespib demonstrated the ability to productively engage the target in cells, mice, and humans.
价 格：￥电议型 号：T69712产 地：中国大陆
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T6960LPU-H71 HCl；PU-H71盐酸盐PU-H71 HCl(873436-91-0 Free base)|||Zelavespib HCl；PU-H71 HCl(873436-91-0 Free b
PU-H71 HCl (Zelavespib HCl) is a novel Hsp90 inhibitor, a novel purine-based analog, and a radiosensitizer that may be a promising agent for CIRT. PU-H71 HCL shows antitumor activity in many preclinical models of malignancy. PU-H71 HCL has an inhibitory effect on the protein expression levels of Rad51 and Ku70, which may be associated with the double chain break repair in the homologous recombination pathway and non-homologous end-joining pathway.
价 格：￥电议型 号：T6960L产 地：中国大陆
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T68765Spirorenone；化合物 SpirorenoneSpirorenone
Spirorenone is an androstadienone derivative as a highly effective aldosterone antagonist. Spirorenone is 8.6 times as potent as spironolactone, but showed a lower affinity for the mineralocorticoid receptors. In phase I clinical trials Spirorenone was absorbed with a half-life of 20-30 min, achieving maximum concentrations of about 100 ng/ml (10 mg) and 260 ng/ml (40 mg) after 1-2 h. Disposition of the parent drug was biphasic with half-lives of 50-60 min (distribution) and 5-6 h (elimination).
价 格：￥电议型 号：T68765产 地：中国大陆
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T68760Luminespib mesylate；化合物 Luminespib mesylateLuminespib mesylate
Luminespib, also known as AUY-922, NVP-AUY922, VER52296, is a derivative of 4,5-diarylisoxazole and a third-generation heat shock protein 90 (Hsp90) inhibitor with potential antineoplastic activity. Hsp90 inhibitor AUY922 has been shown to bind with high affinity to and inhibit Hsp90, resulting in the proteasomal degradation of oncogenic client proteins; the inhibition of cell proliferation; and the elevation of heat shock protein 72 (Hsp72) in a wide range of human tumor cell lines.
价 格：￥电议型 号：T68760产 地：中国大陆
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T6532Hesperadin；化合物HesperadinHesperadin
Hesperadin(IC50=250 nM) effectively inhibits Aurora B. It potently reduces the activity of AMPK, MAPKAP-K1, MKK1, Lck, CHK1 and PHK, but it could not inhibit MKK1 activity in vivo.
价 格：￥电议型 号：T6532产 地：中国大陆
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T64055SPOP-IN-6b dihydrochloride；化合物 SPOP-IN-6b dihydrochlorideSPOP-IN-6b dihydrochloride
SPOP-IN-6b dihydrochloride is a potent inhibitor of spotted POZ protein (SPOP) (IC50: 3.58 μM).
价 格：￥电议型 号：T64055产 地：中国大陆
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T63905Hesperadin hydrochloride；化合物 Hesperadin hydrochlorideHesperadin hydrochloride
Hesperadin hydrochloride is an ATP-competitive indolone inhibitor of Aurora A and B, with an IC50 value of 250 nM for Aurora B.
价 格：￥电议型 号：T63905产 地：中国大陆
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T63425Spirapril hydrochloride；化合物 Spirapril hydrochlorideSpirapril hydrochloride
Spirapril (SCH 33844) hydrochloride is a potent inhibitor of angiotensin-converting enzyme (ACE) and is an orally active prodrug of spiripril. Spirapril hydrochloride can be used to study hypertension and congestive heart failure.
价 格：￥电议型 号：T63425产 地：中国大陆
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T6297Alvespimycin hydrochloride；阿螺旋霉素盐酸盐BMS 826476|||NSC 707545|||KOS-1022|||17-DMAG hydrochloride|||Alve
Alvespimycin hydrochloride (BMS 826476) is a potent HSP90 inhibitor with IC50 of 62 nM. Phase 2.
价 格：￥电议型 号：T6297产 地：中国大陆
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T6290Tanespimycin；坦螺旋霉素17-AAG|||CP 127374|||NSC 330507|||KOS 953；坦螺旋霉素|||17-AAG|||CP 127374|||NSC 330507|
Tanespimycin (KOS 953) (17-AAG) is an inhibitor of Hsp90 that selectively inhibits BT474 tumor cell Hsp90 (IC50: 5 nM).
价 格：￥电议型 号：T6290产 地：中国大陆
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T6284Onalespib；化合物OnalespibAT13387|||Onalespib (AT13387)；AT13387|||Onalespib (AT13387)
Onalespib (AT13387) is a synthetic, orally bioavailable, small-molecule inhibitor of heat shock protein 90 (Hsp90) with potential antineoplastic activity. Onalespib selectively binds to Hsp90, thereby inhibiting its chaperone function and promoting the degradation of oncogenic signaling proteins involved in tumor cell proliferation and survival. Hsp90, a chaperone protein upregulated in a variety of tumor cells, regulates the folding, stability and degradation of many oncogenic signaling protein
价 格：￥电议型 号：T6284产 地：中国大陆
